| Compound name | Brutto | MW | CAS | PubChem CID | Action | Reference | Reference |
|---|---|---|---|---|---|---|---|
| EGCG (Epigallocatechin Gallate) | C22H18O11 | 458.40 | 989-51-5 | 65064 | PKC | Dell'Aica I. (2004) EMBO Rep. 5 418-422 | Tachibana H. (2004) Nat. Struct. Mol. Biol. 11 380 |
| Kinase | % Activity Remaining | Standard Deviation |
|---|---|---|
| AMPK | 66 | 2 |
| Aurora B | 12 | 3 |
| BRSK2 | 23 | 1 |
| BTK | 18 | 0 |
| CAMK1 | 19 | 8 |
| CAMKK beta | 65 | 2 |
| CDK2-Cyclin A | 88 | 4 |
| CHK1 | 72 | 3 |
| CHK2 | 61 | 1 |
| CK1 delta | 90 | 9 |
| CK2 | 89 | 17 |
| CSK | 88 | 10 |
| DYRK1A |
6
|
0 |
| DYRK2 |
0
|
1 |
| DYRK3 |
5
|
0 |
| EF2K | 86 | 2 |
| EPH-A2 | 76 | 0 |
| EPH-B3 |
1
|
0 |
| ERK1 | 17 | 1 |
| ERK2 | 72 | 4 |
| ERK8 | 20 | 0 |
| FGF-R1 |
6
|
0 |
| GSK3 beta | 70 | 6 |
| HIPK2 | 15 | 0 |
| IGF-1R | 19 | 4 |
| IKK beta | 21 | 3 |
| IKK epsilon | 27 | 4 |
| IR | 70 | 5 |
| IRR | 28 | 1 |
| JNK1 | 106 | 8 |
| JNK2 | 84 | 2 |
| Lck | 90 | 3 |
| MAPKAP-K2 | 22 | 1 |
| MARK3 |
6
|
1 |
| MELK | 53 | 1 |
| MKK1 | 58 | 24 |
| MNK1 | 71 | 10 |
| MNK2 | 73 | 7 |
| MSK1 | 40 | 4 |
| MST2 | 37 | 0 |
| MST4 | 24 | 1 |
| NEK2a |
5
|
1 |
| NEK6 | 56 | 4 |
| p38 alpha MAPK | 80 | 8 |
| p38 beta MAPK | 96 | 20 |
| p38 delta MAPK | 102 | 17 |
| p38 gamma MAPK | 98 | 15 |
| PAK4 | 22 | 1 |
| PAK5 | 35 | 1 |
| PAK6 |
8
|
4 |
| PDK1 | 73 | 0 |
| PHK | 75 | 6 |
| PIM1 | 15 | 2 |
| PIM2 | 47 | 0 |
| PIM3 | 17 | 0 |
| PKA | 87 | 1 |
| PKB alpha | 75 | 20 |
| PKB beta |
1
|
0 |
| PKC alpha | 81 | 3 |
| PKC zeta |
2
|
1 |
| PKD1 | 16 | 1 |
| PLK1 |
7
|
2 |
| PRAK |
5
|
2 |
| PRK2 | 82 | 3 |
| ROCK 2 | 74 | 5 |
| RSK1 | 46 | 2 |
| RSK2 |
6
|
6 |
| S6K1 | 37 | 1 |
| SGK1 | 58 | 2 |
| SmMLCK | 51 | 2 |
| Src | 21 | 0 |
| SRPK1 |
5
|
3 |
| SYK | 67 | 8 |
| TBK1 | 65 | 4 |
| VEGFR1 | 20 | 1 |
| YES1 | 12 | 3 |