Compound name | Brutto | MW | CAS | PubChem CID | Action | Reference | Reference |
---|---|---|---|---|---|---|---|
Metformin | C4H11N5 | 129.16 | 1115-70-4 | 4091 | AMP | Ouyang J. (2010) J. Biol. Chem. 2011 Jan. 7 286(1) 1-11 |
Kinase | % Activity Remaining | Standard Deviation |
---|---|---|
ABL | 96 | 2 |
AMPK (hum) | 92 | 5 |
ASK1 | 98 | 0 |
Aurora A | 102 | 7 |
Aurora B | 76 | 4 |
BRK | 81 | 1 |
BRSK1 | 88 | 1 |
BRSK2 | 81 | 0 |
BTK | 78 | 32 |
CAMK1 | 86 | 10 |
CAMKK beta | 92 | 7 |
CDK2-Cyclin A | 96 | 2 |
CDK9-Cyclin T1 | 78 | 7 |
CHK1 | 93 | 1 |
CHK2 | 97 | 4 |
CK1 delta | 89 | 2 |
CK1 gamma 2 | 91 | 9 |
CK2 | 88 | 1 |
CLK2 | 94 | 12 |
CSK | 88 | 1 |
DAPK1 | 91 | 1 |
DDR2 | 109 | 10 |
DYRK1A | 89 | 18 |
DYRK2 | 91 | 9 |
DYRK3 | 97 | 4 |
EF2K | 86 | 0 |
EIF2AK3 | 82 | 1 |
EPH-A2 | 81 | 4 |
EPH-A4 | 89 | 10 |
EPH-B1 | 82 | 5 |
EPH-B2 | 99 | 1 |
EPH-B3 | 93 | 2 |
EPH-B4 | 63 | 5 |
ERK1 | 95 | 2 |
ERK2 | 96 | 1 |
ERK5 | 87 | 1 |
ERK8 | 85 | 8 |
FGF-R1 | 79 | 2 |
GCK | 87 | 4 |
GSK3 beta | 88 | 7 |
HER4 | 77 | 17 |
HIPK1 | 90 | 1 |
HIPK2 | 94 | 1 |
HIPK3 | 96 | 8 |
IGF-1R | 129 | 7 |
IKK beta | 97 | 0 |
IKK epsilon | 86 | 6 |
IR | 95 | 4 |
IRAK1 | 111 | 3 |
IRAK4 | 134 | 59 |
IRR | 97 | 2 |
JAK2 | 85 | 3 |
JNK1 | 90 | 8 |
JNK2 | 75 | 1 |
JNK3 | 92 | 14 |
Lck | 97 | 10 |
LKB1 | 95 | 26 |
MAP4K3 | 94 | 17 |
MAP4K5 | 91 | 15 |
MAPKAP-K2 | 93 | 1 |
MAPKAP-K3 | 91 | 7 |
MARK1 | 93 | 12 |
MARK2 | 98 | 4 |
MARK3 | 95 | 8 |
MARK4 | 94 | 9 |
MEKK1 | 92 | 6 |
MELK | 100 | 14 |
MINK1 | 74 | 9 |
MKK1 | 90 | 6 |
MKK2 | 98 | 9 |
MKK6 | 79 | 3 |
MLK1 | 92 | 3 |
MLK3 | 83 | 1 |
MNK1 | 92 | 3 |
MNK2 | 98 | 11 |
MPSK1 | 87 | 3 |
MSK1 | 92 | 11 |
MST2 | 107 | 13 |
MST3 | 88 | 2 |
MST4 | 97 | 7 |
NEK2a | 106 | 9 |
NEK6 | 88 | 34 |
NUAK1 | 81 | 16 |
OSR1 | 97 | 16 |
p38 alpha MAPK | 80 | 1 |
p38 beta MAPK | 101 | 6 |
p38 delta MAPK | 89 | 4 |
p38 gamma MAPK | 85 | 3 |
PAK2 | 98 | 1 |
PAK4 | 91 | 19 |
PAK5 | 102 | 6 |
PAK6 | 107 | 9 |
PDGFRA | 97 | 3 |
PDK1 | 90 | 6 |
PHK | 103 | 6 |
PIM1 | 103 | 1 |
PIM2 | 103 | 15 |
PIM3 | 89 | 1 |
PINK | 96 | 6 |
PKA | 94 | 9 |
PKB alpha | 101 | 2 |
PKB beta | 96 | 4 |
PKC alpha | 118 | 24 |
PKC gamma | 88 | 9 |
PKC zeta | 104 | 7 |
PKD1 | 89 | 0 |
PLK1 | 95 | 8 |
PRAK | 104 | 7 |
PRK2 | 96 | 3 |
RIPK2 | 95 | 4 |
ROCK 2 | 89 | 4 |
RSK1 | 88 | 11 |
RSK2 | 84 | 3 |
S6K1 | 97 | 6 |
SGK1 | 88 | 1 |
SIK2 | 90 | 1 |
SIK3 | 94 | 10 |
SmMLCK | 93 | 1 |
Src | 87 | 8 |
SRPK1 | 82 | 3 |
STK33 | 94 | 9 |
SYK | 74 | 10 |
TAK1 | 96 | 1 |
TAO1 | 87 | 14 |
TBK1 | 81 | 4 |
TESK1 | 96 | 1 |
TGFBR1 | 93 | 2 |
TIE2 | 90 | 7 |
TLK1 | 90 | 5 |
TrkA | 80 | 11 |
TSSK1 | 81 | 4 |
TTBK1 | 93 | 5 |
TTBK2 | 91 | 4 |
TTK | 108 | 6 |
ULK1 | 93 | 3 |
ULK2 | 106 | 6 |
VEGFR1 | 89 | 6 |
WNK1 | 92 | 20 |
YES1 | 96 | 14 |
ZAP70 | 89 | 1 |
Kinase | % Activity Remaining | Standard Deviation |
---|---|---|
ABL | 94 | 11 |
AMPK (hum) | 97 | 9 |
ASK1 | 97 | 1 |
Aurora A | 100 | 5 |
Aurora B | 83 | 5 |
BRK | 90 | 2 |
BRSK1 | 95 | 4 |
BRSK2 | 93 | 1 |
BTK | 74 | 27 |
CAMK1 | 86 | 5 |
CAMKK beta | 88 | 4 |
CDK2-Cyclin A | 113 | 0 |
CDK9-Cyclin T1 | 92 | 0 |
CHK1 | 93 | 2 |
CHK2 | 93 | 2 |
CK1 delta | 87 | 3 |
CK1 gamma 2 | 104 | 10 |
CK2 | 100 | 4 |
CLK2 | 89 | 3 |
CSK | 92 | 3 |
DAPK1 | 93 | 1 |
DDR2 | 99 | 6 |
DYRK1A | 93 | 2 |
DYRK2 | 84 | 3 |
DYRK3 | 109 | 5 |
EF2K | 101 | 5 |
EIF2AK3 | 87 | 5 |
EPH-A2 | 104 | 24 |
EPH-A4 | 95 | 10 |
EPH-B1 | 98 | 5 |
EPH-B2 | 112 | 8 |
EPH-B3 | 103 | 4 |
EPH-B4 | 77 | 3 |
ERK1 | 102 | 10 |
ERK2 | 100 | 11 |
ERK5 | 94 | 2 |
ERK8 | 101 | 2 |
FGF-R1 | 82 | 4 |
GCK | 95 | 1 |
GSK3 beta | 93 | 14 |
HER4 | 81 | 0 |
HIPK1 | 93 | 8 |
HIPK2 | 112 | 18 |
HIPK3 | 107 | 12 |
IGF-1R | 122 | 5 |
IKK beta | 96 | 6 |
IKK epsilon | 82 | 3 |
IR | 94 | 4 |
IRAK1 | 111 | 3 |
IRAK4 | 98 | 3 |
IRR | 97 | 7 |
JAK2 | 73 | 5 |
JNK1 | 99 | 2 |
JNK2 | 92 | 7 |
JNK3 | 100 | 8 |
Lck | 89 | 1 |
LKB1 | 113 | 7 |
MAP4K3 | 87 | 1 |
MAP4K5 | 95 | 10 |
MAPKAP-K2 | 107 | 17 |
MAPKAP-K3 | 95 | 12 |
MARK1 | 94 | 3 |
MARK2 | 101 | 3 |
MARK3 | 95 | 17 |
MARK4 | 93 | 2 |
MEKK1 | 89 | 11 |
MELK | 95 | 1 |
MINK1 | 75 | 4 |
MKK1 | 78 | 10 |
MKK2 | 101 | 13 |
MKK6 | 78 | 1 |
MLK1 | 106 | 17 |
MLK3 | 83 | 2 |
MNK1 | 95 | 3 |
MNK2 | 93 | 3 |
MPSK1 | 95 | 4 |
MSK1 | 104 | 7 |
MST2 | 112 | 5 |
MST3 | 98 | 1 |
MST4 | 107 | 11 |
NEK2a | 101 | 5 |
NEK6 | 84 | 7 |
NUAK1 | 93 | 18 |
OSR1 | 99 | 6 |
p38 alpha MAPK | 93 | 8 |
p38 beta MAPK | 100 | 4 |
p38 delta MAPK | 101 | 5 |
p38 gamma MAPK | 87 | 11 |
PAK2 | 103 | 9 |
PAK4 | 88 | 1 |
PAK5 | 91 | 8 |
PAK6 | 95 | 10 |
PDGFRA | 92 | 1 |
PDK1 | 100 | 6 |
PHK | 100 | 3 |
PIM1 | 94 | 1 |
PIM2 | 99 | 13 |
PIM3 | 90 | 4 |
PINK | 108 | 3 |
PKA | 97 | 4 |
PKB alpha | 98 | 1 |
PKB beta | 108 | 4 |
PKC alpha | 91 | 5 |
PKC gamma | 103 | 9 |
PKC zeta | 99 | 6 |
PKD1 | 94 | 6 |
PLK1 | 128 | 11 |
PRAK | 100 | 5 |
PRK2 | 95 | 6 |
RIPK2 | 107 | 4 |
ROCK 2 | 94 | 2 |
RSK1 | 94 | 13 |
RSK2 | 83 | 1 |
S6K1 | 102 | 2 |
SGK1 | 102 | 1 |
SIK2 | 96 | 3 |
SIK3 | 87 | 5 |
SmMLCK | 91 | 3 |
Src | 86 | 3 |
SRPK1 | 95 | 1 |
STK33 | 100 | 11 |
SYK | 80 | 5 |
TAK1 | 101 | 10 |
TAO1 | 104 | 7 |
TBK1 | 86 | 4 |
TESK1 | 86 | 7 |
TGFBR1 | 100 | 11 |
TIE2 | 82 | 10 |
TLK1 | 96 | 4 |
TrkA | 78 | 11 |
TSSK1 | 90 | 0 |
TTBK1 | 92 | 3 |
TTBK2 | 90 | 10 |
TTK | 108 | 14 |
ULK1 | 97 | 10 |
ULK2 | 110 | 2 |
VEGFR1 | 89 | 4 |
WNK1 | 97 | 14 |
YES1 | 96 | 17 |
ZAP70 | 93 | 0 |