

Compound name | Brutto | MW | CAS | PubChem CID | Action | Reference | Reference |
---|---|---|---|---|---|---|---|
FMK (Caspase Inhibitor I) | C22H30FN3O7 | 467.50 | 187389-52-2 | 5737 | Caspase | Martin U. (2007) Apoptosis 12 525 | Misaghi S. (2004) Chem. Biol. 11 1677 |
Kinase | % Activity Remaining | Standard Deviation |
---|---|---|
AMPK | 79 | 4 |
Aurora B | 59 | 3 |
Aurora C | 75 | 6 |
BRSK2 | 53 | 6 |
CAMK1 | 77 | 9 |
CAMKK alpha | 70 | 12 |
CAMKK beta | 49 | 3 |
CDK2-Cyclin A | 80 | 7 |
CHK1 | 88 | 4 |
CHK2 | 81 | 9 |
CK1 delta | 63 | 6 |
CK2 | 92 | 10 |
CSK | 55 | 7 |
DYRK1A | 86 | 11 |
DYRK2 | 91 | 8 |
DYRK3 | 68 | 7 |
EF2K | 97 | 8 |
ERK1 | 92 | 6 |
ERK2 | 79 | 5 |
ERK8 | 58 | 4 |
GSK3 beta | 65 | 6 |
HIPK2 | 79 | 11 |
HIPK3 | 79 | 9 |
IKK beta | 92 | 8 |
JNK1 | 81 | 3 |
JNK2 | 83 | 5 |
JNK3 | 89 | 4 |
Lck |
10
|
1 |
MAPKAP-K2 | 94 | 10 |
MAPKAP-K3 | 92 | 6 |
MARK3 | 80 | 3 |
MELK | 65 | 8 |
MKK1 | 80 | 8 |
MNK1 | 42 | 2 |
MNK2 | 65 | 6 |
MSK1 | 75 | 3 |
MST2 | 76 | 4 |
NEK2a | 95 | 4 |
NEK6 | 90 | 4 |
NEK7 | 92 | 8 |
p38 alpha MAPK | 72 | 2 |
p38 beta MAPK | 85 | 4 |
p38 delta MAPK | 103 | 9 |
p38 gamma MAPK | 92 | 7 |
PAK4 | 91 | 1 |
PAK5 | 88 | 6 |
PAK6 | 93 | 5 |
PDK1 | 89 | 10 |
PHK | 93 | 5 |
PIM1 | 61 | 6 |
PIM2 | 85 | 10 |
PIM3 | 56 | 6 |
PKA | 85 | 7 |
PKB alpha | 82 | 3 |
PKB beta | 97 | 4 |
PKC alpha | 85 | 7 |
PKC zeta | 91 | 5 |
PKD1 | 83 | 4 |
PLK1 | 82 | 5 |
PRAK | 97 | 5 |
PRK2 | 83 | 3 |
ROCK 2 | 86 | 7 |
RSK1 | 92 | 6 |
RSK2 | 74 | 2 |
S6K1 | 33 | 2 |
SGK1 | 107 | 8 |
SmMLCK | 82 | 4 |
Src |
10
|
1 |
SRPK1 | 85 | 1 |