| Compound name | Brutto | MW | CAS | PubChem CID | Action | Reference | Reference |
|---|---|---|---|---|---|---|---|
| IC261 | C18H17NO4 | 311.30 | 186611-52-9 | 5288600 | CK1 | Behrend L. (2000) Oncogene 19 5303 | Mashhoon N. (2000) J. Biol. Chem. 275 20052 |
| Kinase | % Activity Remaining Sort descending | Standard Deviation |
|---|---|---|
| CK1 delta |
9
|
2 |
| PIM3 | 41 | 1 |
| PIM1 | 43 | 1 |
| Lck | 49 | 4 |
| CAMK1 | 55 | 5 |
| PKD1 | 62 | 3 |
| CAMKK alpha | 67 | 4 |
| ERK8 | 68 | 2 |
| MST2 | 70 | 1 |
| SmMLCK | 70 | 2 |
| Src | 70 | 4 |
| AMPK | 71 | 2 |
| DYRK1A | 73 | 1 |
| GSK3 beta | 74 | 6 |
| Aurora B | 75 | 3 |
| PIM2 | 75 | 1 |
| MELK | 75 | 8 |
| NEK2a | 75 | 6 |
| PAK6 | 76 | 0 |
| CHK2 | 76 | 4 |
| ROCK 2 | 78 | 0 |
| MNK1 | 79 | 3 |
| SGK1 | 79 | 4 |
| PKC zeta | 80 | 4 |
| CSK | 81 | 4 |
| PRAK | 82 | 5 |
| PKA | 82 | 3 |
| CDK2-Cyclin A | 83 | 4 |
| PAK4 | 84 | 2 |
| PAK5 | 84 | 1 |
| S6K1 | 84 | 2 |
| CAMKK beta | 86 | 2 |
| PHK | 86 | 1 |
| MKK1 | 86 | 2 |
| RSK1 | 87 | 3 |
| PRK2 | 87 | 5 |
| MSK1 | 88 | 1 |
| MAPKAP-K2 | 88 | 4 |
| MARK3 | 88 | 5 |
| BRSK2 | 88 | 4 |
| RSK2 | 89 | 1 |
| DYRK3 | 89 | 3 |
| PDK1 | 89 | 5 |
| IKK beta | 90 | 4 |
| PKB beta | 90 | 3 |
| PKC alpha | 90 | 2 |
| ERK1 | 91 | 6 |
| p38 alpha MAPK | 91 | 4 |
| p38 delta MAPK | 91 | 4 |
| p38 gamma MAPK | 92 | 4 |
| ERK2 | 93 | 4 |
| JNK3 | 93 | 4 |
| PLK1 | 94 | 0 |
| JNK1 | 94 | 2 |
| Aurora C | 94 | 3 |
| MAPKAP-K3 | 94 | 3 |
| PKB alpha | 94 | 5 |
| SRPK1 | 95 | 1 |
| HIPK3 | 95 | 3 |
| NEK6 | 95 | 5 |
| p38 beta MAPK | 96 | 7 |
| HIPK2 | 96 | 6 |
| MNK2 | 97 | 5 |
| CK2 | 97 | 2 |
| DYRK2 | 99 | 6 |
| CHK1 | 99 | 2 |
| EF2K | 100 | 4 |
| JNK2 | 101 | 3 |
| NEK7 | 103 | 4 |