Inhibitor | Harmaline  

Compound name Brutto MW CAS PubChem CID Action Reference Reference
Harmaline   C13H14N2O 214.26 304-21-2 5280951 serotonin, monoamine oxidase Herraiz T. (2013) Drug Test. 1002/dta.1530.

Screening Results Chart

Screening Results Tables

Screen Conc: 1.00µM
Kinase % Activity Remaining Sort ascending Standard Deviation
p38 gamma MAPK 119 5
PIM2 117 1
CHK2 116 5
RSK2 112 0
SmMLCK 111 2
MARK3 110 5
RSK1 109 5
NEK7 107 8
PKD1 107 1
EF2K 107 2
ERK1 107 4
AMPK 105 1
PKB beta 105 1
PAK6 105 2
PIM1 104 6
BRSK2 103 1
CAMK1 103 0
MST2 101 0
GSK3 beta 100 9
CDK2-Cyclin A 100 6
Aurora C 99 8
MAPKAP-K3 97 4
HIPK3 97 0
NEK2a 96 6
MELK 95 0
JNK1 95 3
NEK6 94 1
IKK beta 94 4
PKB alpha 94 0
MKK1 94 2
Src 94 5
MSK1 93 1
S6K1 93 1
CHK1 93 4
p38 beta MAPK 92 0
p38 delta MAPK 92 5
MNK2 92 2
CAMKK alpha 92 1
PKC alpha 90 8
PIM3 90 6
HIPK2 90 1
PAK4 90 1
Aurora B 89 4
SRPK1 89 5
MAPKAP-K2 89 4
JNK3 88 0
CAMKK beta 88 7
PKA 88 1
p38 alpha MAPK 87 4
CK2 87 1
ERK2 86 0
JNK2 85 6
PRK2 85 1
PDK1 85 8
SGK1 85 7
PKC zeta 83 2
PAK5 83 6
PHK 83 6
CSK 81 6
Lck 81 1
MNK1 80 0
PLK1 79 1
ROCK 2 78 6
PRAK 73 1
DYRK2 73 1
CK1 delta 65 5
DYRK3 49 5
ERK8 44 4
DYRK1A 29 4