

Compound name | Brutto | MW | CAS | PubChem CID | Action | Reference | Reference |
---|---|---|---|---|---|---|---|
GF 109203X (Go 6850) | C25H24N4O2 | 412.50 | 133052-90-1 | 2396 | PKC | Hers I. (1999) FEBS Lett. 460 433 | Ku W.-C. (1997) Biochem. Biophys. Res. Commun. 241 730 |
Kinase | % Activity Remaining | Standard Deviation |
---|---|---|
AMPK |
4
|
4 |
CDK2-Cyclin A |
2
|
4 |
CHK1 |
6
|
1 |
CK1 delta | 83 | 7 |
CK2 | 78 | 5 |
CSK | 79 | 17 |
DYRK1A |
0
|
3 |
ERK2 | 75 | 1 |
GSK3 beta |
2
|
0 |
JNK1 | 58 | 4 |
Lck | 27 | 7 |
MAPKAP-K2 | 20 | 1 |
MKK1 | 47 | 9 |
MSK1 |
0
|
3 |
NEK6 | 108 | 4 |
p38 alpha MAPK | 73 | 8 |
p38 beta MAPK | 81 | 3 |
p38 delta MAPK | 102 | 5 |
p38 gamma MAPK | 90 | 2 |
PHK |
0
|
2 |
PKA | 23 | 6 |
PKB alpha | 23 | 0 |
PKC alpha |
0
|
1 |
PKD1 |
5
|
1 |
PRAK | 69 | 3 |
ROCK 2 | 43 | 10 |
RSK1 |
0
|
1 |
S6K1 |
3
|
0 |
SGK1 |
1
|
4 |