Inhibitor | SGK1-Sanofi-ex.290-R  

Compound name Brutto MW CAS PubChem CID Action Reference Reference
SGK1-Sanofi-ex.290-R   C24H25ClN6O5S 545.01 SGK1

Screening Results Chart

Screening Results Tables

Screen Conc: 1.00µM
Kinase % Activity Remaining Standard Deviation
ABL 88 1
AMPK (hum) 15 1
ASK1 104 1
Aurora A 108 12
Aurora B 70 1
BRK 113 9
BRSK1 95 3
BRSK2 102 8
BTK 91 10
CAMK1
3
0
CAMKK beta 77 5
CDK2-Cyclin A 94 14
CDK9-Cyclin T1 105 10
CHK1 95 15
CHK2
9
3
CK1 delta 65 5
CK1 gamma 2 112 9
CK2 100 6
CLK2 88 1
CSK 66 5
DAPK1 87 8
DDR2 80 1
DYRK1A 103 10
DYRK2 100 2
DYRK3 89 13
EF2K 112 14
EIF2AK3 66 0
EPH-A2 109 10
EPH-A4 95 22
EPH-B1 117 10
EPH-B2 120 6
EPH-B3 104 21
EPH-B4 103 11
ERK1 115 16
ERK2 109 8
ERK5 84 13
ERK8 18 0
FGF-R1 104 3
GCK 90 13
GSK3 beta 90 7
HER4 102 17
HIPK1 117 10
HIPK2 50 6
HIPK3 109 9
IGF-1R 88 2
IKK beta 102 0
IKK epsilon 34 5
IR 102 8
IRAK1 93 2
IRAK4 74 12
IRR 96 13
JAK2 112 14
JNK1 101 6
JNK2 105 2
JNK3 104 25
Lck 89 7
LKB1 106 22
MAP4K3
2
0
MAP4K5 19 3
MAPKAP-K2 87 16
MAPKAP-K3 105 27
MARK1 115 19
MARK2 113 9
MARK3 89 3
MARK4 98 10
MEKK1 112 6
MELK 11 0
MINK1 101 14
MKK1 66 8
MKK2 41 11
MKK6 102 17
MLK1
9
2
MLK3
10
4
MNK1 87 5
MNK2 119 23
MPSK1 82 6
MSK1
10
1
MST2 105 23
MST3 57 17
MST4 50 6
NEK2a 74 5
NEK6 88 2
NUAK1 91 11
OSR1 110 4
p38 alpha MAPK 111 2
p38 beta MAPK 99 3
p38 delta MAPK 111 7
p38 gamma MAPK 112 3
PAK2 90 7
PAK4 91 8
PAK5 110 5
PAK6 94 13
PDGFRA 91 8
PDK1 117 34
PHK 97 10
PIM1 83 24
PIM2 105 3
PIM3 105 11
PINK 99 13
PKA 85 6
PKB alpha 49 1
PKB beta 55 7
PKC alpha 113 4
PKC gamma 101 9
PKC zeta 110 17
PKD1 15 4
PLK1 102 4
PRAK 78 11
PRK2 76 6
RIPK2 124 16
ROCK 2 105 7
RSK1
7
0
RSK2 24 2
S6K1
1
0
SGK1
2
1
SIK2 91 1
SIK3 102 9
SmMLCK 23 4
Src 104 16
SRPK1 94 6
STK33 74 2
SYK 88 20
TAK1 101 12
TAO1 110 8
TBK1 62 3
TESK1 77 2
TGFBR1 120 15
TIE2 17 10
TLK1 89 12
TrkA 104 0
TSSK1 98 8
TTBK1 109 16
TTBK2 114 10
TTK 76 3
ULK1 78 2
ULK2 46 2
VEGFR1 82 26
WNK1 110 7
YES1 92 12
ZAP70 98 7