Inhibitor | HG-10-102-01  

Screen Conc: 1.00µM

Kinase	% Activity Remaining Sort ascending	Standard Deviation
IRR	126	5
MAPKAP-K3	120	81
TTBK2	115	11
EPH-B1	115	1
OSR1	108	1
GCK	108	10
MKK1	106	15
EPH-B2	105	7
MSK1	104	8
DDR2	103	16
PRK2	102	12
PDK1	102	11
MST4	101	1
IGF-1R	100	3
GSK3 beta	100	1
MPSK1	100	2
EPH-A4	100	4
PKC zeta	99	10
EIF2AK3	99	19
CSK	97	1
PAK2	97	4
ZAP70	97	4
PLK1	97	23
ULK2	97	9
PIM1	96	8
CK1 gamma 2	96	10
SRPK1	96	1
ERK1	95	16
PKB beta	95	11
PIM2	94	13
MAP4K3	94	11
SGK1	94	3
EPH-B4	94	12
PKC gamma	93	2
EPH-A2	93	9
SIK3	93	6
MEKK1	93	2
Lck	92	4
RSK2	92	7
LKB1	92	1
PRAK	91	0
AMPK (hum)	91	7
MARK1	91	9
CLK2	91	1
MARK3	91	1
MKK2	91	17
TESK1	90	0
PAK6	90	8
IRAK4	90	6
AMPK	89	5
FGF-R1	89	6
HER4	89	4
JNK1	89	8
CDK9-Cyclin T1	89	7
TTBK1	88	8
PAK5	88	3
MELK	88	21
MAPKAP-K2	88	4
p38 gamma MAPK	88	21
p38 delta MAPK	87	0
ROCK 2	87	7
RSK1	87	10
PAK4	87	1
IR	86	4
TBK1	86	3
MINK1	86	4
CAMK1	85	1
HIPK3	85	0
PKA	85	10
MARK2	85	7
MST2	85	17
ABL	84	7
DYRK3	84	1
IRAK1	84	21
Src	84	6
SmMLCK	83	1
BTK	83	8
JAK2	83	8
MST3	83	9
Aurora B	83	1
MAP4K5	83	7
EF2K	83	3
MARK4	82	7
IKK beta	82	2
CDK2-Cyclin A	82	2
TAO1	81	22
YES1	80	3
TrkA	80	14
DYRK1A	79	12
ERK2	79	5
RIPK2	79	6
TIE2	79	3
PDGFRA	79	0
BRSK2	78	11
HIPK1	77	10
HIPK2	77	23
IKK epsilon	77	31
PIM3	77	0
JNK2	76	10
MLK3	75	10
ERK8	74	26
TAK1	74	16
MKK6	74	29
NEK6	73	25
TTK	71	0
p38 alpha MAPK	71	8
MNK1	71	11
S6K1	70	15
ASK1	70	3
PKD1	70	5
PHK	68	11
SYK	68	17
EPH-B3	67	2
PKC alpha	66	6
CHK1	65	29
VEGFR1	65	25
NEK2a	63	1
WNK1	62	20
ULK1	62	10
DAPK1	61	13
STK33	61	1
TLK1	61	7
JNK3	60	1
BRSK1	59	18
p38 beta MAPK	57	11
BRK	56	2
Aurora A	56	4
PKB alpha	53	1
CAMKK beta	52	13
CHK2	52	2
TSSK1	51	3
CK2	50	8
SIK2	49	11
DYRK2	44	7
CK1 delta	44	7
NUAK1	43	1
MLK1	38	3
MNK2	20	9

Screen Conc: 10.00µM

Kinase	% Activity Remaining Sort ascending	Standard Deviation
EPH-B4	113	7
PKC gamma	108	6
MST4	106	9
PLK1	105	4
PAK2	105	4
ERK1	104	22
CSK	103	11
EPH-B2	103	8
MAPKAP-K2	102	2
PKC zeta	101	9
EPH-B3	101	17
TLK1	100	9
PIM1	99	0
WNK1	99	6
MEKK1	98	7
PAK6	98	9
GSK3 beta	98	6
MELK	98	3
PIM2	97	13
MPSK1	97	7
EIF2AK3	97	2
EPH-A2	97	4
TTBK2	97	12
IRR	97	9
MINK1	96	14
CHK2	96	15
Lck	95	5
p38 gamma MAPK	94	11
SRPK1	94	22
HER4	94	2
HIPK1	94	7
EPH-A4	94	7
PKA	94	8
p38 alpha MAPK	93	10
CK1 gamma 2	93	2
TAO1	93	4
MKK1	93	7
p38 beta MAPK	93	6
PRK2	92	10
TTBK1	91	4
SGK1	91	1
TIE2	90	0
LKB1	90	8
YES1	90	5
MARK2	90	6
NEK2a	90	13
DDR2	90	16
CK1 delta	89	9
PDK1	89	8
CK2	88	1
HIPK2	88	6
BTK	88	2
PKC alpha	87	9
TrkA	87	1
FGF-R1	86	10
p38 delta MAPK	86	3
EF2K	86	9
ABL	86	9
EPH-B1	86	5
MKK2	86	10
IRAK4	86	3
ULK1	85	2
PKB alpha	85	1
SYK	85	9
MSK1	84	11
ULK2	84	6
MARK1	84	7
PAK4	84	8
CDK9-Cyclin T1	83	3
TESK1	83	15
IRAK1	83	11
SIK3	82	3
MAP4K5	82	7
ERK8	82	5
OSR1	82	10
ZAP70	81	7
MAPKAP-K3	81	2
AMPK	80	1
DYRK1A	80	2
HIPK3	80	5
PAK5	80	0
JAK2	80	18
IKK beta	80	7
RIPK2	80	2
MST3	80	5
GCK	79	11
Src	79	0
MARK3	78	2
BRSK1	78	0
CLK2	76	5
DYRK3	76	3
IKK epsilon	75	2
MST2	73	10
PIM3	72	4
MARK4	72	6
AMPK (hum)	71	6
ROCK 2	71	2
MAP4K3	70	9
NEK6	69	19
ERK2	69	11
S6K1	67	15
CAMK1	66	3
RSK2	65	10
MKK6	65	7
CDK2-Cyclin A	65	4
PKB beta	64	8
BRSK2	64	5
TTK	57	5
PDGFRA	56	1
SmMLCK	55	3
RSK1	54	2
ASK1	54	3
IGF-1R	51	7
IR	50	7
SIK2	47	0
JNK2	46	3
Aurora A	45	9
CHK1	45	4
MNK1	44	6
PRAK	44	1
MLK3	43	9
Aurora B	42	4
TBK1	42	1
BRK	39	1
JNK1	37	2
VEGFR1	35	2
CAMKK beta	31	3
JNK3	29	10
STK33	28	1
TAK1	25	8
PKD1	25	4
PHK	23	4
DAPK1	23	5
DYRK2	21	6
NUAK1	20	6
TSSK1	19	1
MLK1	18	0
MNK2	7	2