Inhibitor | Piceatannol  

Compound name Brutto MW CAS PubChem CID Action Reference Reference
Piceatannol   C14H12O4 244.20 10083-24-6 667639 PKA, SYK Wang B.H. (1998) Planta Med. 64 195 Keely P.J. and Parise L.V. (1996) J. Biol. Chem. 271 26668

Screening Results Chart

Screening Results Tables

Screen Conc: 1.00µM
Kinase % Activity Remaining Standard Deviation
AMPK 126 2
ASK1 101 9
Aurora A 99 4
Aurora B 96 7
BRSK1 73 5
BRSK2 83 2
BTK 101 11
CAMK1 108 4
CAMKK beta 111 10
CDK2-Cyclin A 111 0
CHK1 88 3
CHK2 107 4
CK1 delta 94 13
CK2 115 8
CLK2 102 10
CSK 108 10
DAPK1 89 3
DYRK1A 76 7
DYRK2 70 4
DYRK3 101 12
EF2K 117 0
EPH-A2 103 4
EPH-A4 116 2
EPH-B1 120 12
EPH-B2 126 8
EPH-B3 104 5
EPH-B4 129 1
ERK1 113 7
ERK2 109 7
ERK8 90 7
FGF-R1 100 5
GCK 118 7
GSK3 beta 104 6
HER4 96 2
HIPK1 98 5
HIPK2 99 2
HIPK3 91 3
IGF-1R 113 6
IKK beta 97 2
IKK epsilon 99 2
IR 61 10
IRAK4 103 8
IRR 86 1
JAK2 96 5
JNK1 104 2
JNK2 112 5
JNK3 96 2
Lck 108 3
LKB1 91 1
MAPKAP-K2 85 3
MAPKAP-K3 119 10
MARK1 102 10
MARK2 87 4
MARK3 82 1
MARK4 98 4
MEKK1 103 10
MELK 121 11
MINK1 111 8
MKK1 89 10
MKK2 109 3
MKK6 99 1
MLK1 87 14
MLK3 84 8
MNK1 98 4
MNK2 108 0
MSK1 105 12
MST2 92 3
MST4 110 4
NEK2a 77 2
NEK6 104 3
NUAK1 79 13
p38 alpha MAPK 73 0
p38 beta MAPK 95 7
p38 delta MAPK 93 5
p38 gamma MAPK 113 1
PAK2 101 6
PAK4 86 11
PAK5 103 15
PAK6 119 10
PDK1 99 8
PHK 102 13
PIM1 87 2
PIM2 102 8
PIM3 72 3
PKA 106 2
PKB alpha 91 6
PKB beta 70 10
PKC alpha 114 11
PKC zeta 108 2
PKD1 101 2
PLK1 125 6
PRAK 110 13
PRK2 86 6
RIPK2 80 7
ROCK 2 66 3
RSK1 93 2
RSK2 115 3
S6K1 92 1
SGK1 109 10
SmMLCK 81 11
Src 81 5
SRPK1 78 3
SYK 100 7
TAK1 99 1
TAO1 114 14
TBK1 113 6
TrkA 110 5
TTK 96 9
VEGFR1 100 12
YES1 110 6
Screen Conc: 10.00µM
Kinase % Activity Remaining Standard Deviation
AMPK 85 11
ASK1 114 8
Aurora A 78 8
Aurora B 63 13
BRSK1 45 0
BRSK2 44 1
BTK 64 2
CAMK1 66 1
CAMKK beta 87 4
CDK2-Cyclin A 107 2
CHK1 125 9
CHK2 69 5
CK1 delta 88 3
CK2 100 1
CLK2 32 3
CSK 108 8
DAPK1 69 3
DYRK1A 28 2
DYRK2 16 1
DYRK3 38 10
EF2K 105 8
EPH-A2 90 8
EPH-A4 108 4
EPH-B1 112 13
EPH-B2 97 14
EPH-B3 99 14
EPH-B4 57 3
ERK1 121 6
ERK2 98 1
ERK8 64 1
FGF-R1 47 5
GCK 78 6
GSK3 beta 87 5
HER4 72 2
HIPK1 94 4
HIPK2 49 2
HIPK3 74 2
IGF-1R 105 5
IKK beta 86 1
IKK epsilon 60 2
IR 36 10
IRAK4 87 8
IRR 57 2
JAK2 72 5
JNK1 100 4
JNK2 111 1
JNK3 116 6
Lck 71 2
LKB1 58 6
MAPKAP-K2 102 13
MAPKAP-K3 92 1
MARK1 69 5
MARK2 80 1
MARK3 51 3
MARK4 89 0
MEKK1 84 8
MELK 77 5
MINK1 68 4
MKK1 87 3
MKK2 109 7
MKK6 101 10
MLK1 32 3
MLK3 34 1
MNK1 84 11
MNK2 96 3
MSK1 86 8
MST2 37 6
MST4 75 13
NEK2a 44 0
NEK6 105 8
NUAK1 47 14
p38 alpha MAPK 77 7
p38 beta MAPK 114 15
p38 delta MAPK 93 3
p38 gamma MAPK 76 11
PAK2 93 7
PAK4 62 8
PAK5 69 13
PAK6 80 6
PDK1 89 10
PHK 71 1
PIM1 25 2
PIM2 59 1
PIM3 31 1
PKA 101 2
PKB alpha 89 10
PKB beta 51 7
PKC alpha 98 0
PKC zeta 51 2
PKD1 75 3
PLK1 101 1
PRAK 95 2
PRK2 88 7
RIPK2 69 3
ROCK 2 82 4
RSK1 72 3
RSK2 65 7
S6K1 87 6
SGK1 85 6
SmMLCK 40 0
Src 48 8
SRPK1 52 1
SYK 113 5
TAK1 102 7
TAO1 82 4
TBK1 73 2
TrkA 76 2
TTK 72 2
VEGFR1 45 6
YES1 65 1