Inhibitor | BX-320  

Screen Conc: 10.00µM

Kinase	% Activity Remaining Sort descending	Standard Deviation
IKK epsilon	3	8
Aurora B	4	0
TBK1	5	0
Aurora C	6	0
MARK3	7	0
PDK1	7	0
MELK	11	0
FGF-R1	13	1
AMPK	13	2
ERK8	18	1
CAMKK beta	19	1
GSK3 beta	22	0
BRSK2	22	3
PAK4	26	0
MKK1	29	1
MNK2	31	1
CHK1	33	0
CDK2-Cyclin A	35	0
RSK1	39	6
Src	40	2
PAK5	40	7
Lck	41	2
RSK2	41	6
PRK2	42	0
DYRK3	44	1
CHK2	45	0
p38 beta MAPK	45	4
SGK1	45	2
PKD1	46	10
CAMKK alpha	47	4
CAMK1	52	5
PIM3	53	4
ROCK 2	56	5
PKB alpha	57	1
PKA	58	3
PAK6	60	0
S6K1	61	5
NEK2a	61	4
SYK	62	3
YES1	62	8
PIM1	63	3
DYRK1A	64	8
JNK2	65	7
IRR	65	7
CSK	66	10
PRAK	66	9
PKC alpha	67	0
MAPKAP-K2	68	1
IKK beta	69	2
PLK1	69	1
SRPK1	69	2
DYRK2	70	0
MST2	70	5
PIM2	71	2
ERK1	72	3
ERK2	73	9
EPH-A2	73	8
p38 delta MAPK	74	9
MNK1	74	4
HIPK2	74	2
PHK	76	3
MSK1	76	8
MAPKAP-K3	76	5
JNK1	78	3
PKC zeta	79	8
p38 gamma MAPK	79	0
PKB beta	79	0
EF2K	83	4
NEK7	84	11
NEK6	91	1
SmMLCK	94	4
p38 alpha MAPK	95	7
CK2	95	6
CK1 delta	96	6
MST4	100	2
HIPK3	100	5
JNK3	102	3

Screen Conc: 1.00µM

Kinase	% Activity Remaining Sort descending	Standard Deviation
Aurora B	6	2
Aurora C	8	0
TBK1	31	1
PDK1	33	0
MARK3	35	3
IKK epsilon	37	4
FGF-R1	44	3
AMPK	46	3
GSK3 beta	55	1
MELK	56	10
ERK8	57	10
MKK1	60	6
CAMKK beta	62	9
MNK2	71	5
CAMK1	71	4
CHK1	71	4
PRK2	71	1
p38 beta MAPK	72	7
BRSK2	72	3
SGK1	75	5
Lck	76	4
ROCK 2	77	4
PAK4	78	7
SRPK1	79	8
EPH-A2	81	5
ERK1	81	8
PKC zeta	82	5
PRAK	82	14
PKB alpha	82	14
Src	84	0
ERK2	84	0
PKD1	85	15
p38 gamma MAPK	86	3
PIM1	86	1
DYRK1A	86	3
DYRK3	86	9
PAK6	88	2
MNK1	88	13
IRR	88	1
RSK2	88	2
RSK1	89	3
CAMKK alpha	89	13
CK1 delta	89	6
CDK2-Cyclin A	90	6
MSK1	91	0
DYRK2	92	0
PAK5	93	1
p38 delta MAPK	93	2
CSK	93	14
NEK2a	94	3
JNK2	95	4
IKK beta	95	9
PLK1	96	7
HIPK2	96	8
JNK3	97	5
PIM3	97	2
MST2	97	3
PKC alpha	98	1
CHK2	99	2
PKA	99	1
YES1	100	2
S6K1	100	7
HIPK3	101	6
PHK	101	1
MAPKAP-K2	102	7
MST4	102	3
SmMLCK	103	4
PIM2	104	9
PKB beta	104	0
CK2	105	10
MAPKAP-K3	106	4
JNK1	106	8
p38 alpha MAPK	107	6
SYK	109	11
EF2K	110	7
NEK7	116	14
NEK6	117	14