Inhibitor | ML-7, Hydrochloride  

Compound name Brutto MW CAS PubChem CID Action Reference Reference
ML-7, Hydrochloride   C15H17IN2O2S • HCl 452.70 110448-33-4 9803932 MLCK Krarup T. (1998) Am. J. Physiol. 275 C239 Saitoh M. (1987) J. Biol. Chem. 262 7796

Screening Results Chart

Screening Results Tables

Screen Conc: 2.00µM
Kinase % Activity Remaining Standard Deviation
AMPK 92 12
Aurora B 82 1
CAMK1 88 6
CDK2-Cyclin A 113 2
CHK1 86 0
CHK2 86 11
CK1 delta 80 7
CK2 101 6
CSK 81 0
DYRK1A 88 12
EF2K 102 6
ERK2 106 6
ERK8 95 3
GSK3 beta 86 5
IKK beta 96 3
JNK1 98 0
JNK3 92 4
Lck 90 8
MAPKAP-K2 101 4
MAPKAP-K3 104 4
MARK3 103 3
MKK1 97 0
MNK1 79 4
MNK2 92 0
MSK1 88 6
MST2 89 9
NEK2a 86 0
NEK6 96 1
NEK7 94 17
p38 alpha MAPK 82 16
p38 beta MAPK 88 1
p38 delta MAPK 93 2
p38 gamma MAPK 100 0
PDK1 82 7
PHK 89 9
PIM2 66 3
PKA 108 3
PKB alpha 101 2
PKB beta 93 5
PKC alpha 80 1
PKD1 101 9
PLK1 107 14
PRAK 91 11
PRK2 57 8
ROCK 2 80 7
RSK1 85 5
RSK2 97 10
S6K1 77 1
SGK1 90 10
SmMLCK 46 2
Src 87 4
SRPK1 97 18
Screen Conc: 20.00µM
Kinase % Activity Remaining Standard Deviation
AMPK 78 4
Aurora B 82 1
Aurora C 66 1
BRSK2 22 4
CAMK1 47 0
CAMKK alpha 82 2
CAMKK beta 91 2
CDK2-Cyclin A 67 5
CHK1 99 0
CHK2 111 4
CK1 delta 85 5
CK2 37 7
CSK 90 7
DYRK1A 54 0
DYRK2 88 2
DYRK3 54 2
EF2K 104 1
ERK1 109 1
ERK2 88 1
ERK8 61 1
GSK3 beta 78 1
HIPK2 41 5
HIPK3 76 2
IKK beta 45 1
JNK1 103 1
JNK2 86 6
JNK3 86 0
Lck 91 0
MAPKAP-K2 56 4
MAPKAP-K3 103 4
MARK3 129 5
MELK 70 2
MKK1 111 9
MNK1 55 6
MNK2 74 0
MSK1 49 1
MST2 90 1
NEK2a 88 1
NEK6 103 5
NEK7 106 0
p38 alpha MAPK 78 1
p38 beta MAPK 87 1
p38 delta MAPK 60 1
p38 gamma MAPK 87 3
PAK4 89 2
PAK5 103 3
PAK6 98 6
PDK1 96 0
PHK 55 0
PIM1 11 0
PIM2 37 5
PIM3
7
0
PKA 52 2
PKB alpha 77 5
PKB beta 77 7
PKC alpha 76 2
PKC zeta 60 3
PKD1 75 1
PLK1 100 0
PRAK 55 8
PRK2 16 0
ROCK 2 54 3
RSK1 64 1
RSK2 73 5
S6K1 50 0
SGK1 95 6
SmMLCK 12 0
Src 98 8
SRPK1 98 5