Inhibitor | KN93  

Screen Conc: 1.00µM

Kinase	% Activity Remaining	Standard Deviation
AMPK	88	4
ASK1	106	4
Aurora A	106	4
Aurora B	83	5
BRSK1	109	1
BRSK2	93	11
BTK	91	4
CAMK1	86	6
CAMKK beta	83	3
CDK2-Cyclin A	120	3
CHK1	86	1
CHK2	111	8
CK1 delta	98	7
CK2	115	5
CLK2	86	7
CSK	107	12
DAPK1	105	8
DYRK1A	110	6
DYRK2	104	5
DYRK3	109	10
EF2K	106	9
EPH-A2	93	2
EPH-A4	104	2
EPH-B1	101	2
EPH-B2	113	5
EPH-B3	98	5
EPH-B4	101	8
ERK1	117	2
ERK2	87	8
ERK8	98	6
FGF-R1	94	1
GCK	113	2
GSK3 beta	99	3
HER4	94	1
HIPK1	102	2
HIPK2	105	2
HIPK3	91	2
IGF-1R	89	12
IKK beta	106	15
IKK epsilon	92	3
IR	97	11
IRAK4	93	0
IRR	106	3
JAK2	103	2
JNK1	94	2
JNK2	101	14
JNK3	96	5
Lck	102	5
LKB1	89	2
MAPKAP-K2	98	6
MAPKAP-K3	89	5
MARK1	95	1
MARK2	84	7
MARK3	110	10
MARK4	103	1
MEKK1	93	2
MELK	96	15
MINK1	110	7
MKK1	111	5
MKK2	93	0
MKK6	107	7
MLK1	108	2
MLK3	96	1
MNK1	100	8
MNK2	118	3
MSK1	107	2
MST2	115	2
MST4	111	4
NEK2a	109	6
NEK6	104	2
NUAK1	104	11
p38 alpha MAPK	112	2
p38 beta MAPK	97	5
p38 delta MAPK	93	7
p38 gamma MAPK	102	14
PAK2	101	8
PAK4	103	14
PAK5	92	3
PAK6	93	1
PDK1	97	5
PHK	114	2
PIM1	86	6
PIM2	103	10
PIM3	87	9
PKA	111	7
PKB alpha	104	2
PKB beta	114	2
PKC alpha	98	3
PKC zeta	113	2
PKD1	99	7
PLK1	92	1
PRAK	102	1
PRK2	82	5
RIPK2	113	0
ROCK 2	95	8
RSK1	117	14
RSK2	96	14
S6K1	97	2
SGK1	102	2
SmMLCK	86	1
Src	103	3
SRPK1	102	13
SYK	108	5
TAK1	90	2
TAO1	101	3
TBK1	87	5
TrkA	97	3
TTK	96	1
VEGFR1	94	6
YES1	92	8

Screen Conc: 10.00µM

Kinase	% Activity Remaining	Standard Deviation
AMPK	77	1
ASK1	103	14
Aurora A	98	8
Aurora B	76	1
BRSK1	83	2
BRSK2	95	3
BTK	89	3
CAMK1	31	1
CAMKK beta	76	9
CDK2-Cyclin A	108	14
CHK1	85	1
CHK2	108	2
CK1 delta	101	8
CK2	117	13
CLK2	70	2
CSK	87	2
DAPK1	82	9
DYRK1A	82	1
DYRK2	81	10
DYRK3	91	13
EF2K	92	12
EPH-A2	83	1
EPH-A4	100	6
EPH-B1	101	3
EPH-B2	90	12
EPH-B3	79	0
EPH-B4	96	6
ERK1	101	1
ERK2	109	12
ERK8	97	7
FGF-R1	80	4
GCK	96	3
GSK3 beta	70	2
HER4	90	1
HIPK1	101	3
HIPK2	100	9
HIPK3	108	12
IGF-1R	66	11
IKK beta	89	1
IKK epsilon	85	8
IR	98	10
IRAK4	79	12
IRR	101	3
JAK2	101	9
JNK1	88	11
JNK2	91	4
JNK3	97	2
Lck	87	2
LKB1	85	2
MAPKAP-K2	88	0
MAPKAP-K3	78	6
MARK1	82	11
MARK2	88	1
MARK3	103	10
MARK4	101	4
MEKK1	98	5
MELK	79	4
MINK1	92	0
MKK1	94	4
MKK2	77	3
MKK6	95	1
MLK1	88	1
MLK3	83	12
MNK1	106	0
MNK2	101	1
MSK1	84	4
MST2	66	1
MST4	106	12
NEK2a	92	1
NEK6	103	13
NUAK1	87	7
p38 alpha MAPK	94	6
p38 beta MAPK	89	4
p38 delta MAPK	86	3
p38 gamma MAPK	104	3
PAK2	87	5
PAK4	96	1
PAK5	60	0
PAK6	100	13
PDK1	99	7
PHK	113	9
PIM1	53	1
PIM2	91	1
PIM3	71	2
PKA	98	2
PKB alpha	89	6
PKB beta	83	1
PKC alpha	89	3
PKC zeta	107	1
PKD1	89	9
PLK1	96	5
PRAK	83	5
PRK2	78	3
RIPK2	94	1
ROCK 2	97	8
RSK1	108	10
RSK2	76	8
S6K1	96	0
SGK1	87	2
SmMLCK	39	4
Src	94	13
SRPK1	91	1
SYK	64	5
TAK1	76	13
TAO1	87	5
TBK1	90	3
TrkA	41	2
TTK	89	9
VEGFR1	77	4
YES1	76	12