Compound name | Brutto | MW | CAS | PubChem CID | Action | Reference | Reference |
---|---|---|---|---|---|---|---|
Piceatannol | C14H12O4 | 244.20 | 10083-24-6 | 667639 | PKA, SYK | Wang B.H. (1998) Planta Med. 64 195 | Keely P.J. and Parise L.V. (1996) J. Biol. Chem. 271 26668 |
Kinase | % Activity Remaining | Standard Deviation |
---|---|---|
AMPK | 126 | 2 |
ASK1 | 101 | 9 |
Aurora A | 99 | 4 |
Aurora B | 96 | 7 |
BRSK1 | 73 | 5 |
BRSK2 | 83 | 2 |
BTK | 101 | 11 |
CAMK1 | 108 | 4 |
CAMKK beta | 111 | 10 |
CDK2-Cyclin A | 111 | 0 |
CHK1 | 88 | 3 |
CHK2 | 107 | 4 |
CK1 delta | 94 | 13 |
CK2 | 115 | 8 |
CLK2 | 102 | 10 |
CSK | 108 | 10 |
DAPK1 | 89 | 3 |
DYRK1A | 76 | 7 |
DYRK2 | 70 | 4 |
DYRK3 | 101 | 12 |
EF2K | 117 | 0 |
EPH-A2 | 103 | 4 |
EPH-A4 | 116 | 2 |
EPH-B1 | 120 | 12 |
EPH-B2 | 126 | 8 |
EPH-B3 | 104 | 5 |
EPH-B4 | 129 | 1 |
ERK1 | 113 | 7 |
ERK2 | 109 | 7 |
ERK8 | 90 | 7 |
FGF-R1 | 100 | 5 |
GCK | 118 | 7 |
GSK3 beta | 104 | 6 |
HER4 | 96 | 2 |
HIPK1 | 98 | 5 |
HIPK2 | 99 | 2 |
HIPK3 | 91 | 3 |
IGF-1R | 113 | 6 |
IKK beta | 97 | 2 |
IKK epsilon | 99 | 2 |
IR | 61 | 10 |
IRAK4 | 103 | 8 |
IRR | 86 | 1 |
JAK2 | 96 | 5 |
JNK1 | 104 | 2 |
JNK2 | 112 | 5 |
JNK3 | 96 | 2 |
Lck | 108 | 3 |
LKB1 | 91 | 1 |
MAPKAP-K2 | 85 | 3 |
MAPKAP-K3 | 119 | 10 |
MARK1 | 102 | 10 |
MARK2 | 87 | 4 |
MARK3 | 82 | 1 |
MARK4 | 98 | 4 |
MEKK1 | 103 | 10 |
MELK | 121 | 11 |
MINK1 | 111 | 8 |
MKK1 | 89 | 10 |
MKK2 | 109 | 3 |
MKK6 | 99 | 1 |
MLK1 | 87 | 14 |
MLK3 | 84 | 8 |
MNK1 | 98 | 4 |
MNK2 | 108 | 0 |
MSK1 | 105 | 12 |
MST2 | 92 | 3 |
MST4 | 110 | 4 |
NEK2a | 77 | 2 |
NEK6 | 104 | 3 |
NUAK1 | 79 | 13 |
p38 alpha MAPK | 73 | 0 |
p38 beta MAPK | 95 | 7 |
p38 delta MAPK | 93 | 5 |
p38 gamma MAPK | 113 | 1 |
PAK2 | 101 | 6 |
PAK4 | 86 | 11 |
PAK5 | 103 | 15 |
PAK6 | 119 | 10 |
PDK1 | 99 | 8 |
PHK | 102 | 13 |
PIM1 | 87 | 2 |
PIM2 | 102 | 8 |
PIM3 | 72 | 3 |
PKA | 106 | 2 |
PKB alpha | 91 | 6 |
PKB beta | 70 | 10 |
PKC alpha | 114 | 11 |
PKC zeta | 108 | 2 |
PKD1 | 101 | 2 |
PLK1 | 125 | 6 |
PRAK | 110 | 13 |
PRK2 | 86 | 6 |
RIPK2 | 80 | 7 |
ROCK 2 | 66 | 3 |
RSK1 | 93 | 2 |
RSK2 | 115 | 3 |
S6K1 | 92 | 1 |
SGK1 | 109 | 10 |
SmMLCK | 81 | 11 |
Src | 81 | 5 |
SRPK1 | 78 | 3 |
SYK | 100 | 7 |
TAK1 | 99 | 1 |
TAO1 | 114 | 14 |
TBK1 | 113 | 6 |
TrkA | 110 | 5 |
TTK | 96 | 9 |
VEGFR1 | 100 | 12 |
YES1 | 110 | 6 |
Kinase | % Activity Remaining | Standard Deviation |
---|---|---|
AMPK | 85 | 11 |
ASK1 | 114 | 8 |
Aurora A | 78 | 8 |
Aurora B | 63 | 13 |
BRSK1 | 45 | 0 |
BRSK2 | 44 | 1 |
BTK | 64 | 2 |
CAMK1 | 66 | 1 |
CAMKK beta | 87 | 4 |
CDK2-Cyclin A | 107 | 2 |
CHK1 | 125 | 9 |
CHK2 | 69 | 5 |
CK1 delta | 88 | 3 |
CK2 | 100 | 1 |
CLK2 | 32 | 3 |
CSK | 108 | 8 |
DAPK1 | 69 | 3 |
DYRK1A | 28 | 2 |
DYRK2 | 16 | 1 |
DYRK3 | 38 | 10 |
EF2K | 105 | 8 |
EPH-A2 | 90 | 8 |
EPH-A4 | 108 | 4 |
EPH-B1 | 112 | 13 |
EPH-B2 | 97 | 14 |
EPH-B3 | 99 | 14 |
EPH-B4 | 57 | 3 |
ERK1 | 121 | 6 |
ERK2 | 98 | 1 |
ERK8 | 64 | 1 |
FGF-R1 | 47 | 5 |
GCK | 78 | 6 |
GSK3 beta | 87 | 5 |
HER4 | 72 | 2 |
HIPK1 | 94 | 4 |
HIPK2 | 49 | 2 |
HIPK3 | 74 | 2 |
IGF-1R | 105 | 5 |
IKK beta | 86 | 1 |
IKK epsilon | 60 | 2 |
IR | 36 | 10 |
IRAK4 | 87 | 8 |
IRR | 57 | 2 |
JAK2 | 72 | 5 |
JNK1 | 100 | 4 |
JNK2 | 111 | 1 |
JNK3 | 116 | 6 |
Lck | 71 | 2 |
LKB1 | 58 | 6 |
MAPKAP-K2 | 102 | 13 |
MAPKAP-K3 | 92 | 1 |
MARK1 | 69 | 5 |
MARK2 | 80 | 1 |
MARK3 | 51 | 3 |
MARK4 | 89 | 0 |
MEKK1 | 84 | 8 |
MELK | 77 | 5 |
MINK1 | 68 | 4 |
MKK1 | 87 | 3 |
MKK2 | 109 | 7 |
MKK6 | 101 | 10 |
MLK1 | 32 | 3 |
MLK3 | 34 | 1 |
MNK1 | 84 | 11 |
MNK2 | 96 | 3 |
MSK1 | 86 | 8 |
MST2 | 37 | 6 |
MST4 | 75 | 13 |
NEK2a | 44 | 0 |
NEK6 | 105 | 8 |
NUAK1 | 47 | 14 |
p38 alpha MAPK | 77 | 7 |
p38 beta MAPK | 114 | 15 |
p38 delta MAPK | 93 | 3 |
p38 gamma MAPK | 76 | 11 |
PAK2 | 93 | 7 |
PAK4 | 62 | 8 |
PAK5 | 69 | 13 |
PAK6 | 80 | 6 |
PDK1 | 89 | 10 |
PHK | 71 | 1 |
PIM1 | 25 | 2 |
PIM2 | 59 | 1 |
PIM3 | 31 | 1 |
PKA | 101 | 2 |
PKB alpha | 89 | 10 |
PKB beta | 51 | 7 |
PKC alpha | 98 | 0 |
PKC zeta | 51 | 2 |
PKD1 | 75 | 3 |
PLK1 | 101 | 1 |
PRAK | 95 | 2 |
PRK2 | 88 | 7 |
RIPK2 | 69 | 3 |
ROCK 2 | 82 | 4 |
RSK1 | 72 | 3 |
RSK2 | 65 | 7 |
S6K1 | 87 | 6 |
SGK1 | 85 | 6 |
SmMLCK | 40 | 0 |
Src | 48 | 8 |
SRPK1 | 52 | 1 |
SYK | 113 | 5 |
TAK1 | 102 | 7 |
TAO1 | 82 | 4 |
TBK1 | 73 | 2 |
TrkA | 76 | 2 |
TTK | 72 | 2 |
VEGFR1 | 45 | 6 |
YES1 | 65 | 1 |