| Compound name | Brutto | MW | CAS | PubChem CID | Action | Reference | Reference |
|---|---|---|---|---|---|---|---|
| KN62 | C38H35N5O6S2 | 721.90 | 127191-97-3 | 5312126 | CaMKII | Minami H. (1994) Biochem. Biophys. Res. Commun. 199 241 |
| Kinase | % Activity Remaining | Standard Deviation |
|---|---|---|
| AMPK | 115 | 1 |
| Aurora B | 89 | 1 |
| Aurora C | 91 | 1 |
| BRSK2 | 96 | 5 |
| CAMK1 | 38 | 4 |
| CAMKK alpha | 85 | 6 |
| CAMKK beta | 88 | 0 |
| CDK2-Cyclin A | 105 | 8 |
| CHK1 | 120 | 11 |
| CHK2 | 123 | 1 |
| CK1 delta | 93 | 8 |
| CK2 | 105 | 3 |
| CSK | 79 | 0 |
| DYRK1A | 38 | 7 |
| DYRK2 | 76 | 0 |
| DYRK3 | 81 | 1 |
| EF2K | 130 | 1 |
| ERK1 | 102 | 6 |
| ERK2 | 92 | 3 |
| ERK8 | 99 | 1 |
| GSK3 beta | 58 | 3 |
| HIPK2 | 99 | 3 |
| HIPK3 | 107 | 6 |
| IKK beta | 63 | 2 |
| JNK1 | 110 | 2 |
| JNK2 | 89 | 2 |
| JNK3 | 79 | 0 |
| Lck | 30 | 0 |
| MAPKAP-K2 | 56 | 4 |
| MAPKAP-K3 | 74 | 5 |
| MARK3 | 90 | 6 |
| MELK | 76 | 7 |
| MKK1 | 93 | 8 |
| MNK1 | 103 | 5 |
| MNK2 | 101 | 1 |
| MSK1 | 81 | 1 |
| MST2 | 102 | 3 |
| NEK2a | 90 | 8 |
| NEK6 | 74 | 2 |
| NEK7 | 91 | 3 |
| p38 alpha MAPK | 91 | 3 |
| p38 beta MAPK | 84 | 2 |
| p38 delta MAPK | 90 | 9 |
| p38 gamma MAPK | 102 | 1 |
| PAK4 | 89 | 8 |
| PAK5 | 104 | 3 |
| PAK6 | 113 | 2 |
| PDK1 | 99 | 0 |
| PHK | 87 | 1 |
| PIM1 | 53 | 0 |
| PIM2 | 87 | 1 |
| PIM3 | 61 | 2 |
| PKA | 76 | 2 |
| PKB alpha | 75 | 0 |
| PKB beta | 83 | 5 |
| PKC alpha | 93 | 5 |
| PKC zeta | 99 | 2 |
| PKD1 | 87 | 0 |
| PLK1 | 95 | 2 |
| PRAK | 45 | 1 |
| PRK2 | 87 | 4 |
| ROCK 2 | 87 | 1 |
| RSK1 | 116 | 3 |
| RSK2 | 60 | 2 |
| S6K1 | 61 | 1 |
| SGK1 | 75 | 1 |
| SmMLCK | 80 | 1 |
| Src | 94 | 4 |
| SRPK1 | 70 | 2 |