Inhibitor | SGK-Sanofi-14i  

Compound name Brutto MW CAS PubChem CID Action Reference Reference
SGK-Sanofi-14i   C18H15ClN6O3S SGK Halland, N (2015) ACS Medicinal Chemistry Letters 6 73-78

Screening Results Chart

Screening Results Tables

Screen Conc: 1.00µM
Kinase % Activity Remaining Standard Deviation
ABL 104 15
AMPK (hum) 83 7
ASK1 98 5
Aurora A 111 4
Aurora B 87 22
BRK 111 6
BRSK1 100 1
BRSK2 87 15
BTK 92 1
CAMK1 66 8
CAMKK beta 117 7
CDK2-Cyclin A 85 2
CDK9-Cyclin T1 111 4
CHK1 73 1
CHK2 75 13
CK1 delta 116 9
CK1 gamma 2 98 15
CK2 87 4
CLK2 97 12
CSK 84 10
DAPK1 103 10
DDR2 103 0
DYRK1A 98 2
DYRK2 123 1
DYRK3 90 45
EF2K 107 22
EIF2AK3 80 15
EPH-A2 98 2
EPH-A4 98 8
EPH-B1 97 19
EPH-B2 97 12
EPH-B3 98 4
EPH-B4 98 11
ERK1 99 3
ERK2 99 2
ERK5 101 7
ERK8 40 2
FGF-R1 92 10
GCK 40 0
GSK3 beta 104 1
HER4 94 12
HIPK1 78 2
HIPK2 15 3
HIPK3 47 4
IGF-1R 119 5
IKK beta 105 8
IKK epsilon 83 12
IR 111 25
IRAK1 80 16
IRAK4 113 5
IRR 91 6
JAK2 81 7
JNK1 91 14
JNK2 106 2
JNK3 99 3
Lck 88 4
LKB1 117 5
MAP4K3 66 11
MAP4K5 39 3
MAPKAP-K2 97 15
MAPKAP-K3 101 5
MARK1 116 14
MARK2 92 4
MARK3 103 9
MARK4 86 6
MEKK1 92 4
MELK 81 4
MINK1 68 3
MKK1 99 5
MKK2 90 9
MKK6 94 5
MLK1 24 2
MLK3 11 1
MNK1 84 10
MNK2 116 13
MPSK1 113 7
MSK1 30 10
MST2 108 5
MST3 102 7
MST4 67 19
NEK2a 109 7
NEK6 100 11
NUAK1 65 3
OSR1 110 15
p38 alpha MAPK 98 9
p38 beta MAPK 91 8
p38 delta MAPK 94 11
p38 gamma MAPK 105 0
PAK2 100 8
PAK4 32 2
PAK5 68 5
PAK6 98 2
PDGFRA 55 9
PDK1 112 16
PHK 122 6
PIM1 105 5
PIM2 134 2
PIM3 104 12
PINK 98 21
PKA 101 2
PKB alpha 104 4
PKB beta 101 7
PKC alpha 108 9
PKC gamma 97 5
PKC zeta 101 9
PKD1 88 1
PLK1 96 1
PRAK 97 3
PRK2 99 14
RIPK2 94 3
ROCK 2 96 11
RSK1 94 1
RSK2 92 0
S6K1
5
0
SGK1
4
0
SIK2 107 15
SIK3 107 15
SmMLCK 93 3
Src 121 6
SRPK1 107 10
STK33 102 9
SYK 84 26
TAK1 63 7
TAO1 75 4
TBK1 61 34
TESK1 105 19
TGFBR1 118 2
TIE2
9
0
TLK1 82 3
TrkA 79 19
TSSK1 103 11
TTBK1 112 7
TTBK2 124 15
TTK 70 14
ULK1 98 8
ULK2 97 6
VEGFR1 68 7
WNK1 97 1
YES1 95 2
ZAP70 112 9