Inhibitor | STOCK2S-26016  

Screen Conc: 1.00µM

Kinase	% Activity Remaining	Standard Deviation
ABL	88	4
AMPK (hum)	88	17
ASK1	101	4
Aurora A	100	1
Aurora B	83	0
BRK	101	3
BRSK1	84	8
BRSK2	101	18
BTK	90	11
CAMK1	96	2
CAMKK beta	95	3
CDK2-Cyclin A	80	7
CDK9-Cyclin T1	83	1
CHK1	90	6
CHK2	90	3
CK1 delta	63	12
CK1 gamma 2	95	11
CK2	120	9
CLK2	89	7
CSK	100	4
DAPK1	102	1
DDR2	101	6
DYRK1A	108	22
DYRK2	100	7
DYRK3	101	1
EF2K	107	8
EIF2AK3	108	9
EPH-A2	104	6
EPH-A4	119	37
EPH-B1	109	2
EPH-B2	109	13
EPH-B3	107	10
EPH-B4	94	4
ERK1	101	3
ERK2	92	9
ERK5	83	6
ERK8	90	9
FGF-R1	93	3
GCK	101	9
GSK3 beta	107	3
HER4	108	7
HIPK1	100	18
HIPK2	102	10
HIPK3	95	8
IGF-1R	94	8
IKK beta	103	14
IKK epsilon	88	16
IR	87	0
IRAK1	94	7
IRAK4	92	21
IRR	103	14
JAK2	92	2
JNK1	106	15
JNK2	93	6
JNK3	96	3
Lck	107	3
LKB1	116	8
MAP4K3	74	11
MAP4K5	82	14
MAPKAP-K2	102	5
MAPKAP-K3	96	3
MARK1	83	3
MARK2	92	5
MARK3	99	4
MARK4	118	51
MEKK1	99	20
MELK	72	10
MINK1	86	9
MKK1	96	4
MKK2	81	5
MKK6	102	10
MLK1	102	1
MLK3	98	5
MNK1	99	8
MNK2	112	27
MPSK1	107	27
MSK1	97	14
MST2	76	4
MST3	108	6
MST4	91	16
NEK2a	102	6
NEK6	100	9
NUAK1	85	4
OSR1	109	10
p38 alpha MAPK	85	8
p38 beta MAPK	113	10
p38 delta MAPK	103	10
p38 gamma MAPK	100	8
PAK2	104	7
PAK4	96	1
PAK5	95	11
PAK6	108	11
PDGFRA	102	9
PDK1	100	1
PHK	92	5
PIM1	98	2
PIM2	99	4
PIM3	90	1
PINK	103	0
PKA	93	5
PKB alpha	94	6
PKB beta	93	14
PKC alpha	88	0
PKC gamma	100	19
PKC zeta	98	4
PKD1	82	7
PLK1	92	5
PRAK	107	11
PRK2	99	2
RIPK2	97	10
ROCK 2	93	5
RSK1	83	3
RSK2	125	0
S6K1	88	17
SGK1	85	23
SIK2	127	31
SIK3	87	2
SmMLCK	101	8
Src	87	0
SRPK1	90	3
STK33	106	18
SYK	95	16
TAK1	101	16
TAO1	98	7
TBK1	99	3
TESK1	90	14
TGFBR1	101	2
TIE2	90	4
TLK1	123	31
TrkA	103	17
TSSK1	61	11
TTBK1	103	1
TTBK2	97	5
TTK	98	3
ULK1	98	5
ULK2	102	4
VEGFR1	63	7
WNK1	115	5
YES1	92	5
ZAP70	100	12

Screen Conc: 10.00µM

Kinase	% Activity Remaining	Standard Deviation
ABL	95	1
AMPK (hum)	94	1
ASK1	107	14
Aurora A	105	4
Aurora B	67	8
BRK	106	3
BRSK1	95	14
BRSK2	70	4
BTK	87	2
CAMK1	92	14
CAMKK beta	103	0
CDK2-Cyclin A	87	5
CDK9-Cyclin T1	97	18
CHK1	92	3
CHK2	81	11
CK1 delta	27	2
CK1 gamma 2	67	2
CK2	108	15
CLK2	83	2
CSK	90	4
DAPK1	93	8
DDR2	110	8
DYRK1A	100	12
DYRK2	81	10
DYRK3	99	7
EF2K	98	0
EIF2AK3	107	8
EPH-A2	95	11
EPH-A4	105	19
EPH-B1	118	14
EPH-B2	92	13
EPH-B3	94	8
EPH-B4	118	10
ERK1	75	3
ERK2	95	2
ERK5	85	13
ERK8	70	3
FGF-R1	74	6
GCK	88	10
GSK3 beta	107	5
HER4	110	9
HIPK1	100	14
HIPK2	106	22
HIPK3	88	4
IGF-1R	103	3
IKK beta	90	14
IKK epsilon	85	2
IR	66	9
IRAK1	64	5
IRAK4	86	7
IRR	87	10
JAK2	88	6
JNK1	94	1
JNK2	83	3
JNK3	101	1
Lck	85	10
LKB1	88	3
MAP4K3	91	1
MAP4K5	77	1
MAPKAP-K2	99	10
MAPKAP-K3	88	8
MARK1	84	4
MARK2	99	7
MARK3	112	12
MARK4	88	27
MEKK1	89	10
MELK	52	8
MINK1	78	15
MKK1	89	9
MKK2	88	26
MKK6	98	3
MLK1	96	0
MLK3	85	3
MNK1	92	12
MNK2	97	17
MPSK1	88	9
MSK1	102	14
MST2	81	20
MST3	105	5
MST4	92	11
NEK2a	100	3
NEK6	100	6
NUAK1	78	2
OSR1	118	8
p38 alpha MAPK	89	18
p38 beta MAPK	106	6
p38 delta MAPK	96	1
p38 gamma MAPK	95	1
PAK2	101	12
PAK4	94	2
PAK5	94	5
PAK6	94	2
PDGFRA	86	7
PDK1	106	11
PHK	86	1
PIM1	85	2
PIM2	88	7
PIM3	72	8
PINK	98	4
PKA	102	4
PKB alpha	97	4
PKB beta	77	3
PKC alpha	90	3
PKC gamma	77	11
PKC zeta	108	2
PKD1	58	11
PLK1	102	0
PRAK	97	4
PRK2	92	9
RIPK2	85	2
ROCK 2	76	4
RSK1	84	10
RSK2	69	15
S6K1	88	1
SGK1	94	7
SIK2	92	13
SIK3	90	1
SmMLCK	99	0
Src	112	1
SRPK1	89	3
STK33	92	1
SYK	78	5
TAK1	83	2
TAO1	92	2
TBK1	108	9
TESK1	98	4
TGFBR1	101	5
TIE2	90	7
TLK1	94	0
TrkA	96	22
TSSK1	79	3
TTBK1	95	6
TTBK2	100	10
TTK	83	3
ULK1	102	11
ULK2	101	14
VEGFR1	41	8
WNK1	111	2
YES1	103	22
ZAP70	127	12