Inhibitor | STOCK1S-50699  

Screen Conc: 1.00µM

Kinase	% Activity Remaining	Standard Deviation
ABL	113	17
AMPK (hum)	108	3
ASK1	107	10
Aurora A	99	1
Aurora B	87	22
BRK	104	14
BRSK1	113	15
BRSK2	94	4
BTK	106	21
CAMK1	97	15
CAMKK beta	104	6
CDK2-Cyclin A	104	14
CDK9-Cyclin T1	101	1
CHK1	106	4
CHK2	99	12
CK1 delta	86	7
CK1 gamma 2	97	1
CK2	107	0
CLK2	89	1
CSK	85	10
DAPK1	103	0
DDR2	102	1
DYRK1A	78	3
DYRK2	91	4
DYRK3	102	6
EF2K	101	6
EIF2AK3	101	1
EPH-A2	116	6
EPH-A4	93	14
EPH-B1	125	24
EPH-B2	102	7
EPH-B3	93	13
EPH-B4	112	5
ERK1	94	11
ERK2	84	11
ERK5	103	8
ERK8	88	12
FGF-R1	96	1
GCK	107	6
GSK3 beta	103	10
HER4	121	8
HIPK1	95	5
HIPK2	110	0
HIPK3	95	1
IGF-1R	95	29
IKK beta	98	10
IKK epsilon	96	8
IR	114	1
IRAK1	82	15
IRAK4	90	10
IRR	105	18
JAK2	110	1
JNK1	97	12
JNK2	97	2
JNK3	105	1
Lck	115	2
LKB1	103	10
MAP4K3	97	1
MAP4K5	103	3
MAPKAP-K2	106	10
MAPKAP-K3	95	1
MARK1	100	14
MARK2	95	2
MARK3	100	7
MARK4	111	32
MEKK1	90	6
MELK	90	4
MINK1	90	6
MKK1	96	14
MKK2	90	2
MKK6	95	6
MLK1	95	4
MLK3	96	8
MNK1	106	19
MNK2	99	12
MPSK1	101	5
MSK1	100	2
MST2	71	6
MST3	110	8
MST4	75	16
NEK2a	107	6
NEK6	99	15
NUAK1	101	5
OSR1	112	5
p38 alpha MAPK	95	3
p38 beta MAPK	121	15
p38 delta MAPK	104	2
p38 gamma MAPK	94	5
PAK2	96	1
PAK4	103	1
PAK5	105	6
PAK6	100	0
PDGFRA	102	2
PDK1	93	14
PHK	103	4
PIM1	94	10
PIM2	93	6
PIM3	82	8
PINK	101	1
PKA	96	12
PKB alpha	85	6
PKB beta	93	2
PKC alpha	80	1
PKC gamma	105	5
PKC zeta	92	3
PKD1	100	11
PLK1	102	0
PRAK	97	6
PRK2	92	13
RIPK2	84	9
ROCK 2	90	2
RSK1	85	5
RSK2	108	10
S6K1	96	9
SGK1	110	14
SIK2	108	22
SIK3	97	0
SmMLCK	95	25
Src	91	5
SRPK1	93	3
STK33	106	1
SYK	92	2
TAK1	100	10
TAO1	96	0
TBK1	111	4
TESK1	104	3
TGFBR1	111	1
TIE2	93	1
TLK1	93	8
TrkA	96	7
TSSK1	96	3
TTBK1	102	9
TTBK2	90	5
TTK	87	18
ULK1	108	8
ULK2	96	8
VEGFR1	84	10
WNK1	103	2
YES1	106	11
ZAP70	112	1

Screen Conc: 10.00µM

Kinase	% Activity Remaining	Standard Deviation
ABL	99	5
AMPK (hum)	112	8
ASK1	101	3
Aurora A	108	6
Aurora B	41	10
BRK	95	32
BRSK1	95	15
BRSK2	61	10
BTK	104	6
CAMK1	95	1
CAMKK beta	96	12
CDK2-Cyclin A	99	20
CDK9-Cyclin T1	102	3
CHK1	97	6
CHK2	88	8
CK1 delta	32	12
CK1 gamma 2	72	10
CK2	82	2
CLK2	90	1
CSK	109	19
DAPK1	115	14
DDR2	110	9
DYRK1A	66	3
DYRK2	85	2
DYRK3	102	6
EF2K	87	2
EIF2AK3	107	7
EPH-A2	103	1
EPH-A4	98	14
EPH-B1	93	11
EPH-B2	106	10
EPH-B3	98	16
EPH-B4	109	13
ERK1	58	2
ERK2	69	8
ERK5	87	16
ERK8	55	7
FGF-R1	77	4
GCK	100	10
GSK3 beta	116	1
HER4	110	12
HIPK1	76	10
HIPK2	116	10
HIPK3	93	7
IGF-1R	83	4
IKK beta	78	3
IKK epsilon	60	6
IR	90	17
IRAK1	57	3
IRAK4	96	17
IRR	72	5
JAK2	125	13
JNK1	87	7
JNK2	96	2
JNK3	103	8
Lck	101	1
LKB1	105	27
MAP4K3	89	3
MAP4K5	103	2
MAPKAP-K2	98	3
MAPKAP-K3	84	8
MARK1	89	14
MARK2	102	8
MARK3	83	20
MARK4	113	8
MEKK1	84	3
MELK	53	1
MINK1	88	0
MKK1	94	8
MKK2	85	3
MKK6	112	9
MLK1	87	4
MLK3	75	3
MNK1	97	7
MNK2	105	16
MPSK1	79	7
MSK1	67	3
MST2	69	11
MST3	110	7
MST4	85	14
NEK2a	103	2
NEK6	91	2
NUAK1	88	8
OSR1	112	2
p38 alpha MAPK	91	5
p38 beta MAPK	98	5
p38 delta MAPK	87	4
p38 gamma MAPK	90	1
PAK2	94	0
PAK4	108	0
PAK5	99	1
PAK6	102	1
PDGFRA	123	16
PDK1	116	4
PHK	104	0
PIM1	73	4
PIM2	84	2
PIM3	84	7
PINK	103	21
PKA	92	7
PKB alpha	65	2
PKB beta	77	3
PKC alpha	88	23
PKC gamma	86	5
PKC zeta	110	1
PKD1	61	4
PLK1	114	21
PRAK	92	1
PRK2	65	17
RIPK2	82	9
ROCK 2	89	1
RSK1	47	18
RSK2	43	8
S6K1	85	16
SGK1	51	2
SIK2	83	10
SIK3	88	3
SmMLCK	99	28
Src	143	5
SRPK1	95	16
STK33	95	3
SYK	64	1
TAK1	68	13
TAO1	93	0
TBK1	84	12
TESK1	112	10
TGFBR1	108	1
TIE2	96	4
TLK1	101	11
TrkA	90	1
TSSK1	72	10
TTBK1	104	0
TTBK2	100	5
TTK	64	17
ULK1	83	5
ULK2	90	1
VEGFR1	23	3
WNK1	104	12
YES1	105	10
ZAP70	112	11