Inhibitor | SGK1-Sanofi-14h  

Compound name Brutto MW CAS PubChem CID Action Reference Reference
SGK1-Sanofi-14h   C17H12Cl2N6O2S 435.29 SGK Halland, N (2015) ACS Medicinal Chemistry Letters , 6,73-78

Screening Results Chart

Screening Results Tables

Screen Conc: 1.00µM
Kinase % Activity Remaining Standard Deviation
ABL 90 6
AMPK (hum) 96 1
ASK1 121 18
Aurora A 100 6
Aurora B 42 7
BRK 100 12
BRSK1 104 6
BRSK2 97 12
BTK 89 6
CAMK1 63 3
CAMKK beta 100 6
CDK2-Cyclin A 104 6
CDK9-Cyclin T1 107 3
CHK1 112 17
CHK2 50 5
CK1 delta 100 4
CK1 gamma 2 81 1
CK2 128 3
CLK2 90 3
CSK 129 9
DAPK1 105 10
DDR2 105 1
DYRK1A 94 4
DYRK2 109 16
DYRK3 94 4
EF2K 98 2
EIF2AK3 81 6
EPH-A2 117 11
EPH-A4 111 5
EPH-B1 98 9
EPH-B2 103 2
EPH-B3 99 10
EPH-B4 99 5
ERK1 95 14
ERK2 99 7
ERK5 119 3
ERK8 38 1
FGF-R1 115 11
GCK 34 3
GSK3 beta 97 3
HER4 103 7
HIPK1 92 9
HIPK2 45 4
HIPK3 98 5
IGF-1R 97 12
IKK beta 100 2
IKK epsilon 69 2
IR 82 8
IRAK1 90 2
IRAK4 108 3
IRR 105 1
JAK2 77 6
JNK1 94 3
JNK2 100 3
JNK3 102 3
Lck 111 12
LKB1 97 1
MAP4K3 25 3
MAP4K5 13 3
MAPKAP-K2 114 9
MAPKAP-K3 122 6
MARK1 130 17
MARK2 95 8
MARK3 95 8
MARK4 106 5
MEKK1 114 14
MELK 67 4
MINK1 71 7
MKK1 72 7
MKK2 70 5
MKK6 91 10
MLK1
10
 0
MLK3
6
 0
MNK1 104 4
MNK2 97 3
MPSK1 114 2
MSK1 31 0
MST2 99 8
MST3 91 7
MST4 104 9
NEK2a 103 1
NEK6 105 5
NUAK1 61 7
OSR1 99 10
p38 alpha MAPK 117 0
p38 beta MAPK 97 5
p38 delta MAPK 114 17
p38 gamma MAPK 104 2
PAK2 110 8
PAK4 46 4
PAK5 87 6
PAK6 101 7
PDGFRA 89 6
PDK1 96 15
PHK 109 1
PIM1 111 4
PIM2 100 15
PIM3 102 10
PINK 99 7
PKA 109 5
PKB alpha 105 20
PKB beta 98 6
PKC alpha 106 6
PKC gamma 111 14
PKC zeta 97 9
PKD1 87 1
PLK1 108 8
PRAK 107 4
PRK2 89 11
RIPK2 95 1
ROCK 2 117 14
RSK1 48 1
RSK2 77 23
S6K1
3
 0
SGK1
6
 1
SIK2 101 1
SIK3 102 12
SmMLCK 101 1
Src 115 12
SRPK1 108 0
STK33 105 8
SYK 101 5
TAK1 45 4
TAO1 90 2
TBK1 94 5
TESK1 111 10
TGFBR1 78 20
TIE2
10
 1
TLK1 112 11
TrkA 101 13
TSSK1 99 8
TTBK1 100 8
TTBK2 110 12
TTK 77 1
ULK1 100 7
ULK2 84 2
VEGFR1 73 1
WNK1 103 8
YES1 95 16
ZAP70 110 16