Inhibitor | AG879 (Tyrphostin)  

Screen Conc: 0.10µM

Kinase	% Activity Remaining	Standard Deviation
AMPK	78	0
BRSK2	87	9
BTK	55	4
CAMK1	85	9
CAMKK beta	78	22
CDK2-Cyclin A	110	1
CHK1	86	1
CHK2	109	23
CK1 delta	95	0
CK2	123	8
CSK	92	15
DYRK1A	84	1
DYRK2	110	8
DYRK3	98	11
EF2K	105	4
EPH-A2	94	12
EPH-B3	96	10
ERK1	88	16
ERK2	91	2
ERK8	96	2
FGF-R1	120	17
GSK3 beta	95	7
HIPK2	118	15
IGF-1R	98	16
IKK beta	109	10
IKK epsilon	78	8
IR	118	7
IRR	88	0
JNK1	99	9
JNK2	90	10
Lck	99	8
MAPKAP-K2	108	11
MARK3	92	6
MELK	76	1
MKK1	95	1
MNK1	101	4
MNK2	84	0
MSK1	82	3
MST2	113	8
MST4	83	0
NEK2a	85	17
NEK6	100	24
p38 alpha MAPK	105	7
p38 beta MAPK	89	6
p38 delta MAPK	93	11
p38 gamma MAPK	98	7
PAK4	105	11
PAK5	585	715
PAK6	86	1
PDK1	100	0
PHK	93	19
PIM1	102	22
PIM2	98	1
PIM3	98	19
PKA	85	3
PKB alpha	103	1
PKB beta	84	3
PKC alpha	101	10
PKC zeta	86	7
PKD1	99	12
PLK1	105	9
PRAK	102	2
PRK2	101	30
ROCK 2	113	10
RSK1	99	9
RSK2	67	2
S6K1	92	4
SGK1	124	15
SmMLCK	85	20
Src	95	11
SRPK1	86	0
SYK	173	70
TBK1	90	6
VEGFR1	92	3
YES1	111	13

Screen Conc: 10.00µM

Kinase	% Activity Remaining	Standard Deviation
AMPK	70	2
BRSK2	66	4
BTK	46	8
CAMK1	88	7
CAMKK beta	44	12
CDK2-Cyclin A	40	0
CHK1	92	19
CHK2	96	14
CK1 delta	92	6
CK2	118	5
CSK	89	6
DYRK1A	56	3
DYRK2	102	31
DYRK3	60	1
EF2K	90	8
EPH-A2	113	11
EPH-B3	55	1
ERK1	90	8
ERK2	87	1
ERK8	37	0
FGF-R1	59	0
GSK3 beta	39	4
HIPK2	21	2
IGF-1R	86	4
IKK beta	105	13
IKK epsilon	63	9
IR	139	52
IRR	45	4
JNK1	87	16
JNK2	70	9
Lck	107	13
MAPKAP-K2	99	2
MARK3	90	7
MELK	8	4
MKK1	83	13
MNK1	99	8
MNK2	76	9
MSK1	88	3
MST2	54	1
MST4	72	14
NEK2a	82	18
NEK6	101	16
p38 alpha MAPK	81	9
p38 beta MAPK	86	8
p38 delta MAPK	86	11
p38 gamma MAPK	92	3
PAK4	56	2
PAK5	519	649
PAK6	80	1
PDK1	96	5
PHK	28	1
PIM1	25	3
PIM2	53	5
PIM3	34	8
PKA	93	10
PKB alpha	94	4
PKB beta	15	9
PKC alpha	78	6
PKC zeta	67	2
PKD1	80	3
PLK1	13	2
PRAK	27	2
PRK2	114	16
ROCK 2	94	0
RSK1	79	1
RSK2	61	4
S6K1	64	14
SGK1	107	13
SmMLCK	52	5
Src	67	0
SRPK1	61	12
SYK	138	2
TBK1	97	1
VEGFR1	50	3
YES1	85	1