Inhibitor |
H-7, Dihydrochloride
Screening Results Tables
Screen Conc:
10.00µM
Kinase |
% Activity Remaining |
Standard Deviation |
AMPK
|
24
|
0
|
Aurora B
|
75
|
4
|
Aurora C
|
61
|
3
|
BRSK2
|
64
|
2
|
CAMK1
|
64
|
7
|
CAMKK alpha
|
69
|
1
|
CAMKK beta
|
85
|
6
|
CDK2-Cyclin A
|
52
|
2
|
CHK1
|
84
|
6
|
CHK2
|
110
|
2
|
CK1 delta
|
86
|
0
|
CK2
|
89
|
2
|
CSK
|
86
|
5
|
DYRK1A
|
85
|
9
|
DYRK2
|
92
|
3
|
DYRK3
|
63
|
2
|
EF2K
|
87
|
4
|
ERK1
|
105
|
2
|
ERK2
|
92
|
2
|
ERK8
|
84
|
1
|
GSK3 beta
|
64
|
4
|
HIPK2
|
92
|
4
|
HIPK3
|
113
|
1
|
IKK beta
|
71
|
5
|
JNK1
|
90
|
1
|
JNK2
|
85
|
1
|
JNK3
|
85
|
0
|
Lck
|
78
|
2
|
MAPKAP-K2
|
82
|
0
|
MAPKAP-K3
|
105
|
1
|
MARK3
|
93
|
1
|
MELK
|
35
|
3
|
MKK1
|
87
|
2
|
MNK1
|
67
|
4
|
MNK2
|
80
|
0
|
MSK1
|
36
|
4
|
MST2
|
69
|
2
|
NEK2a
|
85
|
1
|
NEK6
|
102
|
8
|
NEK7
|
104
|
2
|
p38 alpha MAPK
|
85
|
2
|
p38 beta MAPK
|
109
|
6
|
p38 delta MAPK
|
82
|
3
|
p38 gamma MAPK
|
97
|
0
|
PAK4
|
106
|
6
|
PAK5
|
101
|
7
|
PAK6
|
105
|
1
|
PDK1
|
78
|
3
|
PHK
|
68
|
7
|
PIM1
|
94
|
11
|
PIM2
|
87
|
2
|
PIM3
|
68
|
0
|
PKA
|
48
|
0
|
PKB alpha
|
100
|
5
|
PKB beta
|
81
|
4
|
PKC alpha
|
48
|
3
|
PKC zeta
|
65
|
4
|
PKD1
|
37
|
3
|
PLK1
|
83
|
2
|
PRAK
|
97
|
0
|
PRK2
|
7
|
1
|
ROCK 2
|
15
|
1
|
RSK1
|
16
|
0
|
RSK2
|
38
|
7
|
S6K1
|
90
|
7
|
SGK1
|
84
|
0
|
SmMLCK
|
86
|
2
|
Src
|
84
|
5
|
SRPK1
|
91
|
0
|