| Compound name | Brutto | MW | CAS | PubChem CID | Action | Reference | Reference |
|---|---|---|---|---|---|---|---|
| PS-1145 | C17H11ClN4O | 322.75 | 431898-65-6 | 9949093 | IKK | Castro A.C. (2003) Bioorg. Med. Chem. Lett. 13 2419-2422. |
| Kinase | % Activity Remaining | Standard Deviation |
|---|---|---|
| AMPK | 88 | 4 |
| Aurora B | 70 | 6 |
| Aurora C | 80 | 6 |
| BRSK2 | 90 | 1 |
| CAMK1 | 73 | 1 |
| CAMKK alpha | 80 | 1 |
| CAMKK beta | 69 | 8 |
| CDK2-Cyclin A | 76 | 0 |
| CHK1 | 90 | 5 |
| CHK2 | 102 | 8 |
| CK1 delta | 92 | 1 |
| CK2 | 87 | 1 |
| CSK | 83 | 1 |
| DYRK1A | 47 | 2 |
| DYRK2 | 89 | 1 |
| DYRK3 | 50 | 3 |
| EF2K | 100 | 2 |
| ERK1 | 106 | 8 |
| ERK2 | 84 | 3 |
| ERK8 | 42 | 6 |
| GSK3 beta | 46 | 6 |
| HIPK2 | 67 | 3 |
| HIPK3 | 89 | 2 |
| IKK beta |
4
|
0 |
| IKK epsilon | 81 | 3 |
| JNK1 | 86 | 4 |
| JNK2 | 93 | 1 |
| JNK3 | 92 | 0 |
| Lck | 57 | 3 |
| MAPKAP-K2 | 83 | 4 |
| MAPKAP-K3 | 95 | 9 |
| MARK3 | 89 | 4 |
| MELK | 70 | 1 |
| MKK1 | 83 | 1 |
| MNK1 | 44 | 2 |
| MNK2 | 70 | 2 |
| MSK1 | 99 | 1 |
| MST2 | 88 | 7 |
| NEK2a | 85 | 6 |
| NEK6 | 83 | 1 |
| NEK7 | 103 | 4 |
| p38 alpha MAPK | 89 | 4 |
| p38 beta MAPK | 84 | 6 |
| p38 delta MAPK | 78 | 7 |
| p38 gamma MAPK | 98 | 4 |
| PAK4 | 93 | 1 |
| PAK5 | 87 | 2 |
| PAK6 | 101 | 0 |
| PDK1 | 87 | 3 |
| PHK | 85 | 7 |
| PIM1 | 13 | 1 |
| PIM2 | 47 | 1 |
| PIM3 |
9
|
1 |
| PKA | 86 | 8 |
| PKB alpha | 90 | 1 |
| PKB beta | 101 | 9 |
| PKC alpha | 77 | 2 |
| PKC zeta | 78 | 6 |
| PKD1 | 108 | 4 |
| PLK1 | 98 | 6 |
| PRAK | 85 | 5 |
| PRK2 | 71 | 7 |
| ROCK 2 | 69 | 6 |
| RSK1 | 66 | 1 |
| RSK2 | 82 | 4 |
| S6K1 | 86 | 1 |
| SGK1 | 75 | 0 |
| SmMLCK | 88 | 1 |
| Src | 98 | 5 |
| SRPK1 | 88 | 2 |
| TBK1 | 87 | 1 |