Inhibitor | Piceatannol  

Compound name Brutto MW CAS PubChem CID Action Reference Reference
Piceatannol   C14H12O4 244.20 10083-24-6 667639 PKA, SYK Wang B.H. (1998) Planta Med. 64 195 Keely P.J. and Parise L.V. (1996) J. Biol. Chem. 271 26668

Screening Results Chart

Screening Results Tables

Screen Conc: 10.00µM
Kinase % Activity Remaining Standard Deviation
DYRK2 16 1
PIM1 25 2
DYRK1A 28 2
PIM3 31 1
MLK1 32 3
CLK2 32 3
MLK3 34 1
IR 36 10
MST2 37 6
DYRK3 38 10
SmMLCK 40 0
BRSK2 44 1
NEK2a 44 0
BRSK1 45 0
VEGFR1 45 6
NUAK1 47 14
FGF-R1 47 5
Src 48 8
HIPK2 49 2
PKB beta 51 7
PKC zeta 51 2
MARK3 51 3
SRPK1 52 1
EPH-B4 57 3
IRR 57 2
LKB1 58 6
PIM2 59 1
IKK epsilon 60 2
PAK4 62 8
Aurora B 63 13
ERK8 64 1
BTK 64 2
YES1 65 1
RSK2 65 7
CAMK1 66 1
MINK1 68 4
DAPK1 69 3
CHK2 69 5
RIPK2 69 3
PAK5 69 13
MARK1 69 5
PHK 71 1
Lck 71 2
HER4 72 2
TTK 72 2
RSK1 72 3
JAK2 72 5
TBK1 73 2
HIPK3 74 2
PKD1 75 3
MST4 75 13
p38 gamma MAPK 76 11
TrkA 76 2
MELK 77 5
p38 alpha MAPK 77 7
Aurora A 78 8
GCK 78 6
PAK6 80 6
MARK2 80 1
TAO1 82 4
ROCK 2 82 4
MEKK1 84 8
MNK1 84 11
SGK1 85 6
AMPK 85 11
MSK1 86 8
IKK beta 86 1
S6K1 87 6
GSK3 beta 87 5
IRAK4 87 8
MKK1 87 3
CAMKK beta 87 4
PRK2 88 7
CK1 delta 88 3
MARK4 89 0
PDK1 89 10
PKB alpha 89 10
EPH-A2 90 8
MAPKAP-K3 92 1
PAK2 93 7
p38 delta MAPK 93 3
HIPK1 94 4
PRAK 95 2
MNK2 96 3
EPH-B2 97 14
ERK2 98 1
PKC alpha 98 0
EPH-B3 99 14
JNK1 100 4
CK2 100 1
MKK6 101 10
PKA 101 2
PLK1 101 1
TAK1 102 7
MAPKAP-K2 102 13
EF2K 105 8
IGF-1R 105 5
NEK6 105 8
CDK2-Cyclin A 107 2
EPH-A4 108 4
CSK 108 8
MKK2 109 7
JNK2 111 1
EPH-B1 112 13
SYK 113 5
ASK1 114 8
p38 beta MAPK 114 15
JNK3 116 6
ERK1 121 6
CHK1 125 9
Screen Conc: 1.00µM
Kinase % Activity Remaining Standard Deviation
IR 61 10
ROCK 2 66 3
DYRK2 70 4
PKB beta 70 10
PIM3 72 3
p38 alpha MAPK 73 0
BRSK1 73 5
DYRK1A 76 7
NEK2a 77 2
SRPK1 78 3
NUAK1 79 13
RIPK2 80 7
Src 81 5
SmMLCK 81 11
MARK3 82 1
BRSK2 83 2
MLK3 84 8
MAPKAP-K2 85 3
PRK2 86 6
PAK4 86 11
IRR 86 1
PIM1 87 2
MLK1 87 14
MARK2 87 4
CHK1 88 3
DAPK1 89 3
MKK1 89 10
ERK8 90 7
HIPK3 91 3
LKB1 91 1
PKB alpha 91 6
S6K1 92 1
MST2 92 3
p38 delta MAPK 93 5
RSK1 93 2
CK1 delta 94 13
p38 beta MAPK 95 7
JAK2 96 5
JNK3 96 2
Aurora B 96 7
HER4 96 2
TTK 96 9
IKK beta 97 2
HIPK1 98 5
MNK1 98 4
MARK4 98 4
HIPK2 99 2
TAK1 99 1
Aurora A 99 4
PDK1 99 8
IKK epsilon 99 2
MKK6 99 1
SYK 100 7
FGF-R1 100 5
VEGFR1 100 12
ASK1 101 9
PKD1 101 2
PAK2 101 6
DYRK3 101 12
BTK 101 11
PHK 102 13
PIM2 102 8
CLK2 102 10
MARK1 102 10
MEKK1 103 10
EPH-A2 103 4
IRAK4 103 8
PAK5 103 15
JNK1 104 2
GSK3 beta 104 6
EPH-B3 104 5
NEK6 104 3
MSK1 105 12
PKA 106 2
CHK2 107 4
PKC zeta 108 2
MNK2 108 0
Lck 108 3
CSK 108 10
CAMK1 108 4
ERK2 109 7
MKK2 109 3
SGK1 109 10
PRAK 110 13
TrkA 110 5
YES1 110 6
MST4 110 4
MINK1 111 8
CDK2-Cyclin A 111 0
CAMKK beta 111 10
JNK2 112 5
TBK1 113 6
ERK1 113 7
p38 gamma MAPK 113 1
IGF-1R 113 6
PKC alpha 114 11
TAO1 114 14
CK2 115 8
RSK2 115 3
EPH-A4 116 2
EF2K 117 0
GCK 118 7
MAPKAP-K3 119 10
PAK6 119 10
EPH-B1 120 12
MELK 121 11
PLK1 125 6
EPH-B2 126 8
AMPK 126 2
EPH-B4 129 1