Inhibitor | GF 109203X (Go 6850)  

Compound name Brutto MW CAS PubChem CID Action Reference Reference
GF 109203X (Go 6850)   C25H24N4O2 412.50 133052-90-1 2396 PKC Hers I. (1999) FEBS Lett. 460 433 Ku W.-C. (1997) Biochem. Biophys. Res. Commun. 241 730

Screening Results Chart

Screening Results Tables

Screen Conc: 10.00µM
Kinase % Activity Remaining Standard Deviation
AMPK
4
4
CDK2-Cyclin A
2
4
CHK1
6
1
CK1 delta 83 7
CK2 78 5
CSK 79 17
DYRK1A
0
3
ERK2 75 1
GSK3 beta
2
0
JNK1 58 4
Lck 27 7
MAPKAP-K2 20 1
MKK1 47 9
MSK1
0
3
NEK6 108 4
p38 alpha MAPK 73 8
p38 beta MAPK 81 3
p38 delta MAPK 102 5
p38 gamma MAPK 90 2
PHK
0
2
PKA 23 6
PKB alpha 23 0
PKC alpha
0
1
PKD1
5
1
PRAK 69 3
ROCK 2 43 10
RSK1
0
1
S6K1
3
0
SGK1
1
4