Inhibitor | PI-103  

Screen Conc: 10.00µM

Kinase	% Activity Remaining Sort descending	Standard Deviation
SmMLCK	18	5
DYRK3	21	4
PIM3	27	8
RSK1	41	0
ERK8	45	6
GSK3 beta	48	4
RSK2	51	5
PKC alpha	53	0
PRK2	55	4
MELK	55	2
PHK	56	4
PIM1	60	8
HIPK2	60	0
Lck	62	1
BRSK2	63	1
DYRK1A	64	1
PKB alpha	65	0
CK1 delta	68	0
HIPK3	68	0
MKK1	69	3
CDK2-Cyclin A	70	1
MNK1	71	6
CAMKK beta	72	1
DYRK2	72	1
Aurora C	73	4
MST2	73	5
CAMK1	73	1
CSK	74	2
PAK4	75	5
PKA	77	1
NEK2a	77	9
PIM2	77	4
MARK3	77	2
CK2	77	2
SRPK1	78	2
CAMKK alpha	78	5
PKC zeta	79	4
IKK beta	79	0
PRAK	79	4
PKB beta	79	2
SGK1	79	4
JNK2	81	6
Aurora B	81	1
Src	82	8
NEK6	83	0
MSK1	83	1
MNK2	84	1
CHK1	85	0
p38 alpha MAPK	86	0
PLK1	86	1
PAK5	86	3
S6K1	86	2
ROCK 2	87	5
JNK3	87	0
PKD1	87	7
p38 delta MAPK	87	0
AMPK	88	0
ERK2	90	4
PDK1	91	1
JNK1	95	7
CHK2	97	0
p38 beta MAPK	97	3
MAPKAP-K3	97	7
PAK6	97	0
p38 gamma MAPK	99	2
NEK7	104	4
EF2K	108	4
MAPKAP-K2	110	5
ERK1	114	5

Screen Conc: 1.00µM

Kinase	% Activity Remaining Sort descending	Standard Deviation
SmMLCK	62	5
HIPK2	67	0
MKK1	68	5
PKA	73	6
ERK8	74	3
PKB alpha	74	2
HIPK3	75	6
ROCK 2	75	3
PKB beta	76	5
PKC zeta	76	2
PIM1	77	2
CHK2	78	11
PLK1	79	10
PIM3	79	2
MELK	79	8
CAMKK beta	79	5
DYRK3	79	8
PRK2	80	8
p38 delta MAPK	81	4
S6K1	81	7
DYRK2	81	7
SRPK1	82	8
CK2	82	6
CSK	82	0
PKC alpha	82	4
Aurora B	83	1
PHK	83	5
GSK3 beta	84	10
p38 beta MAPK	85	5
CK1 delta	87	1
DYRK1A	87	5
MAPKAP-K3	88	15
CAMKK alpha	88	7
SGK1	88	2
ERK1	88	6
MNK1	89	6
Lck	89	2
RSK1	90	13
PDK1	90	1
PAK5	90	8
Src	90	7
JNK3	90	6
MST2	91	5
p38 alpha MAPK	91	5
PKD1	92	2
PRAK	92	6
JNK2	93	4
CHK1	94	5
CDK2-Cyclin A	95	5
IKK beta	95	4
MSK1	96	1
BRSK2	96	0
ERK2	96	4
p38 gamma MAPK	97	8
PAK4	97	4
JNK1	97	3
PAK6	98	7
MAPKAP-K2	99	17
MARK3	99	6
Aurora C	103	3
MNK2	103	11
RSK2	104	9
AMPK	105	15
PIM2	106	7
NEK7	106	1
CAMK1	108	7
EF2K	110	13
NEK6	111	6
NEK2a	114	2