Inhibitor | AG879 (Tyrphostin)
Screening Results Tables
Screen Conc: 0.10µM
Kinase |
% Activity Remaining |
Standard Deviation |
AMPK |
78
|
0 |
BRSK2 |
87
|
9 |
BTK |
55
|
4 |
CAMK1 |
85
|
9 |
CAMKK beta |
78
|
22 |
CDK2-Cyclin A |
110
|
1 |
CHK1 |
86
|
1 |
CHK2 |
109
|
23 |
CK1 delta |
95
|
0 |
CK2 |
123
|
8 |
CSK |
92
|
15 |
DYRK1A |
84
|
1 |
DYRK2 |
110
|
8 |
DYRK3 |
98
|
11 |
EF2K |
105
|
4 |
EPH-A2 |
94
|
12 |
EPH-B3 |
96
|
10 |
ERK1 |
88
|
16 |
ERK2 |
91
|
2 |
ERK8 |
96
|
2 |
FGF-R1 |
120
|
17 |
GSK3 beta |
95
|
7 |
HIPK2 |
118
|
15 |
IGF-1R |
98
|
16 |
IKK beta |
109
|
10 |
IKK epsilon |
78
|
8 |
IR |
118
|
7 |
IRR |
88
|
0 |
JNK1 |
99
|
9 |
JNK2 |
90
|
10 |
Lck |
99
|
8 |
MAPKAP-K2 |
108
|
11 |
MARK3 |
92
|
6 |
MELK |
76
|
1 |
MKK1 |
95
|
1 |
MNK1 |
101
|
4 |
MNK2 |
84
|
0 |
MSK1 |
82
|
3 |
MST2 |
113
|
8 |
MST4 |
83
|
0 |
NEK2a |
85
|
17 |
NEK6 |
100
|
24 |
p38 alpha MAPK |
105
|
7 |
p38 beta MAPK |
89
|
6 |
p38 delta MAPK |
93
|
11 |
p38 gamma MAPK |
98
|
7 |
PAK4 |
105
|
11 |
PAK5 |
585
|
715 |
PAK6 |
86
|
1 |
PDK1 |
100
|
0 |
PHK |
93
|
19 |
PIM1 |
102
|
22 |
PIM2 |
98
|
1 |
PIM3 |
98
|
19 |
PKA |
85
|
3 |
PKB alpha |
103
|
1 |
PKB beta |
84
|
3 |
PKC alpha |
101
|
10 |
PKC zeta |
86
|
7 |
PKD1 |
99
|
12 |
PLK1 |
105
|
9 |
PRAK |
102
|
2 |
PRK2 |
101
|
30 |
ROCK 2 |
113
|
10 |
RSK1 |
99
|
9 |
RSK2 |
67
|
2 |
S6K1 |
92
|
4 |
SGK1 |
124
|
15 |
SmMLCK |
85
|
20 |
Src |
95
|
11 |
SRPK1 |
86
|
0 |
SYK |
173
|
70 |
TBK1 |
90
|
6 |
VEGFR1 |
92
|
3 |
YES1 |
111
|
13 |
Screen Conc: 10.00µM
Kinase |
% Activity Remaining |
Standard Deviation |
AMPK |
70
|
2 |
BRSK2 |
66
|
4 |
BTK |
46
|
8 |
CAMK1 |
88
|
7 |
CAMKK beta |
44
|
12 |
CDK2-Cyclin A |
40
|
0 |
CHK1 |
92
|
19 |
CHK2 |
96
|
14 |
CK1 delta |
92
|
6 |
CK2 |
118
|
5 |
CSK |
89
|
6 |
DYRK1A |
56
|
3 |
DYRK2 |
102
|
31 |
DYRK3 |
60
|
1 |
EF2K |
90
|
8 |
EPH-A2 |
113
|
11 |
EPH-B3 |
55
|
1 |
ERK1 |
90
|
8 |
ERK2 |
87
|
1 |
ERK8 |
37
|
0 |
FGF-R1 |
59
|
0 |
GSK3 beta |
39
|
4 |
HIPK2 |
21
|
2 |
IGF-1R |
86
|
4 |
IKK beta |
105
|
13 |
IKK epsilon |
63
|
9 |
IR |
139
|
52 |
IRR |
45
|
4 |
JNK1 |
87
|
16 |
JNK2 |
70
|
9 |
Lck |
107
|
13 |
MAPKAP-K2 |
99
|
2 |
MARK3 |
90
|
7 |
MELK |
8
|
4 |
MKK1 |
83
|
13 |
MNK1 |
99
|
8 |
MNK2 |
76
|
9 |
MSK1 |
88
|
3 |
MST2 |
54
|
1 |
MST4 |
72
|
14 |
NEK2a |
82
|
18 |
NEK6 |
101
|
16 |
p38 alpha MAPK |
81
|
9 |
p38 beta MAPK |
86
|
8 |
p38 delta MAPK |
86
|
11 |
p38 gamma MAPK |
92
|
3 |
PAK4 |
56
|
2 |
PAK5 |
519
|
649 |
PAK6 |
80
|
1 |
PDK1 |
96
|
5 |
PHK |
28
|
1 |
PIM1 |
25
|
3 |
PIM2 |
53
|
5 |
PIM3 |
34
|
8 |
PKA |
93
|
10 |
PKB alpha |
94
|
4 |
PKB beta |
15
|
9 |
PKC alpha |
78
|
6 |
PKC zeta |
67
|
2 |
PKD1 |
80
|
3 |
PLK1 |
13
|
2 |
PRAK |
27
|
2 |
PRK2 |
114
|
16 |
ROCK 2 |
94
|
0 |
RSK1 |
79
|
1 |
RSK2 |
61
|
4 |
S6K1 |
64
|
14 |
SGK1 |
107
|
13 |
SmMLCK |
52
|
5 |
Src |
67
|
0 |
SRPK1 |
61
|
12 |
SYK |
138
|
2 |
TBK1 |
97
|
1 |
VEGFR1 |
50
|
3 |
YES1 |
85
|
1 |