

Compound name | Brutto | MW | CAS | PubChem CID | Action | Reference | Reference |
---|---|---|---|---|---|---|---|
Amgen-NIK-28 | C20H20N4O | 332.40 | NIK | Li K. (2013) Bioorganic and Medicinal Chemistry Letters 23 1238-1244 |
Kinase | % Activity Remaining | Standard Deviation |
---|---|---|
ABL | 104 | 13 |
AMPK (hum) | 109 | 14 |
ASK1 | 110 | 1 |
Aurora A | 102 | 5 |
Aurora B | 90 | 5 |
BRK | 98 | 4 |
BRSK1 | 94 | 1 |
BRSK2 | 101 | 0 |
BTK | 113 | 2 |
CAMK1 | 98 | 19 |
CAMKK beta | 94 | 7 |
CDK2-Cyclin A | 101 | 1 |
CDK9-Cyclin T1 | 100 | 3 |
CHK1 | 105 | 3 |
CHK2 | 65 | 5 |
CK1 delta | 45 | 6 |
CK1 gamma 2 | 103 | 3 |
CK2 | 100 | 9 |
CLK2 | 73 | 3 |
CSK | 124 | 3 |
DAPK1 | 97 | 14 |
DDR2 | 92 | 10 |
DYRK1A | 93 | 12 |
DYRK2 | 91 | 0 |
DYRK3 | 88 | 6 |
EF2K | 97 | 4 |
EIF2AK3 | 71 | 7 |
EPH-A2 | 82 | 7 |
EPH-A4 | 106 | 21 |
EPH-B1 | 105 | 6 |
EPH-B2 | 124 | 7 |
EPH-B3 | 87 | 2 |
EPH-B4 | 89 | 2 |
ERK1 | 97 | 8 |
ERK2 | 115 | 5 |
ERK5 | 81 | 2 |
ERK8 | 96 | 0 |
FGF-R1 | 101 | 14 |
GCK | 99 | 0 |
GSK3 beta | 85 | 2 |
HER4 | 104 | 4 |
HIPK1 |
7
|
0 |
HIPK2 | 77 | 5 |
HIPK3 | 100 | 1 |
IGF-1R | 106 | 21 |
IKK beta | 95 | 18 |
IKK epsilon | 87 | 5 |
IR | 96 | 8 |
IRAK1 | 103 | 8 |
IRAK4 | 75 | 6 |
IRR | 116 | 6 |
JAK2 | 39 | 4 |
JNK1 | 86 | 4 |
JNK2 | 85 | 12 |
JNK3 | 93 | 14 |
Lck | 97 | 5 |
LKB1 | 92 | 15 |
MAP4K3 | 11 | 3 |
MAP4K5 |
5
|
0 |
MAPKAP-K2 | 108 | 10 |
MAPKAP-K3 | 94 | 21 |
MARK1 | 76 | 16 |
MARK2 | 72 | 4 |
MARK3 | 41 | 6 |
MARK4 | 79 | 0 |
MEKK1 | 96 | 1 |
MELK | 87 | 13 |
MINK1 | 58 | 4 |
MKK1 | 57 | 3 |
MKK2 | 75 | 6 |
MKK6 | 79 | 16 |
MLK1 | 30 | 4 |
MLK3 | 12 | 1 |
MNK1 | 89 | 0 |
MNK2 | 95 | 1 |
MPSK1 | 104 | 0 |
MSK1 | 105 | 13 |
MST2 | 99 | 1 |
MST3 | 99 | 2 |
MST4 | 107 | 1 |
NEK2a | 105 | 3 |
NEK6 | 103 | 21 |
NUAK1 | 77 | 6 |
OSR1 | 83 | 1 |
p38 alpha MAPK | 117 | 13 |
p38 beta MAPK | 95 | 5 |
p38 delta MAPK | 86 | 1 |
p38 gamma MAPK | 76 | 0 |
PAK2 | 110 | 2 |
PAK4 | 13 | 3 |
PAK5 | 16 | 1 |
PAK6 | 29 | 1 |
PDGFRA | 88 | 4 |
PDK1 | 111 | 11 |
PHK | 97 | 5 |
PIM1 | 108 | 3 |
PIM2 | 115 | 10 |
PIM3 | 109 | 0 |
PINK | 110 | 6 |
PKA | 102 | 1 |
PKB alpha | 91 | 1 |
PKB beta | 90 | 2 |
PKC alpha | 102 | 15 |
PKC gamma | 105 | 3 |
PKC zeta | 93 | 5 |
PKD1 | 42 | 1 |
PLK1 | 104 | 16 |
PRAK | 109 | 12 |
PRK2 | 95 | 3 |
RIPK2 | 88 | 4 |
ROCK 2 | 97 | 1 |
RSK1 | 83 | 20 |
RSK2 | 89 | 5 |
S6K1 | 97 | 12 |
SGK1 | 110 | 1 |
SIK2 | 81 | 3 |
SIK3 | 103 | 13 |
SmMLCK | 85 | 1 |
Src | 107 | 0 |
SRPK1 | 97 | 10 |
STK33 | 87 | 8 |
SYK | 108 | 4 |
TAK1 | 29 | 1 |
TAO1 | 30 | 0 |
TBK1 | 104 | 2 |
TESK1 | 105 | 3 |
TGFBR1 | 83 | 1 |
TIE2 | 113 | 11 |
TLK1 | 101 | 4 |
TrkA | 127 | 6 |
TSSK1 | 49 | 2 |
TTBK1 | 47 | 10 |
TTBK2 | 52 | 10 |
TTK | 109 | 0 |
ULK1 | 89 | 14 |
ULK2 | 79 | 13 |
VEGFR1 | 67 | 5 |
WNK1 | 107 | 3 |
YES1 | 118 | 8 |
ZAP70 | 98 | 3 |
Kinase | % Activity Remaining | Standard Deviation |
---|---|---|
ABL | 95 | 7 |
AMPK (hum) | 71 | 5 |
ASK1 | 101 | 6 |
Aurora A | 107 | 1 |
Aurora B | 72 | 3 |
BRK | 87 | 4 |
BRSK1 | 91 | 5 |
BRSK2 | 84 | 7 |
BTK | 117 | 21 |
CAMK1 | 69 | 12 |
CAMKK beta | 99 | 2 |
CDK2-Cyclin A | 97 | 21 |
CDK9-Cyclin T1 | 126 | 1 |
CHK1 | 102 | 5 |
CHK2 | 16 | 3 |
CK1 delta | 15 | 3 |
CK1 gamma 2 | 92 | 1 |
CK2 | 90 | 3 |
CLK2 | 27 | 5 |
CSK | 119 | 19 |
DAPK1 | 82 | 1 |
DDR2 | 104 | 4 |
DYRK1A | 72 | 13 |
DYRK2 | 76 | 1 |
DYRK3 | 61 | 2 |
EF2K | 83 | 9 |
EIF2AK3 | 24 | 4 |
EPH-A2 | 90 | 2 |
EPH-A4 | 119 | 30 |
EPH-B1 | 101 | 11 |
EPH-B2 | 131 | 16 |
EPH-B3 | 87 | 3 |
EPH-B4 | 98 | 1 |
ERK1 | 96 | 6 |
ERK2 | 95 | 5 |
ERK5 | 47 | 3 |
ERK8 | 85 | 0 |
FGF-R1 | 62 | 2 |
GCK | 37 | 1 |
GSK3 beta | 30 | 2 |
HER4 | 108 | 10 |
HIPK1 |
3
|
0 |
HIPK2 | 39 | 2 |
HIPK3 | 86 | 26 |
IGF-1R | 118 | 8 |
IKK beta | 82 | 4 |
IKK epsilon | 28 | 10 |
IR | 72 | 5 |
IRAK1 | 97 | 7 |
IRAK4 | 53 | 10 |
IRR | 103 | 9 |
JAK2 |
10
|
2 |
JNK1 | 86 | 17 |
JNK2 | 86 | 6 |
JNK3 | 89 | 10 |
Lck | 94 | 6 |
LKB1 | 81 | 6 |
MAP4K3 |
2
|
1 |
MAP4K5 |
5
|
1 |
MAPKAP-K2 | 108 | 10 |
MAPKAP-K3 | 104 | 7 |
MARK1 | 38 | 15 |
MARK2 | 42 | 1 |
MARK3 |
10
|
1 |
MARK4 | 39 | 3 |
MEKK1 | 94 | 2 |
MELK | 71 | 2 |
MINK1 | 16 | 0 |
MKK1 | 22 | 2 |
MKK2 | 39 | 7 |
MKK6 | 46 | 24 |
MLK1 |
5
|
0 |
MLK3 |
2
|
0 |
MNK1 | 108 | 4 |
MNK2 | 92 | 1 |
MPSK1 | 89 | 7 |
MSK1 | 102 | 7 |
MST2 | 65 | 2 |
MST3 | 72 | 2 |
MST4 | 63 | 3 |
NEK2a | 92 | 5 |
NEK6 | 92 | 13 |
NUAK1 | 33 | 3 |
OSR1 | 88 | 8 |
p38 alpha MAPK | 113 | 7 |
p38 beta MAPK | 100 | 0 |
p38 delta MAPK | 88 | 6 |
p38 gamma MAPK | 34 | 1 |
PAK2 | 96 | 11 |
PAK4 |
2
|
2 |
PAK5 |
3
|
1 |
PAK6 |
5
|
1 |
PDGFRA | 96 | 13 |
PDK1 | 101 | 1 |
PHK | 80 | 3 |
PIM1 | 92 | 5 |
PIM2 | 108 | 7 |
PIM3 | 89 | 3 |
PINK | 102 | 4 |
PKA | 89 | 2 |
PKB alpha | 54 | 1 |
PKB beta | 46 | 4 |
PKC alpha | 102 | 7 |
PKC gamma | 97 | 2 |
PKC zeta | 89 | 8 |
PKD1 |
9
|
3 |
PLK1 | 103 | 1 |
PRAK | 103 | 10 |
PRK2 | 86 | 6 |
RIPK2 | 73 | 5 |
ROCK 2 | 94 | 1 |
RSK1 | 81 | 15 |
RSK2 | 94 | 4 |
S6K1 | 101 | 8 |
SGK1 | 68 | 0 |
SIK2 | 77 | 5 |
SIK3 | 87 | 10 |
SmMLCK | 31 | 0 |
Src | 82 | 10 |
SRPK1 | 94 | 17 |
STK33 | 52 | 0 |
SYK | 117 | 7 |
TAK1 |
6
|
0 |
TAO1 |
7
|
2 |
TBK1 | 90 | 5 |
TESK1 | 97 | 4 |
TGFBR1 | 84 | 9 |
TIE2 | 97 | 12 |
TLK1 | 99 | 17 |
TrkA | 115 | 11 |
TSSK1 | 13 | 0 |
TTBK1 |
8
|
1 |
TTBK2 | 12 | 5 |
TTK | 100 | 1 |
ULK1 | 81 | 16 |
ULK2 | 61 | 7 |
VEGFR1 | 22 | 2 |
WNK1 | 103 | 15 |
YES1 | 107 | 14 |
ZAP70 | 103 | 11 |