Inhibitor | KN93  

Screen Conc: 10.00µM

Kinase	% Activity Remaining Sort descending	Standard Deviation
CAMK1	31	1
SmMLCK	39	4
TrkA	41	2
PIM1	53	1
PAK5	60	0
SYK	64	5
IGF-1R	66	11
MST2	66	1
GSK3 beta	70	2
CLK2	70	2
PIM3	71	2
RSK2	76	8
YES1	76	12
Aurora B	76	1
CAMKK beta	76	9
TAK1	76	13
MKK2	77	3
AMPK	77	1
VEGFR1	77	4
MAPKAP-K3	78	6
PRK2	78	3
MELK	79	4
EPH-B3	79	0
IRAK4	79	12
FGF-R1	80	4
DYRK2	81	10
DYRK1A	82	1
MARK1	82	11
DAPK1	82	9
EPH-A2	83	1
PKB beta	83	1
MLK3	83	12
PRAK	83	5
BRSK1	83	2
MSK1	84	4
LKB1	85	2
IKK epsilon	85	8
CHK1	85	1
p38 delta MAPK	86	3
TAO1	87	5
CSK	87	2
NUAK1	87	7
Lck	87	2
SGK1	87	2
PAK2	87	5
MLK1	88	1
MAPKAP-K2	88	0
JNK1	88	11
MARK2	88	1
PKB alpha	89	6
BTK	89	3
TTK	89	9
IKK beta	89	1
p38 beta MAPK	89	4
PKC alpha	89	3
PKD1	89	9
HER4	90	1
EPH-B2	90	12
TBK1	90	3
SRPK1	91	1
JNK2	91	4
DYRK3	91	13
PIM2	91	1
EF2K	92	12
NEK2a	92	1
MINK1	92	0
MKK1	94	4
Src	94	13
RIPK2	94	1
p38 alpha MAPK	94	6
MKK6	95	1
BRSK2	95	3
GCK	96	3
PLK1	96	5
PAK4	96	1
S6K1	96	0
EPH-B4	96	6
ERK8	97	7
JNK3	97	2
ROCK 2	97	8
Aurora A	98	8
IR	98	10
PKA	98	2
MEKK1	98	5
PDK1	99	7
EPH-A4	100	6
HIPK2	100	9
PAK6	100	13
CK1 delta	101	8
MNK2	101	1
ERK1	101	1
HIPK1	101	3
EPH-B1	101	3
JAK2	101	9
IRR	101	3
MARK4	101	4
ASK1	103	14
NEK6	103	13
MARK3	103	10
p38 gamma MAPK	104	3
MNK1	106	0
MST4	106	12
PKC zeta	107	1
CHK2	108	2
RSK1	108	10
CDK2-Cyclin A	108	14
HIPK3	108	12
ERK2	109	12
PHK	113	9
CK2	117	13

Screen Conc: 1.00µM

Kinase	% Activity Remaining Sort descending	Standard Deviation
PRK2	82	5
Aurora B	83	5
CAMKK beta	83	3
MARK2	84	7
CLK2	86	7
PIM1	86	6
CAMK1	86	6
SmMLCK	86	1
CHK1	86	1
TBK1	87	5
PIM3	87	9
ERK2	87	8
AMPK	88	4
LKB1	89	2
MAPKAP-K3	89	5
IGF-1R	89	12
TAK1	90	2
HIPK3	91	2
BTK	91	4
PLK1	92	1
YES1	92	8
PAK5	92	3
IKK epsilon	92	3
p38 delta MAPK	93	7
PAK6	93	1
IRAK4	93	0
MKK2	93	0
BRSK2	93	11
MEKK1	93	2
EPH-A2	93	2
VEGFR1	94	6
FGF-R1	94	1
HER4	94	1
JNK1	94	2
MARK1	95	1
ROCK 2	95	8
JNK3	96	5
RSK2	96	14
TTK	96	1
MELK	96	15
MLK3	96	1
p38 beta MAPK	97	5
PDK1	97	5
IR	97	11
S6K1	97	2
TrkA	97	3
CK1 delta	98	7
PKC alpha	98	3
EPH-B3	98	5
ERK8	98	6
MAPKAP-K2	98	6
GSK3 beta	99	3
PKD1	99	7
MNK1	100	8
JNK2	101	14
TAO1	101	3
EPH-B1	101	2
PAK2	101	8
EPH-B4	101	8
Lck	102	5
p38 gamma MAPK	102	14
PRAK	102	1
SGK1	102	2
SRPK1	102	13
HIPK1	102	2
PAK4	103	14
JAK2	103	2
MARK4	103	1
PIM2	103	10
Src	103	3
EPH-A4	104	2
DYRK2	104	5
NEK6	104	2
PKB alpha	104	2
NUAK1	104	11
HIPK2	105	2
DAPK1	105	8
ASK1	106	4
Aurora A	106	4
IKK beta	106	15
IRR	106	3
EF2K	106	9
CSK	107	12
MSK1	107	2
MKK6	107	7
SYK	108	5
MLK1	108	2
DYRK3	109	10
NEK2a	109	6
BRSK1	109	1
DYRK1A	110	6
MARK3	110	10
MINK1	110	7
CHK2	111	8
MST4	111	4
MKK1	111	5
PKA	111	7
p38 alpha MAPK	112	2
PKC zeta	113	2
EPH-B2	113	5
RIPK2	113	0
GCK	113	2
PKB beta	114	2
PHK	114	2
CK2	115	5
MST2	115	2
RSK1	117	14
ERK1	117	2
MNK2	118	3
CDK2-Cyclin A	120	3