| Compound name | Brutto | MW | CAS | PubChem CID | Action | Reference | Reference |
|---|---|---|---|---|---|---|---|
| Gö 6976 | C24H18N4O | 378.40 | 136194-77-9 | 3501 | PKC | Gschwendt M. (1996) FEBS Lett. 392 77 | Wenzel-Seifert K. (1994) Biochem. Biophys. Res. Commun. 200 1536 |
| Kinase | % Activity Remaining | Standard Deviation |
|---|---|---|
| AMPK | 16 | 3 |
| Aurora B | 23 | 0 |
| Aurora C | 26 | 3 |
| BRSK2 | 48 | 6 |
| CAMK1 | 99 | 3 |
| CAMKK alpha | 37 | 4 |
| CAMKK beta | 16 | 4 |
| CDK2-Cyclin A |
10
|
0 |
| CHK1 |
1
|
0 |
| CHK2 | 53 | 3 |
| CK1 delta | 88 | 3 |
| CK2 | 88 | 4 |
| CSK | 74 | 3 |
| DYRK1A | 33 | 6 |
| DYRK2 | 60 | 8 |
| DYRK3 | 33 | 6 |
| EF2K | 109 | 3 |
| ERK1 | 60 | 7 |
| ERK2 | 46 | 2 |
| ERK8 | 36 | 4 |
| GSK3 beta | 24 | 4 |
| HIPK2 | 27 | 3 |
| HIPK3 | 58 | 2 |
| IKK beta | 76 | 0 |
| JNK1 | 58 | 2 |
| JNK2 | 79 | 0 |
| JNK3 | 70 | 0 |
| Lck | 53 | 6 |
| MAPKAP-K2 | 118 | 3 |
| MAPKAP-K3 | 104 | 7 |
| MARK3 | 16 | 1 |
| MELK | 17 | 2 |
| MKK1 | 50 | 1 |
| MNK1 | 69 | 0 |
| MNK2 | 34 | 0 |
| MSK1 |
7
|
0 |
| MST2 |
0
|
0 |
| NEK2a | 84 | 1 |
| NEK6 | 97 | 6 |
| NEK7 | 108 | 1 |
| p38 alpha MAPK | 116 | 4 |
| p38 beta MAPK | 125 | 5 |
| p38 delta MAPK | 78 | 1 |
| p38 gamma MAPK | 83 | 8 |
| PAK4 |
5
|
0 |
| PAK5 |
7
|
0 |
| PAK6 |
8
|
0 |
| PDK1 | 11 | 0 |
| PHK |
1
|
1 |
| PIM1 | 21 | 1 |
| PIM2 | 65 | 3 |
| PIM3 |
5
|
0 |
| PKA | 64 | 5 |
| PKB alpha | 85 | 1 |
| PKB beta | 87 | 1 |
| PKC alpha |
1
|
0 |
| PKC zeta | 80 | 4 |
| PKD1 |
6
|
0 |
| PLK1 | 80 | 1 |
| PRAK | 83 | 3 |
| PRK2 |
4
|
2 |
| ROCK 2 | 59 | 4 |
| RSK1 |
9
|
2 |
| RSK2 |
5
|
0 |
| S6K1 | 16 | 0 |
| SGK1 | 59 | 5 |
| SmMLCK | 31 | 1 |
| Src | 74 | 2 |
| SRPK1 | 92 | 5 |