Inhibitor | KN62  

Compound name Brutto MW CAS PubChem CID Action Reference Reference
KN62   C38H35N5O6S2 721.90 127191-97-3 5312126 CaMKII Minami H. (1994) Biochem. Biophys. Res. Commun. 199 241

Screening Results Chart

Screening Results Tables

Screen Conc: 10.00µM
Kinase % Activity Remaining Sort descending Standard Deviation
Lck 30 0
CAMK1 38 4
DYRK1A 38 7
PRAK 45 1
PIM1 53 0
MAPKAP-K2 56 4
GSK3 beta 58 3
RSK2 60 2
PIM3 61 2
S6K1 61 1
IKK beta 63 2
SRPK1 70 2
MAPKAP-K3 74 5
NEK6 74 2
PKB alpha 75 0
SGK1 75 1
PKA 76 2
MELK 76 7
DYRK2 76 0
JNK3 79 0
CSK 79 0
SmMLCK 80 1
MSK1 81 1
DYRK3 81 1
PKB beta 83 5
p38 beta MAPK 84 2
CAMKK alpha 85 6
PIM2 87 1
ROCK 2 87 1
PRK2 87 4
PKD1 87 0
PHK 87 1
CAMKK beta 88 0
Aurora B 89 1
JNK2 89 2
PAK4 89 8
MARK3 90 6
p38 delta MAPK 90 9
NEK2a 90 8
Aurora C 91 1
p38 alpha MAPK 91 3
NEK7 91 3
ERK2 92 3
PKC alpha 93 5
CK1 delta 93 8
MKK1 93 8
Src 94 4
PLK1 95 2
BRSK2 96 5
PKC zeta 99 2
HIPK2 99 3
ERK8 99 1
PDK1 99 0
MNK2 101 1
MST2 102 3
p38 gamma MAPK 102 1
ERK1 102 6
MNK1 103 5
PAK5 104 3
CK2 105 3
CDK2-Cyclin A 105 8
HIPK3 107 6
JNK1 110 2
PAK6 113 2
AMPK 115 1
RSK1 116 3
CHK1 120 11
CHK2 123 1
EF2K 130 1