Inhibitor | LY294002  

Screen Conc: 5.00µM

Kinase	% Activity Remaining	Standard Deviation
AMPK	105	0
Aurora B	83	9
Aurora C	86	13
BRSK2	110	9
CAMK1	96	5
CAMKK beta	74	7
CDK2-Cyclin A	44	1
CHK1	97	5
CHK2	81	0
CK1 delta	78	0
CK2	40	7
CSK	118	10
DYRK1A	91	4
DYRK2	95	7
DYRK3	69	5
EF2K	114	1
EPH-A2	142	1
ERK1	80	2
ERK2	93	3
ERK8	87	5
FGF-R1	94	10
GSK3 beta	56	3
HIPK2	43	9
HIPK3	93	4
IKK beta	68	4
IKK epsilon	96	2
IRR	72	0
JNK1	119	1
JNK2	105	1
JNK3	100	6
Lck	103	6
MAPKAP-K2	117	0
MAPKAP-K3	120	1
MARK3	66	0
MELK	103	4
MKK1	86	4
MNK1	87	6
MNK2	108	3
MSK1	101	8
MST2	92	7
MST4	78	10
NEK2a	90	12
NEK6	97	7
NEK7	90	0
p38 alpha MAPK	112	13
p38 beta MAPK	97	10
p38 delta MAPK	112	6
p38 gamma MAPK	95	4
PAK4	84	5
PAK5	107	15
PAK6	104	6
PDK1	92	2
PHK	99	3
PIM1	11	1
PIM2	94	3
PIM3	19	0
PKA	102	6
PKB alpha	111	10
PKB beta	87	6
PKC alpha	77	4
PKC zeta	102	0
PKD1	87	7
PLK1	21	0
PRAK	81	10
PRK2	74	3
ROCK 2	102	8
RSK1	102	2
RSK2	128	3
S6K1	92	2
SGK1	110	9
SmMLCK	119	8
Src	98	5
SRPK1	111	3
SYK	110	5
TBK1	116	5
YES1	95	2

Screen Conc: 10.00µM

Kinase	% Activity Remaining	Standard Deviation
AMPK	96	7
Aurora B	69	3
Aurora C	84	2
BRSK2	103	4
CAMK1	87	14
CAMKK alpha	71	4
CAMKK beta	71	4
CDK2-Cyclin A	80	1
CHK1	82	12
CHK2	83	0
CK1 delta	56	3
CK2	23	5
CSK	103	2
DYRK1A	75	9
DYRK2	94	3
DYRK3	78	2
EF2K	83	3
EPH-A2	94	4
ERK1	85	7
ERK2	88	11
ERK8	69	4
FGF-R1	95	2
GSK3 beta	37	3
HIPK2	38	1
HIPK3	77	2
IKK beta	67	4
IKK epsilon	100	3
IRR	55	8
JNK1	92	5
JNK2	97	2
JNK3	86	2
Lck	96	2
MAPKAP-K2	102	3
MAPKAP-K3	119	4
MARK3	79	13
MELK	85	8
MKK1	85	0
MNK1	77	5
MNK2	94	4
MSK1	103	0
MST2	84	0
MST4	90	1
NEK2a	90	8
NEK6	103	4
NEK7	86	0
p38 alpha MAPK	101	10
p38 beta MAPK	100	5
p38 delta MAPK	101	13
p38 gamma MAPK	89	3
PAK4	67	4
PAK5	92	5
PAK6	99	0
PDK1	88	2
PHK	94	9
PIM1	8	1
PIM2	65	1
PIM3	13	2
PKA	97	0
PKB alpha	95	3
PKB beta	81	8
PKC alpha	76	6
PKC zeta	114	5
PKD1	105	2
PLK1	26	0
PRAK	83	6
PRK2	74	7
ROCK 2	89	10
RSK1	92	3
RSK2	103	4
S6K1	90	2
SGK1	104	4
SmMLCK	88	7
Src	105	10
SRPK1	100	5
SYK	115	9
TBK1	102	4
YES1	90	3

Screen Conc: 50.00µM

Kinase	% Activity Remaining	Standard Deviation
AMPK	85	2
Aurora B	68	7
Aurora C	72	3
BRSK2	44	1
CAMK1	72	1
CAMKK alpha	63	1
CAMKK beta	49	5
CDK2-Cyclin A	60	1
CHK1	79	0
CHK2	103	2
CK1 delta	32	0
CK2	2	3
CSK	60	1
DYRK1A	24	2
DYRK2	79	5
DYRK3	39	1
EF2K	44	4
ERK1	88	1
ERK2	89	7
ERK8	41	2
GSK3 beta	8	0
HIPK2	7	0
HIPK3	25	1
IKK beta	45	1
JNK1	91	1
JNK2	83	1
JNK3	80	0
Lck	40	3
MAPKAP-K2	84	7
MAPKAP-K3	88	1
MARK3	82	0
MELK	52	4
MKK1	78	0
MNK1	77	2
MNK2	81	1
MSK1	72	1
MST2	61	1
NEK2a	73	4
NEK6	69	1
NEK7	80	8
p38 alpha MAPK	94	5
p38 beta MAPK	109	4
p38 delta MAPK	66	5
p38 gamma MAPK	95	1
PAK4	70	6
PAK5	77	8
PAK6	80	7
PDK1	74	7
PHK	42	5
PIM1	3	1
PIM2	33	5
PIM3	2	0
PKA	60	1
PKB alpha	67	5
PKB beta	77	7
PKC alpha	49	3
PKC zeta	73	8
PKD1	78	0
PLK1	4	0
PRAK	55	2
PRK2	45	0
ROCK 2	84	6
RSK1	36	1
RSK2	57	9
S6K1	76	1
SGK1	67	0
SmMLCK	43	2
Src	81	3
SRPK1	71	1