

Compound name | Brutto | MW | CAS | PubChem CID | Action | Reference | Reference |
---|---|---|---|---|---|---|---|
A-769662 | C20H12N2O3S | 360.39 | 844499-71-4 | 54708532 | AMPK Activator | Cool B. (2006) Cell Metabolism 3 403-416 |
Kinase | % Activity Remaining | Standard Deviation |
---|---|---|
AMPK | 135 | 15 |
ASK1 | 140 | 5 |
Aurora A | 93 | 7 |
Aurora B | 53 | 0 |
BRSK1 | 76 | 5 |
BRSK2 | 64 | 4 |
BTK | 52 | 5 |
CAMK1 | 68 | 3 |
CAMKK beta | 87 | 5 |
CDK2-Cyclin A | 100 | 3 |
CHK1 | 69 | 2 |
CHK2 | 79 | 4 |
CK1 delta | 88 | 5 |
CK2 | 110 | 5 |
CLK2 | 81 | 2 |
CSK | 79 | 2 |
DAPK1 | 107 | 1 |
DYRK1A | 75 | 3 |
DYRK2 | 63 | 0 |
DYRK3 | 54 | 6 |
EF2K | 89 | 4 |
EPH-A2 | 82 | 7 |
EPH-A4 | 93 | 1 |
EPH-B1 | 110 | 6 |
EPH-B2 | 93 | 5 |
EPH-B3 | 81 | 11 |
EPH-B4 | 82 | 8 |
ERK1 | 83 | 3 |
ERK2 | 103 | 8 |
ERK8 | 81 | 3 |
FGF-R1 | 109 | 11 |
GCK | 76 | 5 |
GSK3 beta | 80 | 1 |
HER4 | 33 | 7 |
HIPK1 | 74 | 7 |
HIPK2 | 99 | 6 |
HIPK3 | 97 | 1 |
IGF-1R | 94 | 8 |
IKK beta | 86 | 0 |
IKK epsilon | 69 | 4 |
IR | 103 | 1 |
IRAK4 | 82 | 4 |
IRR | 88 | 5 |
JAK2 | 83 | 6 |
JNK1 | 99 | 5 |
JNK2 | 94 | 1 |
JNK3 | 75 | 3 |
Lck | 88 | 5 |
LKB1 | 86 | 3 |
MAPKAP-K2 | 77 | 1 |
MAPKAP-K3 | 57 | 1 |
MARK1 | 59 | 3 |
MARK2 | 64 | 4 |
MARK3 | 78 | 4 |
MARK4 | 92 | 6 |
MEKK1 | 26 | 5 |
MELK | 46 | 1 |
MINK1 | 65 | 6 |
MKK1 | 79 | 1 |
MKK2 | 74 | 3 |
MKK6 | 85 | 15 |
MLK1 | 59 | 4 |
MLK3 | 43 | 6 |
MNK1 | 104 | 2 |
MNK2 | 102 | 3 |
MSK1 | 69 | 3 |
MST2 | 60 | 10 |
MST4 | 74 | 5 |
NEK2a | 73 | 1 |
NEK6 | 104 | 6 |
NUAK1 | 61 | 7 |
p38 alpha MAPK | 97 | 2 |
p38 beta MAPK | 89 | 2 |
p38 delta MAPK | 107 | 7 |
p38 gamma MAPK | 95 | 3 |
PAK2 | 94 | 2 |
PAK4 | 52 | 8 |
PAK5 | 58 | 2 |
PAK6 | 69 | 3 |
PDK1 | 93 | 3 |
PHK | 96 | 0 |
PIM1 | 26 | 2 |
PIM2 | 71 | 5 |
PIM3 | 18 | 1 |
PKA | 89 | 1 |
PKB alpha | 94 | 0 |
PKB beta | 56 | 5 |
PKC alpha | 94 | 6 |
PKC zeta | 96 | 7 |
PKD1 | 62 | 6 |
PLK1 | 88 | 1 |
PRAK | 52 | 4 |
PRK2 | 85 | 8 |
RIPK2 | 110 | 4 |
ROCK 2 | 91 | 2 |
RSK1 | 80 | 7 |
RSK2 | 74 | 4 |
S6K1 | 78 | 1 |
SGK1 | 103 | 1 |
SmMLCK | 76 | 2 |
Src | 44 | 5 |
SRPK1 | 107 | 0 |
SYK | 106 | 0 |
TAK1 | 83 | 3 |
TAO1 | 83 | 4 |
TBK1 | 67 | 8 |
TrkA | 69 | 2 |
TTK | 76 | 2 |
VEGFR1 | 65 | 4 |
YES1 | 96 | 7 |
Kinase | % Activity Remaining | Standard Deviation |
---|---|---|
AMPK | 67 | 3 |
Aurora B | 25 | 2 |
Aurora C | 30 | 4 |
BRSK2 | 63 | 4 |
CAMK1 | 45 | 0 |
CAMKK beta | 48 | 9 |
CDK2-Cyclin A | 84 | 6 |
CHK1 | 98 | 4 |
CHK2 | 52 | 4 |
CK1 delta | 60 | 6 |
CK2 | 95 | 0 |
CSK | 46 | 1 |
DYRK1A | 60 | 10 |
DYRK2 | 84 | 0 |
DYRK3 | 47 | 4 |
EF2K | 73 | 3 |
EPH-A2 | 64 | 6 |
ERK1 | 102 | 3 |
ERK2 | 74 | 2 |
ERK8 | 36 | 4 |
FGF-R1 | 95 | 11 |
GSK3 beta | 17 | 4 |
HIPK2 | 58 | 2 |
HIPK3 | 52 | 2 |
IKK beta | 60 | 0 |
IKK epsilon | 47 | 1 |
IRR | 90 | 4 |
JNK1 | 102 | 3 |
JNK2 | 89 | 10 |
JNK3 | 70 | 4 |
Lck | 58 | 4 |
MAPKAP-K2 | 32 | 2 |
MAPKAP-K3 | 48 | 1 |
MARK3 | 87 | 4 |
MELK | 64 | 5 |
MKK1 | 27 | 10 |
MNK1 | 66 | 4 |
MNK2 | 80 | 4 |
MSK1 | 39 | 4 |
MST2 | 36 | 0 |
MST4 | 57 | 3 |
NEK2a | 52 | 9 |
NEK6 | 94 | 8 |
NEK7 | 102 | 4 |
p38 alpha MAPK | 122 | 12 |
p38 beta MAPK | 84 | 4 |
p38 delta MAPK | 116 | 12 |
p38 gamma MAPK | 80 | 6 |
PAK4 | 38 | 0 |
PAK5 | 50 | 6 |
PAK6 | 92 | 11 |
PDK1 | 81 | 0 |
PHK | 65 | 3 |
PIM1 |
5
|
0 |
PIM2 | 17 | 0 |
PIM3 |
5
|
0 |
PKA | 41 | 10 |
PKB alpha | 62 | 1 |
PKB beta | 37 | 5 |
PKC alpha | 60 | 0 |
PKC zeta | 67 | 6 |
PKD1 | 25 | 12 |
PLK1 | 28 | 1 |
PRAK | 25 | 1 |
PRK2 | 85 | 9 |
ROCK 2 | 49 | 7 |
RSK1 |
9
|
0 |
RSK2 | 27 | 7 |
S6K1 | 66 | 5 |
SGK1 | 54 | 1 |
SmMLCK | 39 | 12 |
Src | 65 | 13 |
SRPK1 | 42 | 8 |
SYK | 36 | 3 |
TBK1 | 55 | 4 |
YES1 | 13 | 2 |
Kinase | % Activity Remaining | Standard Deviation |
---|---|---|
AMPK | 62 | 5 |
ASK1 | 250 | 7 |
Aurora A | 64 | 4 |
Aurora B | 22 | 2 |
BRSK1 | 51 | 4 |
BRSK2 | 28 | 1 |
BTK |
10
|
1 |
CAMK1 |
7
|
1 |
CAMKK beta | 78 | 4 |
CDK2-Cyclin A | 121 | 0 |
CHK1 | 43 | 3 |
CHK2 | 33 | 3 |
CK1 delta | 88 | 4 |
CK2 | 86 | 5 |
CLK2 | 30 | 4 |
CSK | 82 | 10 |
DAPK1 | 83 | 5 |
DYRK1A | 26 | 3 |
DYRK2 | 33 | 2 |
DYRK3 |
6
|
1 |
EF2K | 64 | 5 |
EPH-A2 | 40 | 5 |
EPH-A4 | 64 | 4 |
EPH-B1 | 97 | 4 |
EPH-B2 | 13 | 2 |
EPH-B3 | 55 | 4 |
EPH-B4 | 49 | 4 |
ERK1 | 63 | 11 |
ERK2 | 49 | 10 |
ERK8 | 24 | 4 |
FGF-R1 | 50 | 8 |
GCK | 14 | 2 |
GSK3 beta | 46 | 6 |
HER4 |
8
|
4 |
HIPK1 | 35 | 2 |
HIPK2 | 19 | 3 |
HIPK3 | 43 | 6 |
IGF-1R | 65 | 5 |
IKK beta | 39 | 3 |
IKK epsilon | 12 | 0 |
IR | 69 | 9 |
IRAK4 | 34 | 3 |
IRR | 51 | 6 |
JAK2 | 32 | 1 |
JNK1 | 93 | 8 |
JNK2 | 88 | 1 |
JNK3 | 62 | 11 |
Lck | 58 | 5 |
LKB1 | 65 | 6 |
MAPKAP-K2 | 30 | 4 |
MAPKAP-K3 |
8
|
3 |
MARK1 | 68 | 6 |
MARK2 | 49 | 2 |
MARK3 | 38 | 4 |
MARK4 | 45 | 4 |
MEKK1 |
7
|
0 |
MELK | 21 | 0 |
MINK1 |
5
|
0 |
MKK1 | 29 | 3 |
MKK2 | 19 | 0 |
MKK6 | 84 | 10 |
MLK1 | 18 | 2 |
MLK3 |
4
|
1 |
MNK1 | 93 | 5 |
MNK2 | 86 | 1 |
MSK1 | 42 | 7 |
MST2 | 20 | 0 |
MST4 | 14 | 0 |
NEK2a | 19 | 0 |
NEK6 | 137 | 5 |
NUAK1 |
10
|
0 |
p38 alpha MAPK | 90 | 5 |
p38 beta MAPK | 77 | 3 |
p38 delta MAPK | 124 | 10 |
p38 gamma MAPK | 83 | 6 |
PAK2 | 63 | 8 |
PAK4 | 41 | 2 |
PAK5 | 39 | 1 |
PAK6 | 82 | 8 |
PDK1 | 90 | 2 |
PHK | 73 | 1 |
PIM1 |
7
|
1 |
PIM2 | 18 | 1 |
PIM3 |
7
|
2 |
PKA | 95 | 10 |
PKB alpha | 78 | 2 |
PKB beta | 11 | 2 |
PKC alpha | 90 | 11 |
PKC zeta | 28 | 6 |
PKD1 | 24 | 1 |
PLK1 | 25 | 2 |
PRAK | 15 | 4 |
PRK2 | 59 | 2 |
RIPK2 | 139 | 3 |
ROCK 2 | 75 | 5 |
RSK1 | 12 | 5 |
RSK2 | 13 | 2 |
S6K1 | 38 | 1 |
SGK1 | 48 | 1 |
SmMLCK | 20 | 0 |
Src |
10
|
1 |
SRPK1 | 35 | 1 |
SYK | 42 | 10 |
TAK1 | 72 | 8 |
TAO1 | 18 | 1 |
TBK1 | 29 | 2 |
TrkA | 28 | 4 |
TTK | 48 | 1 |
VEGFR1 | 11 | 2 |
YES1 | 16 | 0 |