Inhibitor | JNKIN7  

Screen Conc: 0.10µM

Kinase	% Activity Remaining	Standard Deviation
ABL	77	9
AMPK	92	12
ASK1	96	9
Aurora A	107	7
Aurora B	74	1
BRK	81	11
BRSK1	94	4
BRSK2	82	8
BTK	86	22
CAMK1	87	12
CAMKK beta	87	10
CDK2-Cyclin A	85	0
CDK9-Cyclin T1	22	4
CHK1	74	17
CHK2	89	2
CK1 delta	63	5
CK1 gamma 2	88	1
CK2	80	1
CLK2	49	2
CSK	109	20
DAPK1	90	8
DDR2	89	7
DYRK1A	97	2
DYRK2	82	20
DYRK3	81	9
EF2K	97	5
EIF2AK3	90	2
EPH-A2	110	7
EPH-A4	92	5
EPH-B1	93	9
EPH-B2	101	9
EPH-B3	101	6
EPH-B4	105	2
ERK1	110	16
ERK2	99	16
ERK8	46	5
FGF-R1	94	19
GCK	45	4
GSK3 beta	88	8
HER4	108	32
HIPK1	86	11
HIPK2	85	10
HIPK3	113	0
IGF-1R	75	22
IKK beta	76	16
IKK epsilon	97	4
IR	81	1
IRAK1	26	14
IRAK4	86	12
IRR	72	1
JAK2	85	10
JNK1	9	2
JNK2	81	8
JNK3	15	2
Lck	95	0
LKB1	78	3
MAPKAP-K2	91	1
MAPKAP-K3	104	9
MARK1	91	9
MARK2	94	1
MARK3	101	5
MARK4	85	3
MEKK1	85	11
MELK	71	0
MINK1	92	9
MKK1	98	6
MKK2	87	19
MKK6	97	13
MLK1	72	0
MLK3	79	1
MNK1	84	16
MNK2	92	5
MPSK1	108	3
MSK1	88	9
MST2	83	10
MST3	94	3
MST4	98	2
NEK2a	93	1
NEK6	88	12
NUAK1	35	1
OSR1	99	2
p38 alpha MAPK	98	0
p38 beta MAPK	96	5
p38 delta MAPK	106	7
p38 gamma MAPK	90	10
PAK2	102	2
PAK4	84	8
PAK5	89	1
PAK6	87	4
PDK1	89	14
PHK	94	10
PIM1	97	3
PIM2	96	8
PIM3	97	6
PKA	97	5
PKB alpha	92	5
PKB beta	93	13
PKC alpha	89	4
PKC gamma	96	4
PKC zeta	112	3
PKD1	105	37
PLK1	91	9
PRAK	96	17
PRK2	99	0
RIPK2	74	21
ROCK 2	89	10
RSK1	95	21
RSK2	80	11
S6K1	88	2
SGK1	105	20
SIK2	78	1
SIK3	81	4
SmMLCK	96	6
Src	93	9
SRPK1	105	16
STK33	92	8
SYK	89	17
TAK1	67	4
TAO1	96	1
TBK1	77	5
TESK1	90	16
TIE2	94	5
TLK1	99	7
TrkA	96	24
TSSK1	88	3
TTBK1	88	13
TTK	83	6
ULK1	37	1
ULK2	50	5
VEGFR1	59	4
WNK1	103	17
YES1	80	17
ZAP70	82	1

Screen Conc: 1.00µM

Kinase	% Activity Remaining	Standard Deviation
ABL	85	12
AMPK	87	4
ASK1	100	1
Aurora A	97	3
Aurora B	73	1
BRK	81	16
BRSK1	86	6
BRSK2	76	6
BTK	85	14
CAMK1	92	4
CAMKK beta	35	4
CDK2-Cyclin A	72	2
CDK9-Cyclin T1	42	2
CHK1	88	2
CHK2	73	1
CK1 delta	33	0
CK1 gamma 2	88	4
CK2	81	10
CLK2	18	5
CSK	103	7
DAPK1	83	2
DDR2	108	9
DYRK1A	85	6
DYRK2	56	2
DYRK3	79	6
EF2K	101	1
EIF2AK3	99	9
EPH-A2	125	17
EPH-A4	105	2
EPH-B1	86	19
EPH-B2	103	10
EPH-B3	118	20
EPH-B4	109	6
ERK1	109	9
ERK2	114	17
ERK8	20	8
FGF-R1	95	14
GCK	20	1
GSK3 beta	56	1
HER4	106	7
HIPK1	78	10
HIPK2	46	4
HIPK3	101	22
IGF-1R	102	8
IKK beta	63	2
IKK epsilon	98	8
IR	77	24
IRAK1	5	0
IRAK4	88	6
IRR	64	6
JAK2	77	8
JNK1	4	1
JNK2	19	9
JNK3	16	0
Lck	101	1
LKB1	91	18
MAPKAP-K2	106	11
MAPKAP-K3	101	4
MARK1	80	1
MARK2	85	2
MARK3	76	2
MARK4	83	16
MEKK1	100	8
MELK	48	1
MINK1	69	2
MKK1	113	9
MKK2	102	13
MKK6	91	0
MLK1	39	0
MLK3	59	8
MNK1	95	23
MNK2	84	21
MPSK1	103	8
MSK1	91	6
MST2	64	6
MST3	93	15
MST4	104	1
NEK2a	105	21
NEK6	96	0
NUAK1	82	10
OSR1	105	7
p38 alpha MAPK	113	3
p38 beta MAPK	82	6
p38 delta MAPK	100	4
p38 gamma MAPK	103	0
PAK2	93	1
PAK4	66	6
PAK5	91	8
PAK6	103	8
PDK1	98	4
PHK	83	0
PIM1	114	6
PIM2	102	8
PIM3	84	6
PKA	108	15
PKB alpha	104	5
PKB beta	106	18
PKC alpha	97	8
PKC gamma	101	5
PKC zeta	103	4
PKD1	82	9
PLK1	106	1
PRAK	85	8
PRK2	92	3
RIPK2	42	1
ROCK 2	71	2
RSK1	77	31
RSK2	80	4
S6K1	112	4
SGK1	105	9
SIK2	67	7
SIK3	64	12
SmMLCK	85	1
Src	72	10
SRPK1	104	4
STK33	91	12
SYK	72	5
TAK1	39	1
TAO1	95	20
TBK1	79	11
TESK1	98	10
TIE2	84	15
TLK1	98	8
TrkA	82	11
TSSK1	101	7
TTBK1	79	8
TTK	77	3
ULK1	63	13
ULK2	69	7
VEGFR1	32	2
WNK1	117	8
YES1	58	4
ZAP70	123	1