| Compound name | Brutto | MW | CAS | PubChem CID | Action | Reference | Reference |
|---|---|---|---|---|---|---|---|
| GF 109203X (Go 6850) | C25H24N4O2 | 412.50 | 133052-90-1 | 2396 | PKC | Hers I. (1999) FEBS Lett. 460 433 | Ku W.-C. (1997) Biochem. Biophys. Res. Commun. 241 730 |
| Kinase | % Activity Remaining | Standard Deviation |
|---|---|---|
| AMPK |
4
|
4 |
| CDK2-Cyclin A |
2
|
4 |
| CHK1 |
6
|
1 |
| CK1 delta | 83 | 7 |
| CK2 | 78 | 5 |
| CSK | 79 | 17 |
| DYRK1A |
0
|
3 |
| ERK2 | 75 | 1 |
| GSK3 beta |
2
|
0 |
| JNK1 | 58 | 4 |
| Lck | 27 | 7 |
| MAPKAP-K2 | 20 | 1 |
| MKK1 | 47 | 9 |
| MSK1 |
0
|
3 |
| NEK6 | 108 | 4 |
| p38 alpha MAPK | 73 | 8 |
| p38 beta MAPK | 81 | 3 |
| p38 delta MAPK | 102 | 5 |
| p38 gamma MAPK | 90 | 2 |
| PHK |
0
|
2 |
| PKA | 23 | 6 |
| PKB alpha | 23 | 0 |
| PKC alpha |
0
|
1 |
| PKD1 |
5
|
1 |
| PRAK | 69 | 3 |
| ROCK 2 | 43 | 10 |
| RSK1 |
0
|
1 |
| S6K1 |
3
|
0 |
| SGK1 |
1
|
4 |