Inhibitor | Harmane  

Compound name Brutto MW CAS PubChem CID Action Reference Reference
Harmane   C12H10N2 182.22 486-84-0 5281404 serotonin, monoamine oxidase Smith KL. (2013) J Psychopharmacol. 162-70

Screening Results Chart

Screening Results Tables

Screen Conc: 1.00µM
Kinase % Activity Remaining Standard Deviation
AMPK 111 12
Aurora B 105 2
Aurora C 86 2
BRSK2 100 1
CAMK1 90 3
CAMKK alpha 85 5
CAMKK beta 92 4
CDK2-Cyclin A 102 6
CHK1 98 3
CHK2 91 3
CK1 delta 98 6
CK2 84 7
CSK 81 5
DYRK1A 44 3
DYRK2 83 5
DYRK3 72 3
EF2K 100 3
ERK1 106 0
ERK2 95 6
ERK8 69 0
GSK3 beta 108 1
HIPK2 104 5
HIPK3 104 0
IKK beta 76 8
JNK1 92 3
JNK2 84 5
JNK3 89 2
Lck 93 1
MAPKAP-K2 109 3
MAPKAP-K3 103 6
MARK3 128 3
MELK 82 2
MKK1 90 5
MNK1 82 1
MNK2 111 4
MSK1 90 11
MST2 80 1
NEK2a 78 0
NEK6 90 1
NEK7 104 0
p38 alpha MAPK 74 1
p38 beta MAPK 90 7
p38 delta MAPK 89 1
p38 gamma MAPK 96 9
PAK4 103 5
PAK5 97 8
PAK6 104 3
PDK1 89 7
PHK 102 3
PIM1 93 1
PIM2 85 1
PIM3 80 0
PKA 94 2
PKB alpha 103 2
PKB beta 91 7
PKC alpha 90 5
PKC zeta 89 2
PKD1 87 1
PLK1 80 2
PRAK 84 8
PRK2 84 5
ROCK 2 104 1
RSK1 98 0
RSK2 94 1
S6K1 94 3
SGK1 86 4
SmMLCK 100 3
Src 83 2
SRPK1 80 2