| Compound name | Brutto | MW | CAS | PubChem CID | Action | Reference | Reference |
|---|---|---|---|---|---|---|---|
| FMK (Caspase Inhibitor I) | C22H30FN3O7 | 467.50 | 187389-52-2 | 5737 | Caspase | Martin U. (2007) Apoptosis 12 525 | Misaghi S. (2004) Chem. Biol. 11 1677 |
| Kinase | % Activity Remaining | Standard Deviation |
|---|---|---|
| AMPK | 79 | 4 |
| Aurora B | 59 | 3 |
| Aurora C | 75 | 6 |
| BRSK2 | 53 | 6 |
| CAMK1 | 77 | 9 |
| CAMKK alpha | 70 | 12 |
| CAMKK beta | 49 | 3 |
| CDK2-Cyclin A | 80 | 7 |
| CHK1 | 88 | 4 |
| CHK2 | 81 | 9 |
| CK1 delta | 63 | 6 |
| CK2 | 92 | 10 |
| CSK | 55 | 7 |
| DYRK1A | 86 | 11 |
| DYRK2 | 91 | 8 |
| DYRK3 | 68 | 7 |
| EF2K | 97 | 8 |
| ERK1 | 92 | 6 |
| ERK2 | 79 | 5 |
| ERK8 | 58 | 4 |
| GSK3 beta | 65 | 6 |
| HIPK2 | 79 | 11 |
| HIPK3 | 79 | 9 |
| IKK beta | 92 | 8 |
| JNK1 | 81 | 3 |
| JNK2 | 83 | 5 |
| JNK3 | 89 | 4 |
| Lck |
10
|
1 |
| MAPKAP-K2 | 94 | 10 |
| MAPKAP-K3 | 92 | 6 |
| MARK3 | 80 | 3 |
| MELK | 65 | 8 |
| MKK1 | 80 | 8 |
| MNK1 | 42 | 2 |
| MNK2 | 65 | 6 |
| MSK1 | 75 | 3 |
| MST2 | 76 | 4 |
| NEK2a | 95 | 4 |
| NEK6 | 90 | 4 |
| NEK7 | 92 | 8 |
| p38 alpha MAPK | 72 | 2 |
| p38 beta MAPK | 85 | 4 |
| p38 delta MAPK | 103 | 9 |
| p38 gamma MAPK | 92 | 7 |
| PAK4 | 91 | 1 |
| PAK5 | 88 | 6 |
| PAK6 | 93 | 5 |
| PDK1 | 89 | 10 |
| PHK | 93 | 5 |
| PIM1 | 61 | 6 |
| PIM2 | 85 | 10 |
| PIM3 | 56 | 6 |
| PKA | 85 | 7 |
| PKB alpha | 82 | 3 |
| PKB beta | 97 | 4 |
| PKC alpha | 85 | 7 |
| PKC zeta | 91 | 5 |
| PKD1 | 83 | 4 |
| PLK1 | 82 | 5 |
| PRAK | 97 | 5 |
| PRK2 | 83 | 3 |
| ROCK 2 | 86 | 7 |
| RSK1 | 92 | 6 |
| RSK2 | 74 | 2 |
| S6K1 | 33 | 2 |
| SGK1 | 107 | 8 |
| SmMLCK | 82 | 4 |
| Src |
10
|
1 |
| SRPK1 | 85 | 1 |