Inhibitor | 1 NM-PP1 (PP1 Analog II)  

Compound name Brutto MW CAS PubChem CID Action Reference Reference
1 NM-PP1 (PP1 Analog II)   C20H21N5 331.40 221244-14-0 5154691 Src Ira G. (2004) Nature 431 1011 Papa F.R. (2003) Science 302 1533

Screening Results Chart

Screening Results Tables

Screen Conc: 10.00µM
Kinase Sort ascending % Activity Remaining Standard Deviation
SRPK1 93 0
Src
7
0
SmMLCK 71 1
SGK1 99 5
S6K1 82 6
RSK2 68 2
RSK1 56 6
ROCK 2 76 1
PRK2 97 2
PRAK 62 1
PLK1 94 0
PKD1
3
0
PKC zeta 84 4
PKC alpha 79 2
PKB beta 91 4
PKB alpha 62 1
PKA
7
1
PIM3 87 3
PIM2 103 2
PIM1 94 0
PHK 78 3
PDK1 101 0
PAK6 65 5
PAK5 47 0
PAK4 50 8
p38 gamma MAPK 98 2
p38 delta MAPK 94 4
p38 beta MAPK 15 5
p38 alpha MAPK
8
1
NEK7 109 8
NEK6 110 1
NEK2a 91 5
MST2
9
0
MSK1 69 2
MNK2 98 5
MNK1 105 0
MKK1 76 6
MELK 23 0
MARK3 54 2
MAPKAP-K3 93 1
MAPKAP-K2 114 7
Lck
3
0
JNK3 79 1
JNK2 63 4
JNK1 85 4
IKK beta 95 0
HIPK3 103 3
HIPK2 71 3
GSK3 beta 92 3
ERK8 48 0
ERK2 32 7
ERK1 45 1
EF2K 105 2
DYRK3 58 4
DYRK2 112 5
DYRK1A 66 2
CSK
6
1
CK2 91 2
CK1 delta 14 2
CHK2 44 3
CHK1 105 0
CDK2-Cyclin A 42 5
CAMKK beta 76 2
CAMKK alpha 89 4
CAMK1 46 1
BRSK2 97 4
Aurora C 73 1
Aurora B 82 0
AMPK 96 2
Screen Conc: 1.00µM
Kinase Sort ascending % Activity Remaining Standard Deviation
SRPK1 99 3
Src 29 6
SmMLCK 80 7
SGK1 98 1
S6K1 91 7
RSK2 97 1
RSK1 83 2
ROCK 2 83 0
PRK2 109 5
PRAK 89 0
PLK1 95 4
PKD1 13 0
PKC zeta 82 1
PKC alpha 81 1
PKB beta 97 4
PKB alpha 82 1
PKA 32 2
PIM3 99 2
PIM2 101 4
PIM1 103 3
PHK 80 5
PDK1 96 1
PAK6 88 0
PAK5 74 0
PAK4 71 6
p38 gamma MAPK 95 0
p38 delta MAPK 97 1
p38 beta MAPK 53 4
p38 alpha MAPK 41 2
NEK7 110 2
NEK6 94 3
NEK2a 101 6
MST2 45 2
MSK1 78 1
MNK2 114 1
MNK1 109 8
MKK1 112 2
MELK 66 2
MARK3 71 6
MAPKAP-K3 96 1
MAPKAP-K2 98 3
Lck 18 2
JNK3 98 8
JNK2 78 1
JNK1 90 0
IKK beta 98 2
HIPK3 96 3
HIPK2 95 4
GSK3 beta 90 3
ERK8 76 0
ERK2 64 3
ERK1 84 5
EF2K 99 2
DYRK3 80 4
DYRK2 94 2
DYRK1A 92 8
CSK 36 2
CK2 80 7
CK1 delta 56 4
CHK2 83 2
CHK1 96 7
CDK2-Cyclin A 85 4
CAMKK beta 102 6
CAMKK alpha 100 1
CAMK1 83 6
BRSK2 101 3
Aurora C 76 1
Aurora B 105 2
AMPK 86 2