Inhibitor |
AG879 (Tyrphostin)
Screening Results Tables
Screen Conc:
0.10µM
Kinase |
% Activity Remaining |
Standard Deviation |
AMPK
|
78
|
0
|
BRSK2
|
87
|
9
|
BTK
|
55
|
4
|
CAMK1
|
85
|
9
|
CAMKK beta
|
78
|
22
|
CDK2-Cyclin A
|
110
|
1
|
CHK1
|
86
|
1
|
CHK2
|
109
|
23
|
CK1 delta
|
95
|
0
|
CK2
|
123
|
8
|
CSK
|
92
|
15
|
DYRK1A
|
84
|
1
|
DYRK2
|
110
|
8
|
DYRK3
|
98
|
11
|
EF2K
|
105
|
4
|
EPH-A2
|
94
|
12
|
EPH-B3
|
96
|
10
|
ERK1
|
88
|
16
|
ERK2
|
91
|
2
|
ERK8
|
96
|
2
|
FGF-R1
|
120
|
17
|
GSK3 beta
|
95
|
7
|
HIPK2
|
118
|
15
|
IGF-1R
|
98
|
16
|
IKK beta
|
109
|
10
|
IKK epsilon
|
78
|
8
|
IR
|
118
|
7
|
IRR
|
88
|
0
|
JNK1
|
99
|
9
|
JNK2
|
90
|
10
|
Lck
|
99
|
8
|
MAPKAP-K2
|
108
|
11
|
MARK3
|
92
|
6
|
MELK
|
76
|
1
|
MKK1
|
95
|
1
|
MNK1
|
101
|
4
|
MNK2
|
84
|
0
|
MSK1
|
82
|
3
|
MST2
|
113
|
8
|
MST4
|
83
|
0
|
NEK2a
|
85
|
17
|
NEK6
|
100
|
24
|
p38 alpha MAPK
|
105
|
7
|
p38 beta MAPK
|
89
|
6
|
p38 delta MAPK
|
93
|
11
|
p38 gamma MAPK
|
98
|
7
|
PAK4
|
105
|
11
|
PAK5
|
585
|
715
|
PAK6
|
86
|
1
|
PDK1
|
100
|
0
|
PHK
|
93
|
19
|
PIM1
|
102
|
22
|
PIM2
|
98
|
1
|
PIM3
|
98
|
19
|
PKA
|
85
|
3
|
PKB alpha
|
103
|
1
|
PKB beta
|
84
|
3
|
PKC alpha
|
101
|
10
|
PKC zeta
|
86
|
7
|
PKD1
|
99
|
12
|
PLK1
|
105
|
9
|
PRAK
|
102
|
2
|
PRK2
|
101
|
30
|
ROCK 2
|
113
|
10
|
RSK1
|
99
|
9
|
RSK2
|
67
|
2
|
S6K1
|
92
|
4
|
SGK1
|
124
|
15
|
SmMLCK
|
85
|
20
|
Src
|
95
|
11
|
SRPK1
|
86
|
0
|
SYK
|
173
|
70
|
TBK1
|
90
|
6
|
VEGFR1
|
92
|
3
|
YES1
|
111
|
13
|
Screen Conc:
10.00µM
Kinase |
% Activity Remaining |
Standard Deviation |
AMPK
|
70
|
2
|
BRSK2
|
66
|
4
|
BTK
|
46
|
8
|
CAMK1
|
88
|
7
|
CAMKK beta
|
44
|
12
|
CDK2-Cyclin A
|
40
|
0
|
CHK1
|
92
|
19
|
CHK2
|
96
|
14
|
CK1 delta
|
92
|
6
|
CK2
|
118
|
5
|
CSK
|
89
|
6
|
DYRK1A
|
56
|
3
|
DYRK2
|
102
|
31
|
DYRK3
|
60
|
1
|
EF2K
|
90
|
8
|
EPH-A2
|
113
|
11
|
EPH-B3
|
55
|
1
|
ERK1
|
90
|
8
|
ERK2
|
87
|
1
|
ERK8
|
37
|
0
|
FGF-R1
|
59
|
0
|
GSK3 beta
|
39
|
4
|
HIPK2
|
21
|
2
|
IGF-1R
|
86
|
4
|
IKK beta
|
105
|
13
|
IKK epsilon
|
63
|
9
|
IR
|
139
|
52
|
IRR
|
45
|
4
|
JNK1
|
87
|
16
|
JNK2
|
70
|
9
|
Lck
|
107
|
13
|
MAPKAP-K2
|
99
|
2
|
MARK3
|
90
|
7
|
MELK
|
8
|
4
|
MKK1
|
83
|
13
|
MNK1
|
99
|
8
|
MNK2
|
76
|
9
|
MSK1
|
88
|
3
|
MST2
|
54
|
1
|
MST4
|
72
|
14
|
NEK2a
|
82
|
18
|
NEK6
|
101
|
16
|
p38 alpha MAPK
|
81
|
9
|
p38 beta MAPK
|
86
|
8
|
p38 delta MAPK
|
86
|
11
|
p38 gamma MAPK
|
92
|
3
|
PAK4
|
56
|
2
|
PAK5
|
519
|
649
|
PAK6
|
80
|
1
|
PDK1
|
96
|
5
|
PHK
|
28
|
1
|
PIM1
|
25
|
3
|
PIM2
|
53
|
5
|
PIM3
|
34
|
8
|
PKA
|
93
|
10
|
PKB alpha
|
94
|
4
|
PKB beta
|
15
|
9
|
PKC alpha
|
78
|
6
|
PKC zeta
|
67
|
2
|
PKD1
|
80
|
3
|
PLK1
|
13
|
2
|
PRAK
|
27
|
2
|
PRK2
|
114
|
16
|
ROCK 2
|
94
|
0
|
RSK1
|
79
|
1
|
RSK2
|
61
|
4
|
S6K1
|
64
|
14
|
SGK1
|
107
|
13
|
SmMLCK
|
52
|
5
|
Src
|
67
|
0
|
SRPK1
|
61
|
12
|
SYK
|
138
|
2
|
TBK1
|
97
|
1
|
VEGFR1
|
50
|
3
|
YES1
|
85
|
1
|