Inhibitor | Harmine  

Screen Conc: 1.00µM

Kinase	% Activity Remaining	Standard Deviation
AMPK	83	16
Aurora B	82	1
Aurora C	83	1
BRSK2	107	8
BTK	91	5
CAMK1	100	3
CAMKK alpha	87	1
CAMKK beta	96	6
CDK2-Cyclin A	81	8
CHK1	88	3
CHK2	69	0
CK1 delta	82	9
CK2	89	18
CSK	109	10
DYRK1A	9	0
DYRK2	28	3
DYRK3	33	9
EF2K	102	9
EPH-A2	101	0
EPH-B3	105	15
ERK1	107	44
ERK2	89	7
ERK8	77	11
FGF-R1	105	8
GSK3 beta	95	15
HIPK2	69	6
HIPK3	87	7
IGF-1R	104	4
IKK beta	105	4
IKK epsilon	92	11
IR	105	4
IRR	37	0
JNK1	100	14
JNK2	92	10
JNK3	77	0
Lck	96	16
MAPKAP-K2	87	8
MAPKAP-K3	97	5
MARK3	112	17
MELK	79	8
MKK1	98	1
MNK1	81	2
MNK2	84	7
MSK1	90	3
MST2	93	2
MST4	97	5
NEK2a	96	4
NEK6	91	8
NEK7	107	1
p38 alpha MAPK	89	1
p38 beta MAPK	106	23
p38 delta MAPK	111	0
p38 gamma MAPK	89	10
PAK4	82	10
PAK5	117	5
PAK6	106	4
PDK1	101	7
PHK	95	13
PIM1	84	0
PIM2	113	10
PIM3	79	6
PKA	94	4
PKB alpha	91	7
PKB beta	103	8
PKC alpha	105	5
PKC zeta	103	13
PKD1	83	2
PLK1	103	4
PRAK	91	3
PRK2	91	9
ROCK 2	97	7
RSK1	114	13
RSK2	91	2
S6K1	93	1
SGK1	90	3
SmMLCK	85	2
Src	83	5
SRPK1	82	12
SYK	91	34
TBK1	98	1
VEGFR1	108	0
YES1	87	16

Screen Conc: 10.00µM

Kinase	% Activity Remaining	Standard Deviation
AMPK	72	1
Aurora B	81	2
Aurora C	83	1
BRSK2	83	3
BTK	84	10
CAMK1	94	4
CAMKK alpha	95	4
CAMKK beta	81	1
CDK2-Cyclin A	86	4
CHK1	99	9
CHK2	100	0
CK1 delta	60	4
CK2	68	5
CSK	86	3
DYRK1A	2	2
DYRK2	15	0
DYRK3	6	0
EF2K	104	8
EPH-A2	107	0
EPH-B3	105	21
ERK1	95	5
ERK2	95	5
ERK8	80	1
FGF-R1	120	26
GSK3 beta	87	0
HIPK2	108	7
HIPK3	87	8
IGF-1R	106	42
IKK beta	73	9
IKK epsilon	87	15
IR	100	2
IRR	33	10
JNK1	89	3
JNK2	91	5
JNK3	91	0
Lck	81	2
MAPKAP-K2	110	4
MAPKAP-K3	98	6
MARK3	83	3
MELK	80	2
MKK1	73	4
MNK1	82	4
MNK2	80	4
MSK1	83	5
MST2	85	7
MST4	90	1
NEK2a	94	1
NEK6	87	1
NEK7	108	1
p38 alpha MAPK	100	7
p38 beta MAPK	103	4
p38 delta MAPK	88	1
p38 gamma MAPK	80	3
PAK4	96	3
PAK5	92	5
PAK6	83	5
PDK1	87	1
PHK	85	5
PIM1	86	1
PIM2	88	7
PIM3	64	1
PKA	80	9
PKB alpha	101	7
PKB beta	90	1
PKC alpha	82	4
PKC zeta	83	1
PKD1	80	9
PLK1	97	1
PRAK	90	2
PRK2	86	4
ROCK 2	80	4
RSK1	105	6
RSK2	104	3
S6K1	93	3
SGK1	83	1
SmMLCK	87	7
Src	88	9
SRPK1	85	7
SYK	85	16
TBK1	89	1
VEGFR1	95	3
YES1	83	21