Inhibitor | 2-Aminopurine
Compound name |
Brutto |
MW |
CAS |
PubChem CID |
Action |
Reference |
Reference |
2-Aminopurine |
C5H5N5 |
135.13 |
452-06-2 |
9955 |
PKR |
|
|
Screening Results Tables
Screen Conc: 100.00µM
Kinase |
% Activity Remaining |
Standard Deviation |
ABL |
83
|
7 |
AMPK |
73
|
6 |
AMPK (hum) |
80
|
11 |
ASK1 |
44
|
3 |
Aurora A |
64
|
3 |
Aurora B |
23
|
2 |
BRK |
47
|
5 |
BRSK1 |
79
|
8 |
BRSK2 |
81
|
3 |
BTK |
67
|
3 |
CAMK1 |
85
|
5 |
CAMKK beta |
87
|
1 |
CDK2-Cyclin A |
81
|
2 |
CDK9-Cyclin T1 |
72
|
9 |
CHK1 |
57
|
9 |
CHK2 |
21
|
0 |
CK1 delta |
24
|
4 |
CK1 gamma 2 |
16
|
1 |
CK2 |
89
|
5 |
CLK2 |
37
|
4 |
CSK |
91
|
17 |
DAPK1 |
77
|
7 |
DDR2 |
82
|
11 |
DYRK1A |
64
|
3 |
DYRK2 |
68
|
6 |
DYRK3 |
72
|
5 |
EF2K |
88
|
3 |
EIF2AK3 |
89
|
0 |
EPH-A2 |
83
|
1 |
EPH-A4 |
84
|
4 |
EPH-B1 |
108
|
7 |
EPH-B2 |
95
|
10 |
EPH-B3 |
105
|
36 |
EPH-B4 |
90
|
10 |
ERK1 |
78
|
8 |
ERK2 |
78
|
0 |
ERK5 |
67
|
1 |
ERK8 |
79
|
10 |
FGF-R1 |
109
|
18 |
GCK |
20
|
0 |
GSK3 beta |
89
|
12 |
HER4 |
72
|
0 |
HIPK1 |
104
|
15 |
HIPK2 |
76
|
2 |
HIPK3 |
92
|
2 |
IGF-1R |
75
|
23 |
IKK beta |
55
|
4 |
IKK epsilon |
62
|
5 |
IR |
106
|
8 |
IRAK1 |
65
|
10 |
IRAK4 |
76
|
7 |
IRR |
73
|
5 |
JAK2 |
30
|
0 |
JNK1 |
81
|
6 |
JNK2 |
83
|
8 |
JNK3 |
83
|
6 |
Lck |
79
|
3 |
LKB1 |
82
|
9 |
MAP4K3 |
50
|
6 |
MAP4K5 |
67
|
3 |
MAPKAP-K2 |
40
|
3 |
MAPKAP-K3 |
70
|
3 |
MARK1 |
67
|
0 |
MARK2 |
69
|
2 |
MARK3 |
61
|
5 |
MARK4 |
74
|
5 |
MEKK1 |
78
|
0 |
MELK |
63
|
2 |
MINK1 |
63
|
3 |
MKK1 |
56
|
5 |
MKK2 |
63
|
2 |
MKK6 |
91
|
6 |
MLK1 |
29
|
6 |
MLK3 |
18
|
5 |
MNK1 |
67
|
7 |
MNK2 |
75
|
2 |
MPSK1 |
89
|
4 |
MSK1 |
84
|
4 |
MST2 |
63
|
1 |
MST3 |
81
|
2 |
MST4 |
72
|
3 |
NEK2a |
60
|
14 |
NEK6 |
88
|
10 |
NUAK1 |
33
|
0 |
OSR1 |
80
|
7 |
p38 alpha MAPK |
85
|
4 |
p38 beta MAPK |
83
|
0 |
p38 delta MAPK |
97
|
6 |
p38 gamma MAPK |
75
|
0 |
PAK2 |
100
|
10 |
PAK4 |
44
|
5 |
PAK5 |
64
|
0 |
PAK6 |
82
|
5 |
PDGFRA |
79
|
3 |
PDK1 |
67
|
1 |
PHK |
76
|
2 |
PIM1 |
122
|
0 |
PIM2 |
102
|
7 |
PIM3 |
76
|
4 |
PINK |
90
|
11 |
PKA |
93
|
7 |
PKB alpha |
99
|
5 |
PKB beta |
83
|
7 |
PKC alpha |
104
|
27 |
PKC gamma |
84
|
6 |
PKC zeta |
78
|
3 |
PKD1 |
65
|
7 |
PLK1 |
76
|
1 |
PRAK |
75
|
0 |
PRK2 |
73
|
8 |
RIPK2 |
43
|
1 |
ROCK 2 |
64
|
2 |
RSK1 |
81
|
2 |
RSK2 |
79
|
8 |
S6K1 |
85
|
15 |
SGK1 |
63
|
1 |
SIK2 |
43
|
2 |
SIK3 |
56
|
2 |
SmMLCK |
75
|
2 |
Src |
73
|
1 |
SRPK1 |
96
|
1 |
STK33 |
67
|
6 |
SYK |
102
|
8 |
TAK1 |
54
|
2 |
TAO1 |
66
|
3 |
TBK1 |
73
|
4 |
TESK1 |
60
|
4 |
TGFBR1 |
101
|
2 |
TIE2 |
85
|
1 |
TLK1 |
108
|
7 |
TrkA |
73
|
13 |
TSSK1 |
44
|
8 |
TTBK1 |
80
|
12 |
TTBK2 |
74
|
6 |
TTK |
82
|
1 |
ULK1 |
57
|
2 |
ULK2 |
69
|
0 |
VEGFR1 |
29
|
3 |
WNK1 |
87
|
2 |
YES1 |
94
|
6 |
ZAP70 |
101
|
4 |