Inhibitor | KT5720  

Compound name Brutto MW CAS PubChem CID Action Reference Reference
KT5720   C32H31N3O5 537.60 108068-98-0 454202 PKA Simpson CS. Morris BJ. (1995) Neuroscience 68 97-106 Cabell L. Audesirk G. (1993) Int. J. Dev. Neurosci. 11 357

Screening Results Chart

Screening Results Tables

Screen Conc: 1.00µM
Kinase % Activity Remaining Sort descending Standard Deviation
PDK1
3
0
PHK
5
0
PIM3
7
0
PRK2
10
2
PKD1 12 4
MNK2 13 3
Aurora B 14 4
BRSK2 14 2
MELK 14 1
Aurora C 15 0
AMPK 15 2
CHK1 18 1
RSK1 18 0
RSK2 19 6
SGK1 20 0
MKK1 24 2
MST2 26 4
CAMKK beta 27 0
MAPKAP-K2 28 1
MARK3 29 2
PAK4 36 4
JNK1 38 0
DYRK1A 38 8
MSK1 39 1
DYRK3 40 7
PIM1 40 0
JNK3 43 0
PKA 50 8
SmMLCK 54 5
ERK8 57 2
Lck 59 7
CHK2 59 6
PKC alpha 60 8
CAMKK alpha 60 1
MNK1 61 0
IKK beta 62 7
PAK5 62 7
JNK2 63 1
CDK2-Cyclin A 65 1
DYRK2 66 1
ERK2 66 1
CSK 67 1
PIM2 67 5
p38 gamma MAPK 69 5
SRPK1 69 4
PAK6 70 2
PRAK 71 6
GSK3 beta 76 4
CAMK1 76 6
HIPK2 77 3
Src 78 5
ERK1 79 0
NEK2a 79 4
PLK1 81 0
PKB beta 82 6
CK2 84 1
ROCK 2 85 1
p38 beta MAPK 90 2
PKB alpha 91 4
S6K1 93 9
EF2K 95 0
p38 alpha MAPK 96 4
CK1 delta 97 2
MAPKAP-K3 98 1
NEK6 99 6
NEK7 102 8
PKC zeta 106 3
p38 delta MAPK 111 4
HIPK3 112 0