Inhibitor | CKI-7  

Screen Conc: 25.00µM

Kinase	% Activity Remaining Sort descending	Standard Deviation
CK1 delta	12	0
SGK1	25	2
MNK1	26	0
PIM1	28	1
PIM3	28	0
ERK8	29	6
AMPK	29	5
DYRK1A	39	6
MSK1	42	2
BRSK2	42	1
DYRK3	46	1
PRK2	47	3
RSK1	48	3
S6K1	49	5
PKC zeta	52	0
PKB alpha	54	1
PIM2	55	6
IRR	60	4
PKD1	60	3
CDK2-Cyclin A	62	4
RSK2	63	4
MELK	63	4
CHK2	64	0
CK2	65	1
PKA	65	6
ROCK 2	65	8
IKK epsilon	70	4
EPH-A2	71	0
PHK	72	5
GSK3 beta	75	4
MKK1	76	2
DYRK2	76	2
SYK	76	11
MNK2	76	0
PAK6	78	3
Aurora B	78	0
MARK3	78	5
CSK	79	5
p38 delta MAPK	79	8
PLK1	81	4
PRAK	81	4
CAMK1	82	3
Lck	83	6
FGF-R1	83	7
PDK1	83	3
SmMLCK	84	7
NEK2a	85	4
MAPKAP-K2	85	3
PAK5	86	7
CAMKK beta	86	3
CHK1	86	2
JNK2	86	9
PKC alpha	86	2
SRPK1	86	2
MAPKAP-K3	86	7
HIPK3	86	7
CAMKK alpha	86	4
IKK beta	87	2
TBK1	87	9
PAK4	88	3
PKB beta	89	4
NEK6	90	2
JNK1	91	0
MST2	91	0
Src	92	1
EF2K	94	6
MST4	95	3
Aurora C	95	3
HIPK2	98	7
ERK2	100	2
ERK1	101	3
p38 beta MAPK	101	9
p38 gamma MAPK	101	3
JNK3	102	0
NEK7	102	3
p38 alpha MAPK	103	4
YES1	110	12

Screen Conc: 2.50µM

Kinase	% Activity Remaining Sort descending	Standard Deviation
CK1 delta	62	3
PIM2	72	1
MKK1	72	12
PRK2	73	10
MNK1	76	8
S6K1	76	0
AMPK	78	1
CHK2	79	9
MST4	80	3
Lck	81	4
PKC alpha	82	2
IKK beta	82	5
GSK3 beta	82	5
JNK1	82	8
JNK2	83	3
JNK3	84	12
DYRK1A	84	0
SGK1	85	10
p38 alpha MAPK	87	6
CHK1	87	5
MAPKAP-K2	88	3
p38 gamma MAPK	89	3
Src	89	2
CSK	89	16
Aurora B	90	1
NEK2a	91	0
PRAK	91	1
CAMK1	91	7
PKD1	92	1
ROCK 2	92	11
MNK2	93	0
RSK1	93	2
p38 beta MAPK	94	5
MAPKAP-K3	94	6
NEK6	94	4
ERK8	95	4
PDK1	95	11
PKB beta	96	3
PKB alpha	97	2
MARK3	98	7
CDK2-Cyclin A	98	14
SRPK1	99	6
PKA	99	6
CK2	100	4
NEK7	100	7
ERK2	101	6
RSK2	103	3
PHK	103	2
PLK1	105	13
MSK1	110	36
EF2K	111	4
SmMLCK	122	13