Inhibitor | Chloroquine  

Screen Conc: 1.00µM

Kinase	% Activity Remaining Sort descending	Standard Deviation
PHK	76	4
NEK2a	79	5
IKK epsilon	79	2
PKC alpha	81	24
TIE2	84	1
YES1	85	4
MST3	85	19
BRK	88	8
TSSK1	89	8
PRAK	89	18
PKB beta	90	1
HIPK3	91	11
EPH-A4	92	9
MNK2	92	24
MAPKAP-K2	92	13
ZAP70	92	3
BRSK1	94	7
MINK1	94	5
MNK1	95	33
ULK2	95	37
CK1 delta	96	2
TBK1	97	15
ERK8	97	6
MKK2	97	16
PKA	98	1
CHK1	98	3
IRR	98	8
CDK9-Cyclin T1	99	28
PIM1	99	3
CK2	99	8
ERK5	100	2
BRSK2	100	24
PIM3	100	1
JNK1	101	3
ASK1	101	15
PAK5	101	11
PIM2	101	19
CAMK1	102	5
MARK2	102	20
MST4	102	3
EPH-B2	102	7
TLK1	102	8
EPH-B3	102	7
S6K1	103	12
PDGFRA	103	7
CSK	103	7
p38 alpha MAPK	103	12
IKK beta	103	9
DYRK2	104	0
VEGFR1	104	8
p38 delta MAPK	105	16
MPSK1	105	1
WNK1	105	5
TrkA	105	2
AMPK (hum)	106	4
ERK2	106	8
MAP4K5	106	13
SmMLCK	107	16
MSK1	107	8
PKB alpha	107	12
TTBK2	108	1
MELK	108	15
ABL	108	6
OSR1	108	12
TTK	108	2
Aurora A	108	7
MKK1	108	24
DDR2	108	3
MLK3	109	7
Lck	109	15
PINK	109	9
PAK4	109	3
IRAK4	109	7
CK1 gamma 2	109	0
ERK1	110	3
DAPK1	110	15
NEK6	110	4
CLK2	111	1
PRK2	111	16
PAK6	111	2
IR	111	6
MEKK1	111	11
AMPK	111	17
TTBK1	111	3
DYRK1A	112	2
MARK3	112	1
PKC gamma	112	1
CAMKK beta	113	16
DYRK3	113	14
IRAK1	113	7
p38 gamma MAPK	113	1
GCK	113	3
RSK1	113	4
RSK2	113	1
MAPKAP-K3	113	6
EIF2AK3	113	7
TAO1	114	6
MARK4	114	4
CDK2-Cyclin A	114	19
JAK2	114	8
SRPK1	114	20
LKB1	114	10
SGK1	115	2
HER4	115	22
TAK1	115	1
PLK1	115	23
HIPK1	115	13
MLK1	115	9
EPH-B4	115	6
FGF-R1	116	20
HIPK2	117	4
TESK1	117	18
RIPK2	117	9
BTK	117	26
EPH-B1	117	17
SYK	117	7
MARK1	118	2
STK33	118	15
PAK2	119	12
EPH-A2	119	11
p38 beta MAPK	119	25
Aurora B	119	8
JNK2	120	6
JNK3	120	16
MST2	120	2
PDK1	120	6
SIK2	121	1
SIK3	121	14
ULK1	121	4
MAP4K3	122	22
MKK6	122	22
ROCK 2	123	3
NUAK1	123	22
TGFBR1	123	13
IGF-1R	126	30
PKC zeta	126	19
GSK3 beta	127	12
EF2K	127	15
Src	127	13
CHK2	128	24
PKD1	133	19

Screen Conc: 10.00µM

Kinase	% Activity Remaining Sort descending	Standard Deviation
IKK beta	76	4
TIE2	81	8
PHK	83	26
PRAK	84	7
DYRK2	89	0
PIM1	90	6
LKB1	90	7
PAK4	91	9
CK1 delta	92	5
BRSK1	93	22
DAPK1	94	7
S6K1	94	1
p38 alpha MAPK	95	13
TBK1	96	11
PIM3	96	2
MARK1	96	9
MARK3	97	14
EPH-B4	97	21
PAK5	97	9
PKB alpha	98	1
MST3	98	5
IRAK1	99	2
CDK2-Cyclin A	99	8
TrkA	99	15
EPH-B2	100	11
MKK1	100	17
CSK	100	5
IKK epsilon	100	22
YES1	100	7
IR	100	11
JNK1	100	9
EPH-A2	100	9
EPH-A4	100	8
MARK4	101	5
NEK2a	101	31
ABL	101	10
MSK1	101	3
ERK2	101	3
HIPK3	101	11
NEK6	102	0
ZAP70	102	2
PKA	102	8
PKC alpha	103	10
ASK1	103	5
p38 delta MAPK	103	1
TLK1	103	7
PRK2	103	3
SmMLCK	103	20
ULK2	104	2
MELK	104	10
ERK8	104	5
BRK	104	6
CAMKK beta	104	14
MLK3	104	4
CAMK1	104	5
Src	105	2
TSSK1	105	6
MAPKAP-K3	105	18
AMPK (hum)	105	4
TAO1	105	11
DYRK3	106	8
CHK1	106	10
p38 beta MAPK	106	10
MST4	106	2
IRR	106	27
MST2	107	3
EIF2AK3	107	12
HIPK1	107	9
JNK2	107	13
DYRK1A	107	8
BRSK2	108	19
ERK1	108	7
p38 gamma MAPK	108	9
MEKK1	108	5
MPSK1	108	15
ULK1	108	11
MARK2	108	6
EPH-B3	109	3
Lck	109	16
NUAK1	109	5
SGK1	109	14
ERK5	109	12
MAPKAP-K2	109	1
PINK	109	23
MLK1	109	1
CLK2	109	5
VEGFR1	110	15
OSR1	110	13
PDGFRA	110	6
TTK	110	1
PKC gamma	111	1
FGF-R1	111	8
PAK6	111	4
PIM2	111	26
Aurora A	111	27
SYK	111	1
SRPK1	111	1
RSK1	111	5
AMPK	111	19
PDK1	112	0
IRAK4	112	3
IGF-1R	112	25
CK1 gamma 2	112	5
MINK1	112	17
TTBK2	112	0
SIK2	114	8
MAP4K3	114	16
ROCK 2	114	1
MKK2	115	21
GCK	115	9
MNK1	115	0
RIPK2	115	2
JNK3	116	10
TAK1	116	1
GSK3 beta	116	3
MAP4K5	116	11
PKB beta	117	37
DDR2	117	5
RSK2	117	2
PAK2	118	7
TGFBR1	118	18
TESK1	118	15
CHK2	119	28
HER4	119	23
JAK2	119	17
CK2	119	3
WNK1	119	3
PKC zeta	121	6
STK33	121	24
CDK9-Cyclin T1	121	12
PLK1	121	2
MNK2	123	5
BTK	124	8
EF2K	124	5
TTBK1	124	2
SIK3	125	7
EPH-B1	125	27
Aurora B	126	2
HIPK2	128	4
PKD1	129	44
MKK6	130	15