

Compound name | Brutto | MW | CAS | PubChem CID | Action | Reference | Reference |
---|---|---|---|---|---|---|---|
ML-9, Hydrochloride | C15H17ClN2O2S • HCl | 361.30 | 105637-50-1 | 108047 | MLCK | Reig J.A. (1993) Neurochem. Res. 18 317 | Nagatsu T. (1987) Biochem. Biophys. Res. Commun. 143 1045 |
Kinase | % Activity Remaining | Standard Deviation |
---|---|---|
AMPK | 85 | 14 |
Aurora B | 63 | 2 |
CAMK1 | 74 | 8 |
CDK2-Cyclin A | 57 | 2 |
CHK1 | 86 | 5 |
CHK2 | 77 | 5 |
CK1 delta | 91 | 3 |
CK2 | 78 | 4 |
CSK | 80 | 8 |
DYRK1A | 84 | 16 |
EF2K | 88 | 12 |
ERK2 | 96 | 7 |
ERK8 | 84 | 10 |
GSK3 beta | 80 | 5 |
IKK beta | 71 | 1 |
JNK1 | 84 | 9 |
JNK3 | 76 | 1 |
Lck | 75 | 0 |
MAPKAP-K2 | 85 | 4 |
MAPKAP-K3 | 97 | 6 |
MARK3 | 103 | 5 |
MKK1 | 58 | 14 |
MNK1 | 66 | 0 |
MNK2 | 81 | 9 |
MSK1 | 30 | 1 |
MST2 | 82 | 0 |
NEK2a | 83 | 0 |
NEK6 | 103 | 14 |
NEK7 | 92 | 8 |
p38 alpha MAPK | 88 | 3 |
p38 beta MAPK | 80 | 4 |
p38 delta MAPK | 65 | 13 |
p38 gamma MAPK | 91 | 4 |
PDK1 | 96 | 7 |
PHK | 95 | 5 |
PIM2 | 63 | 0 |
PKA | 61 | 3 |
PKB alpha | 89 | 5 |
PKB beta | 92 | 4 |
PKC alpha | 72 | 2 |
PKD1 | 85 | 8 |
PLK1 | 101 | 6 |
PRAK | 77 | 1 |
PRK2 | 15 | 0 |
ROCK 2 | 28 | 0 |
RSK1 | 43 | 8 |
RSK2 | 67 | 6 |
S6K1 | 32 | 6 |
SGK1 | 82 | 11 |
SmMLCK | 95 | 40 |
Src | 82 | 3 |
SRPK1 | 87 | 16 |
Kinase | % Activity Remaining | Standard Deviation |
---|---|---|
AMPK | 32 | 3 |
Aurora B | 57 | 2 |
Aurora C | 73 | 3 |
BRSK2 |
2
|
5 |
CAMK1 | 17 | 3 |
CAMKK alpha | 108 | 1 |
CAMKK beta | 75 | 1 |
CDK2-Cyclin A | 13 | 1 |
CHK1 | 94 | 2 |
CHK2 | 108 | 5 |
CK1 delta | 58 | 3 |
CK2 | 25 | 2 |
CSK | 78 | 2 |
DYRK1A | 46 | 5 |
DYRK2 | 79 | 6 |
DYRK3 | 30 | 2 |
EF2K | 122 | 1 |
ERK1 | 91 | 1 |
ERK2 | 91 | 8 |
ERK8 | 50 | 2 |
GSK3 beta | 88 | 1 |
HIPK2 | 43 | 1 |
HIPK3 | 68 | 5 |
IKK beta | 67 | 1 |
JNK1 | 115 | 1 |
JNK2 | 92 | 4 |
JNK3 | 92 | 0 |
Lck | 81 | 1 |
MAPKAP-K2 | 69 | 4 |
MAPKAP-K3 | 79 | 2 |
MARK3 | 130 | 1 |
MELK | 66 | 7 |
MKK1 | 75 | 3 |
MNK1 | 28 | 4 |
MNK2 | 40 | 2 |
MSK1 | 11 | 3 |
MST2 | 74 | 4 |
NEK2a | 94 | 3 |
NEK6 | 105 | 1 |
NEK7 | 122 | 6 |
p38 alpha MAPK | 92 | 6 |
p38 beta MAPK | 86 | 1 |
p38 delta MAPK | 88 | 4 |
p38 gamma MAPK | 87 | 4 |
PAK4 | 94 | 1 |
PAK5 | 85 | 4 |
PAK6 | 108 | 4 |
PDK1 | 87 | 2 |
PHK | 47 | 6 |
PIM1 |
7
|
0 |
PIM2 | 43 | 6 |
PIM3 |
7
|
0 |
PKA | 25 | 5 |
PKB alpha | 44 | 4 |
PKB beta | 58 | 3 |
PKC alpha | 27 | 0 |
PKC zeta | 50 | 5 |
PKD1 | 48 | 5 |
PLK1 | 98 | 7 |
PRAK | 37 | 6 |
PRK2 |
1
|
1 |
ROCK 2 |
6
|
0 |
RSK1 | 12 | 0 |
RSK2 | 19 | 1 |
S6K1 | 13 | 1 |
SGK1 | 59 | 4 |
SmMLCK | 31 | 0 |
Src | 100 | 1 |
SRPK1 | 92 | 1 |