Inhibitor | Harmalol  

Compound name Brutto MW CAS PubChem CID Action Reference Reference
Harmalol   C12H12N2O • HCl • 2H2O 272.73 6028-00-8 5353656 serotonin, monoamine oxidase Riba J. (2012) Drug Test. 610-6.

Screening Results Chart

Screening Results Tables

Screen Conc: 1.00µM
Kinase % Activity Remaining Standard Deviation
AMPK 109 1
Aurora B 90 7
Aurora C 90 5
BRSK2 98 4
CAMK1 101 3
CAMKK alpha 102 1
CAMKK beta 90 1
CDK2-Cyclin A 100 1
CHK1 84 5
CHK2 121 1
CK1 delta 93 9
CK2 90 0
CSK 83 6
DYRK1A 67 6
DYRK2 86 4
DYRK3 71 2
EF2K 101 6
ERK1 106 0
ERK2 94 5
ERK8 62 3
GSK3 beta 88 3
HIPK2 100 1
HIPK3 93 8
IKK beta 73 1
JNK1 102 3
JNK2 99 6
JNK3 112 0
Lck 92 1
MAPKAP-K2 88 1
MAPKAP-K3 98 9
MARK3 131 8
MELK 76 0
MKK1 86 1
MNK1 97 1
MNK2 106 5
MSK1 95 1
MST2 90 3
NEK2a 82 4
NEK6 93 1
NEK7 108 7
p38 alpha MAPK 96 2
p38 beta MAPK 95 3
p38 delta MAPK 89 4
p38 gamma MAPK 104 1
PAK4 104 6
PAK5 95 4
PAK6 91 1
PDK1 92 5
PHK 87 3
PIM1 91 1
PIM2 100 1
PIM3 71 0
PKA 90 3
PKB alpha 88 1
PKB beta 81 1
PKC alpha 91 1
PKC zeta 87 0
PKD1 110 2
PLK1 82 0
PRAK 84 2
PRK2 86 2
ROCK 2 90 7
RSK1 99 9
RSK2 83 7
S6K1 94 8
SGK1 85 2
SmMLCK 107 9
Src 85 5
SRPK1 88 8