| Compound name | Brutto | MW | CAS | PubChem CID | Action | Reference | Reference |
|---|---|---|---|---|---|---|---|
| Sirolimus | C51H79NO13 | 914.20 | 53123-88-9 | 5284616 | p70S6K, mTOR | Powell D.J. (2003) Mol. Cell Biol. 23 7794 | Braun W. (1995) FASEB J. 9 63 |
| Kinase | % Activity Remaining | Standard Deviation |
|---|---|---|
| AMPK | 87 | 2 |
| Aurora B | 86 | 5 |
| Aurora C | 97 | 5 |
| BRSK2 | 90 | 4 |
| CAMK1 | 97 | 0 |
| CAMKK alpha | 80 | 8 |
| CAMKK beta | 82 | 1 |
| CDK2-Cyclin A | 92 | 3 |
| CHK1 | 97 | 6 |
| CHK2 | 92 | 2 |
| CK1 delta | 88 | 1 |
| CK2 | 92 | 9 |
| CSK | 83 | 1 |
| DYRK1A | 91 | 1 |
| DYRK2 | 83 | 8 |
| DYRK3 | 87 | 1 |
| EF2K | 94 | 0 |
| ERK1 | 100 | 1 |
| ERK2 | 93 | 4 |
| ERK8 | 96 | 5 |
| GSK3 beta | 83 | 5 |
| HIPK2 | 93 | 6 |
| HIPK3 | 108 | 4 |
| IKK beta | 82 | 3 |
| JNK1 | 90 | 8 |
| JNK2 | 81 | 0 |
| JNK3 | 80 | 0 |
| Lck | 79 | 6 |
| MAPKAP-K2 | 108 | 4 |
| MAPKAP-K3 | 104 | 4 |
| MARK3 | 88 | 3 |
| MELK | 74 | 4 |
| MKK1 | 93 | 4 |
| MNK1 | 83 | 1 |
| MNK2 | 101 | 3 |
| MSK1 | 85 | 2 |
| MST2 | 90 | 5 |
| NEK2a | 82 | 5 |
| NEK6 | 95 | 3 |
| NEK7 | 102 | 5 |
| p38 alpha MAPK | 74 | 4 |
| p38 beta MAPK | 83 | 0 |
| p38 delta MAPK | 92 | 4 |
| p38 gamma MAPK | 80 | 7 |
| PAK4 | 81 | 1 |
| PAK5 | 89 | 8 |
| PAK6 | 88 | 1 |
| PDK1 | 84 | 0 |
| PHK | 95 | 2 |
| PIM1 | 91 | 2 |
| PIM2 | 117 | 0 |
| PIM3 | 88 | 1 |
| PKA | 77 | 1 |
| PKB alpha | 91 | 3 |
| PKB beta | 84 | 9 |
| PKC alpha | 88 | 3 |
| PKC zeta | 92 | 5 |
| PKD1 | 92 | 2 |
| PLK1 | 78 | 3 |
| PRAK | 91 | 2 |
| PRK2 | 78 | 1 |
| ROCK 2 | 103 | 3 |
| RSK1 | 90 | 3 |
| RSK2 | 97 | 5 |
| S6K1 | 105 | 7 |
| SGK1 | 93 | 1 |
| SmMLCK | 107 | 1 |
| Src | 85 | 0 |
| SRPK1 | 84 | 1 |