Inhibitor | Gö 6976  

Compound name Brutto MW CAS PubChem CID Action Reference Reference
Gö 6976   C24H18N4O 378.40 136194-77-9 3501 PKC Gschwendt M. (1996) FEBS Lett. 392 77 Wenzel-Seifert K. (1994) Biochem. Biophys. Res. Commun. 200 1536

Screening Results Chart

Screening Results Tables

Screen Conc: 0.10µM
Kinase % Activity Remaining Standard Deviation
AMPK 16 3
Aurora B 23 0
Aurora C 26 3
BRSK2 48 6
CAMK1 99 3
CAMKK alpha 37 4
CAMKK beta 16 4
CDK2-Cyclin A
10
0
CHK1
1
0
CHK2 53 3
CK1 delta 88 3
CK2 88 4
CSK 74 3
DYRK1A 33 6
DYRK2 60 8
DYRK3 33 6
EF2K 109 3
ERK1 60 7
ERK2 46 2
ERK8 36 4
GSK3 beta 24 4
HIPK2 27 3
HIPK3 58 2
IKK beta 76 0
JNK1 58 2
JNK2 79 0
JNK3 70 0
Lck 53 6
MAPKAP-K2 118 3
MAPKAP-K3 104 7
MARK3 16 1
MELK 17 2
MKK1 50 1
MNK1 69 0
MNK2 34 0
MSK1
7
0
MST2
0
0
NEK2a 84 1
NEK6 97 6
NEK7 108 1
p38 alpha MAPK 116 4
p38 beta MAPK 125 5
p38 delta MAPK 78 1
p38 gamma MAPK 83 8
PAK4
5
0
PAK5
7
0
PAK6
8
0
PDK1 11 0
PHK
1
1
PIM1 21 1
PIM2 65 3
PIM3
5
0
PKA 64 5
PKB alpha 85 1
PKB beta 87 1
PKC alpha
1
0
PKC zeta 80 4
PKD1
6
0
PLK1 80 1
PRAK 83 3
PRK2
4
2
ROCK 2 59 4
RSK1
9
2
RSK2
5
0
S6K1 16 0
SGK1 59 5
SmMLCK 31 1
Src 74 2
SRPK1 92 5