Inhibitor | Harmalol  

Compound name Brutto MW CAS PubChem CID Action Reference Reference
Harmalol   C12H12N2O • HCl • 2H2O 272.73 6028-00-8 5353656 serotonin, monoamine oxidase Riba J. (2012) Drug Test. 610-6.

Screening Results Chart

Screening Results Tables

Screen Conc: 1.00µM
Kinase % Activity Remaining Sort descending Standard Deviation
ERK8 62 3
DYRK1A 67 6
DYRK3 71 2
PIM3 71 0
IKK beta 73 1
MELK 76 0
PKB beta 81 1
NEK2a 82 4
PLK1 82 0
RSK2 83 7
CSK 83 6
CHK1 84 5
PRAK 84 2
Src 85 5
SGK1 85 2
DYRK2 86 4
PRK2 86 2
MKK1 86 1
PHK 87 3
PKC zeta 87 0
GSK3 beta 88 3
SRPK1 88 8
MAPKAP-K2 88 1
PKB alpha 88 1
p38 delta MAPK 89 4
PKA 90 3
ROCK 2 90 7
Aurora B 90 7
Aurora C 90 5
MST2 90 3
CAMKK beta 90 1
CK2 90 0
PKC alpha 91 1
PIM1 91 1
PAK6 91 1
PDK1 92 5
Lck 92 1
NEK6 93 1
HIPK3 93 8
CK1 delta 93 9
S6K1 94 8
ERK2 94 5
p38 beta MAPK 95 3
MSK1 95 1
PAK5 95 4
p38 alpha MAPK 96 2
MNK1 97 1
MAPKAP-K3 98 9
BRSK2 98 4
JNK2 99 6
RSK1 99 9
CDK2-Cyclin A 100 1
HIPK2 100 1
PIM2 100 1
EF2K 101 6
CAMK1 101 3
JNK1 102 3
CAMKK alpha 102 1
p38 gamma MAPK 104 1
PAK4 104 6
ERK1 106 0
MNK2 106 5
SmMLCK 107 9
NEK7 108 7
AMPK 109 1
PKD1 110 2
JNK3 112 0
CHK2 121 1
MARK3 131 8