Inhibitor | PD 184352 (CI-1040)  

Screen Conc: 1.00µM

Kinase	% Activity Remaining	Standard Deviation
AMPK	80	4
Aurora B	77	4
Aurora C	82	4
BRSK2	83	5
CAMK1	81	4
CAMKK alpha	87	2
CAMKK beta	90	1
CDK2-Cyclin A	79	3
CHK1	84	6
CHK2	110	4
CK1 delta	99	5
CK2	102	0
CSK	77	6
DYRK1A	86	6
DYRK2	93	7
DYRK3	88	3
EF2K	80	1
ERK1	106	6
ERK2	102	5
ERK8	107	2
GSK3 beta	65	4
HIPK2	85	5
HIPK3	94	9
IKK beta	88	4
JNK1	101	4
JNK2	95	3
JNK3	94	0
Lck	70	2
MAPKAP-K2	85	3
MAPKAP-K3	81	5
MARK3	80	2
MELK	64	2
MKK1	45	0
MNK1	92	4
MNK2	101	4
MSK1	88	7
MST2	68	1
NEK2a	86	0
NEK6	89	2
NEK7	110	4
p38 alpha MAPK	109	3
p38 beta MAPK	104	5
p38 delta MAPK	87	1
p38 gamma MAPK	96	1
PAK4	95	1
PAK5	82	7
PAK6	75	1
PDK1	82	0
PHK	70	2
PIM1	84	8
PIM2	94	2
PIM3	56	1
PKA	66	3
PKB alpha	92	8
PKB beta	103	1
PKC alpha	64	2
PKC zeta	81	6
PKD1	100	1
PLK1	90	4
PRAK	81	2
PRK2	69	4
ROCK 2	82	7
RSK1	48	5
RSK2	58	6
S6K1	87	1
SGK1	84	3
SmMLCK	86	7
Src	100	1
SRPK1	85	0

Screen Conc: 10.00µM

Kinase	% Activity Remaining	Standard Deviation
AMPK	108	3
Aurora B	70	1
Aurora C	96	9
BRSK2	82	5
CAMK1	69	4
CAMKK alpha	77	1
CAMKK beta	90	1
CDK2-Cyclin A	88	8
CHK1	113	1
CHK2	95	8
CK1 delta	100	1
CK2	90	10
CSK	81	2
DYRK1A	80	2
DYRK2	76	2
DYRK3	104	2
EF2K	97	0
ERK1	86	0
ERK2	83	3
ERK8	94	2
GSK3 beta	78	6
HIPK2	151	5
HIPK3	95	6
IKK beta	92	0
JNK1	92	1
JNK2	110	4
JNK3	108	4
Lck	85	2
MAPKAP-K2	81	5
MAPKAP-K3	84	8
MARK3	98	2
MELK	82	3
MKK1	12	1
MNK1	92	9
MNK2	99	3
MSK1	91	5
MST2	89	1
NEK2a	98	1
NEK6	90	6
NEK7	93	1
p38 alpha MAPK	86	7
p38 beta MAPK	96	7
p38 delta MAPK	93	2
p38 gamma MAPK	87	3
PAK4	82	3
PAK5	98	9
PAK6	100	1
PDK1	79	4
PHK	98	2
PIM1	75	3
PIM2	92	1
PIM3	66	4
PKA	87	0
PKB alpha	87	7
PKB beta	80	0
PKC alpha	88	2
PKC zeta	72	0
PKD1	85	3
PLK1	82	0
PRAK	82	1
PRK2	83	1
ROCK 2	86	0
RSK1	124	11
RSK2	92	4
S6K1	89	1
SGK1	101	6
SmMLCK	105	3
Src	90	5
SRPK1	94	4