Inhibitor | AG879 (Tyrphostin)  

Screen Conc: 10.00µM

Kinase Sort ascending	% Activity Remaining	Standard Deviation
YES1	85	1
VEGFR1	50	3
TBK1	97	1
SYK	138	2
SRPK1	61	12
Src	67	0
SmMLCK	52	5
SGK1	107	13
S6K1	64	14
RSK2	61	4
RSK1	79	1
ROCK 2	94	0
PRK2	114	16
PRAK	27	2
PLK1	13	2
PKD1	80	3
PKC zeta	67	2
PKC alpha	78	6
PKB beta	15	9
PKB alpha	94	4
PKA	93	10
PIM3	34	8
PIM2	53	5
PIM1	25	3
PHK	28	1
PDK1	96	5
PAK6	80	1
PAK5	519	649
PAK4	56	2
p38 gamma MAPK	92	3
p38 delta MAPK	86	11
p38 beta MAPK	86	8
p38 alpha MAPK	81	9
NEK6	101	16
NEK2a	82	18
MST4	72	14
MST2	54	1
MSK1	88	3
MNK2	76	9
MNK1	99	8
MKK1	83	13
MELK	8	4
MARK3	90	7
MAPKAP-K2	99	2
Lck	107	13
JNK2	70	9
JNK1	87	16
IRR	45	4
IR	139	52
IKK epsilon	63	9
IKK beta	105	13
IGF-1R	86	4
HIPK2	21	2
GSK3 beta	39	4
FGF-R1	59	0
ERK8	37	0
ERK2	87	1
ERK1	90	8
EPH-B3	55	1
EPH-A2	113	11
EF2K	90	8
DYRK3	60	1
DYRK2	102	31
DYRK1A	56	3
CSK	89	6
CK2	118	5
CK1 delta	92	6
CHK2	96	14
CHK1	92	19
CDK2-Cyclin A	40	0
CAMKK beta	44	12
CAMK1	88	7
BTK	46	8
BRSK2	66	4
AMPK	70	2

Screen Conc: 0.10µM

Kinase Sort ascending	% Activity Remaining	Standard Deviation
YES1	111	13
VEGFR1	92	3
TBK1	90	6
SYK	173	70
SRPK1	86	0
Src	95	11
SmMLCK	85	20
SGK1	124	15
S6K1	92	4
RSK2	67	2
RSK1	99	9
ROCK 2	113	10
PRK2	101	30
PRAK	102	2
PLK1	105	9
PKD1	99	12
PKC zeta	86	7
PKC alpha	101	10
PKB beta	84	3
PKB alpha	103	1
PKA	85	3
PIM3	98	19
PIM2	98	1
PIM1	102	22
PHK	93	19
PDK1	100	0
PAK6	86	1
PAK5	585	715
PAK4	105	11
p38 gamma MAPK	98	7
p38 delta MAPK	93	11
p38 beta MAPK	89	6
p38 alpha MAPK	105	7
NEK6	100	24
NEK2a	85	17
MST4	83	0
MST2	113	8
MSK1	82	3
MNK2	84	0
MNK1	101	4
MKK1	95	1
MELK	76	1
MARK3	92	6
MAPKAP-K2	108	11
Lck	99	8
JNK2	90	10
JNK1	99	9
IRR	88	0
IR	118	7
IKK epsilon	78	8
IKK beta	109	10
IGF-1R	98	16
HIPK2	118	15
GSK3 beta	95	7
FGF-R1	120	17
ERK8	96	2
ERK2	91	2
ERK1	88	16
EPH-B3	96	10
EPH-A2	94	12
EF2K	105	4
DYRK3	98	11
DYRK2	110	8
DYRK1A	84	1
CSK	92	15
CK2	123	8
CK1 delta	95	0
CHK2	109	23
CHK1	86	1
CDK2-Cyclin A	110	1
CAMKK beta	78	22
CAMK1	85	9
BTK	55	4
BRSK2	87	9
AMPK	78	0