Inhibitor | KN62  

Compound name Brutto MW CAS PubChem CID Action Reference Reference
KN62   C38H35N5O6S2 721.90 127191-97-3 5312126 CaMKII Minami H. (1994) Biochem. Biophys. Res. Commun. 199 241

Screening Results Chart

Screening Results Tables

Screen Conc: 10.00µM
Kinase % Activity Remaining Standard Deviation
AMPK 115 1
Aurora B 89 1
Aurora C 91 1
BRSK2 96 5
CAMK1 38 4
CAMKK alpha 85 6
CAMKK beta 88 0
CDK2-Cyclin A 105 8
CHK1 120 11
CHK2 123 1
CK1 delta 93 8
CK2 105 3
CSK 79 0
DYRK1A 38 7
DYRK2 76 0
DYRK3 81 1
EF2K 130 1
ERK1 102 6
ERK2 92 3
ERK8 99 1
GSK3 beta 58 3
HIPK2 99 3
HIPK3 107 6
IKK beta 63 2
JNK1 110 2
JNK2 89 2
JNK3 79 0
Lck 30 0
MAPKAP-K2 56 4
MAPKAP-K3 74 5
MARK3 90 6
MELK 76 7
MKK1 93 8
MNK1 103 5
MNK2 101 1
MSK1 81 1
MST2 102 3
NEK2a 90 8
NEK6 74 2
NEK7 91 3
p38 alpha MAPK 91 3
p38 beta MAPK 84 2
p38 delta MAPK 90 9
p38 gamma MAPK 102 1
PAK4 89 8
PAK5 104 3
PAK6 113 2
PDK1 99 0
PHK 87 1
PIM1 53 0
PIM2 87 1
PIM3 61 2
PKA 76 2
PKB alpha 75 0
PKB beta 83 5
PKC alpha 93 5
PKC zeta 99 2
PKD1 87 0
PLK1 95 2
PRAK 45 1
PRK2 87 4
ROCK 2 87 1
RSK1 116 3
RSK2 60 2
S6K1 61 1
SGK1 75 1
SmMLCK 80 1
Src 94 4
SRPK1 70 2