Inhibitor | CKI-7  

Screen Conc: 2.50µM

Kinase	% Activity Remaining	Standard Deviation
AMPK	78	1
Aurora B	90	1
CAMK1	91	7
CDK2-Cyclin A	98	14
CHK1	87	5
CHK2	79	9
CK1 delta	62	3
CK2	100	4
CSK	89	16
DYRK1A	84	0
EF2K	111	4
ERK2	101	6
ERK8	95	4
GSK3 beta	82	5
IKK beta	82	5
JNK1	82	8
JNK2	83	3
JNK3	84	12
Lck	81	4
MAPKAP-K2	88	3
MAPKAP-K3	94	6
MARK3	98	7
MKK1	72	12
MNK1	76	8
MNK2	93	0
MSK1	110	36
MST4	80	3
NEK2a	91	0
NEK6	94	4
NEK7	100	7
p38 alpha MAPK	87	6
p38 beta MAPK	94	5
p38 gamma MAPK	89	3
PDK1	95	11
PHK	103	2
PIM2	72	1
PKA	99	6
PKB alpha	97	2
PKB beta	96	3
PKC alpha	82	2
PKD1	92	1
PLK1	105	13
PRAK	91	1
PRK2	73	10
ROCK 2	92	11
RSK1	93	2
RSK2	103	3
S6K1	76	0
SGK1	85	10
SmMLCK	122	13
Src	89	2
SRPK1	99	6

Screen Conc: 25.00µM

Kinase	% Activity Remaining	Standard Deviation
AMPK	29	5
Aurora B	78	0
Aurora C	95	3
BRSK2	42	1
CAMK1	82	3
CAMKK alpha	86	4
CAMKK beta	86	3
CDK2-Cyclin A	62	4
CHK1	86	2
CHK2	64	0
CK1 delta	12	0
CK2	65	1
CSK	79	5
DYRK1A	39	6
DYRK2	76	2
DYRK3	46	1
EF2K	94	6
EPH-A2	71	0
ERK1	101	3
ERK2	100	2
ERK8	29	6
FGF-R1	83	7
GSK3 beta	75	4
HIPK2	98	7
HIPK3	86	7
IKK beta	87	2
IKK epsilon	70	4
IRR	60	4
JNK1	91	0
JNK2	86	9
JNK3	102	0
Lck	83	6
MAPKAP-K2	85	3
MAPKAP-K3	86	7
MARK3	78	5
MELK	63	4
MKK1	76	2
MNK1	26	0
MNK2	76	0
MSK1	42	2
MST2	91	0
MST4	95	3
NEK2a	85	4
NEK6	90	2
NEK7	102	3
p38 alpha MAPK	103	4
p38 beta MAPK	101	9
p38 delta MAPK	79	8
p38 gamma MAPK	101	3
PAK4	88	3
PAK5	86	7
PAK6	78	3
PDK1	83	3
PHK	72	5
PIM1	28	1
PIM2	55	6
PIM3	28	0
PKA	65	6
PKB alpha	54	1
PKB beta	89	4
PKC alpha	86	2
PKC zeta	52	0
PKD1	60	3
PLK1	81	4
PRAK	81	4
PRK2	47	3
ROCK 2	65	8
RSK1	48	3
RSK2	63	4
S6K1	49	5
SGK1	25	2
SmMLCK	84	7
Src	92	1
SRPK1	86	2
SYK	76	11
TBK1	87	9
YES1	110	12