Compound name | Brutto | MW | CAS | PubChem CID | Action | Reference | Reference |
---|---|---|---|---|---|---|---|
Gö 6976 | C24H18N4O | 378.40 | 136194-77-9 | 3501 | PKC | Gschwendt M. (1996) FEBS Lett. 392 77 | Wenzel-Seifert K. (1994) Biochem. Biophys. Res. Commun. 200 1536 |
Kinase | % Activity Remaining | Standard Deviation |
---|---|---|
AMPK | 16 | 3 |
Aurora B | 23 | 0 |
Aurora C | 26 | 3 |
BRSK2 | 48 | 6 |
CAMK1 | 99 | 3 |
CAMKK alpha | 37 | 4 |
CAMKK beta | 16 | 4 |
CDK2-Cyclin A |
10
|
0 |
CHK1 |
1
|
0 |
CHK2 | 53 | 3 |
CK1 delta | 88 | 3 |
CK2 | 88 | 4 |
CSK | 74 | 3 |
DYRK1A | 33 | 6 |
DYRK2 | 60 | 8 |
DYRK3 | 33 | 6 |
EF2K | 109 | 3 |
ERK1 | 60 | 7 |
ERK2 | 46 | 2 |
ERK8 | 36 | 4 |
GSK3 beta | 24 | 4 |
HIPK2 | 27 | 3 |
HIPK3 | 58 | 2 |
IKK beta | 76 | 0 |
JNK1 | 58 | 2 |
JNK2 | 79 | 0 |
JNK3 | 70 | 0 |
Lck | 53 | 6 |
MAPKAP-K2 | 118 | 3 |
MAPKAP-K3 | 104 | 7 |
MARK3 | 16 | 1 |
MELK | 17 | 2 |
MKK1 | 50 | 1 |
MNK1 | 69 | 0 |
MNK2 | 34 | 0 |
MSK1 |
7
|
0 |
MST2 |
0
|
0 |
NEK2a | 84 | 1 |
NEK6 | 97 | 6 |
NEK7 | 108 | 1 |
p38 alpha MAPK | 116 | 4 |
p38 beta MAPK | 125 | 5 |
p38 delta MAPK | 78 | 1 |
p38 gamma MAPK | 83 | 8 |
PAK4 |
5
|
0 |
PAK5 |
7
|
0 |
PAK6 |
8
|
0 |
PDK1 | 11 | 0 |
PHK |
1
|
1 |
PIM1 | 21 | 1 |
PIM2 | 65 | 3 |
PIM3 |
5
|
0 |
PKA | 64 | 5 |
PKB alpha | 85 | 1 |
PKB beta | 87 | 1 |
PKC alpha |
1
|
0 |
PKC zeta | 80 | 4 |
PKD1 |
6
|
0 |
PLK1 | 80 | 1 |
PRAK | 83 | 3 |
PRK2 |
4
|
2 |
ROCK 2 | 59 | 4 |
RSK1 |
9
|
2 |
RSK2 |
5
|
0 |
S6K1 | 16 | 0 |
SGK1 | 59 | 5 |
SmMLCK | 31 | 1 |
Src | 74 | 2 |
SRPK1 | 92 | 5 |