

Compound name | Brutto | MW | CAS | PubChem CID | Action | Reference | Reference |
---|---|---|---|---|---|---|---|
KN62 | C38H35N5O6S2 | 721.90 | 127191-97-3 | 5312126 | CaMKII | Minami H. (1994) Biochem. Biophys. Res. Commun. 199 241 |
Kinase | % Activity Remaining | Standard Deviation |
---|---|---|
AMPK | 115 | 1 |
Aurora B | 89 | 1 |
Aurora C | 91 | 1 |
BRSK2 | 96 | 5 |
CAMK1 | 38 | 4 |
CAMKK alpha | 85 | 6 |
CAMKK beta | 88 | 0 |
CDK2-Cyclin A | 105 | 8 |
CHK1 | 120 | 11 |
CHK2 | 123 | 1 |
CK1 delta | 93 | 8 |
CK2 | 105 | 3 |
CSK | 79 | 0 |
DYRK1A | 38 | 7 |
DYRK2 | 76 | 0 |
DYRK3 | 81 | 1 |
EF2K | 130 | 1 |
ERK1 | 102 | 6 |
ERK2 | 92 | 3 |
ERK8 | 99 | 1 |
GSK3 beta | 58 | 3 |
HIPK2 | 99 | 3 |
HIPK3 | 107 | 6 |
IKK beta | 63 | 2 |
JNK1 | 110 | 2 |
JNK2 | 89 | 2 |
JNK3 | 79 | 0 |
Lck | 30 | 0 |
MAPKAP-K2 | 56 | 4 |
MAPKAP-K3 | 74 | 5 |
MARK3 | 90 | 6 |
MELK | 76 | 7 |
MKK1 | 93 | 8 |
MNK1 | 103 | 5 |
MNK2 | 101 | 1 |
MSK1 | 81 | 1 |
MST2 | 102 | 3 |
NEK2a | 90 | 8 |
NEK6 | 74 | 2 |
NEK7 | 91 | 3 |
p38 alpha MAPK | 91 | 3 |
p38 beta MAPK | 84 | 2 |
p38 delta MAPK | 90 | 9 |
p38 gamma MAPK | 102 | 1 |
PAK4 | 89 | 8 |
PAK5 | 104 | 3 |
PAK6 | 113 | 2 |
PDK1 | 99 | 0 |
PHK | 87 | 1 |
PIM1 | 53 | 0 |
PIM2 | 87 | 1 |
PIM3 | 61 | 2 |
PKA | 76 | 2 |
PKB alpha | 75 | 0 |
PKB beta | 83 | 5 |
PKC alpha | 93 | 5 |
PKC zeta | 99 | 2 |
PKD1 | 87 | 0 |
PLK1 | 95 | 2 |
PRAK | 45 | 1 |
PRK2 | 87 | 4 |
ROCK 2 | 87 | 1 |
RSK1 | 116 | 3 |
RSK2 | 60 | 2 |
S6K1 | 61 | 1 |
SGK1 | 75 | 1 |
SmMLCK | 80 | 1 |
Src | 94 | 4 |
SRPK1 | 70 | 2 |