Inhibitor | SGK1-Sanofi-14n  

Compound name Brutto MW CAS PubChem CID Action Reference Reference
SGK1-Sanofi-14n   C17H12CIFN6O2S 418.83 SGK Halland, N (2015) ACS Medicinal Chemistry Letters 6 73-78

Screening Results Chart

Screening Results Tables

Screen Conc: 1.00µM
Kinase % Activity Remaining Standard Deviation
ABL 105 35
AMPK (hum) 79 8
ASK1 142 4
Aurora A 110 3
Aurora B 39 3
BRK 103 12
BRSK1 94 7
BRSK2 91 1
BTK 83 2
CAMK1 56 1
CAMKK beta 94 1
CDK2-Cyclin A 101 2
CDK9-Cyclin T1 115 1
CHK1 97 5
CHK2 64 6
CK1 delta 102 6
CK1 gamma 2 95 14
CK2 100 4
CLK2 90 10
CSK 100 8
DAPK1 110 10
DDR2 101 1
DYRK1A 97 10
DYRK2 101 6
DYRK3 95 14
EF2K 98 10
EIF2AK3 83 4
EPH-A2 108 6
EPH-A4 94 2
EPH-B1 114 5
EPH-B2 104 2
EPH-B3 99 4
EPH-B4 109 17
ERK1 99 2
ERK2 94 3
ERK5 101 5
ERK8 51 25
FGF-R1 109 7
GCK 34 9
GSK3 beta 95 7
HER4 119 5
HIPK1 96 15
HIPK2 64 8
HIPK3 102 5
IGF-1R 82 16
IKK beta 102 4
IKK epsilon 67 1
IR 98 10
IRAK1 100 0
IRAK4 100 6
IRR 100 6
JAK2 80 9
JNK1 104 6
JNK2 90 4
JNK3 89 9
Lck 101 8
LKB1 90 0
MAP4K3 39 3
MAP4K5 34 1
MAPKAP-K2 104 12
MAPKAP-K3 110 6
MARK1 106 5
MARK2 105 1
MARK3 113 13
MARK4 93 1
MEKK1 104 3
MELK 78 2
MINK1 75 8
MKK1 77 10
MKK2 80 9
MKK6 94 10
MLK1
8
 2
MLK3
6
 1
MNK1 80 2
MNK2 79 1
MPSK1 93 15
MSK1 41 7
MST2 95 3
MST3 98 9
MST4 102 3
NEK2a 96 2
NEK6 91 5
NUAK1 64 7
OSR1 95 4
p38 alpha MAPK 92 13
p38 beta MAPK 92 15
p38 delta MAPK 90 13
p38 gamma MAPK 98 9
PAK2 113 13
PAK4 47 5
PAK5 81 4
PAK6 86 0
PDGFRA 73 2
PDK1 104 16
PHK 105 1
PIM1 103 0
PIM2 110 12
PIM3 92 3
PINK 107 8
PKA 102 11
PKB alpha 93 5
PKB beta 102 28
PKC alpha 102 9
PKC gamma 99 8
PKC zeta 91 7
PKD1 87 3
PLK1 93 21
PRAK 112 26
PRK2 98 7
RIPK2 108 16
ROCK 2 105 0
RSK1 56 2
RSK2 79 17
S6K1
2
 0
SGK1
6
 3
SIK2 98 1
SIK3 94 6
SmMLCK 104 3
Src 109 25
SRPK1 93 1
STK33 88 2
SYK 88 2
TAK1 38 0
TAO1 77 3
TBK1 83 3
TESK1 108 1
TGFBR1 80 10
TIE2
10
 3
TLK1 109 8
TrkA 108 3
TSSK1 94 2
TTBK1 101 5
TTBK2 107 7
TTK 72 2
ULK1 99 3
ULK2 89 1
VEGFR1 80 12
WNK1 102 1
YES1 88 0
ZAP70 90 11