Inhibitor | BMS345541 (IKK Inhibitor III)  

Compound name Brutto MW CAS PubChem CID Action Reference Reference
BMS345541 (IKK Inhibitor III)   C14H17N5 255.32 547757-23-3 9926054 IKBKB Du Z. (2012) J Interferon Cytokine Res. 368-77

Screening Results Chart

Screening Results Tables

Screen Conc: 1.00µM
Kinase % Activity Remaining Standard Deviation
AMPK 97 4
Aurora A 117 6
Aurora B 107 35
BRSK1 102 8
BRSK2 103 6
BTK 105 17
CAMK1 85 26
CAMKK beta 105 1
CDK2-Cyclin A 97 9
CHK1 129 19
CHK2 121 7
CK1 delta 104 19
CK2 116 8
CLK2 102 12
CSK 135 1
DAPK1 109 8
DYRK1A 108 2
DYRK2 89 8
DYRK3 107 1
EF2K 117 12
EPH-A2 98 11
EPH-A4 103 7
EPH-B2 126 9
EPH-B3 97 5
EPH-B4 111 9
ERK1 121 7
ERK2 116 23
ERK8 93 5
FGF-R1 103 12
GCK 110 3
GSK3 beta 102 19
HER4 145 13
HIPK1 101 9
HIPK2 98 3
HIPK3 106 4
IGF-1R 81 3
IKK beta 57 2
IKK epsilon 119 13
IR 109 1
IRAK4 127 19
IRR 94 3
JAK2 111 12
JNK1 111 19
JNK2 116 2
JNK3 104 20
Lck 109 9
LKB1 99 6
MAPKAP-K2 111 3
MAPKAP-K3 129 15
MARK1 109 2
MARK2 118 6
MARK3 97 11
MARK4 107 3
MEKK1 101 2
MELK 103 5
MINK1 117 25
MKK1 113 10
MLK1 104 34
MLK3 123 16
MNK1 97 22
MNK2 119 3
MSK1 93 7
MST2 86 8
MST4 94 1
NEK2a 117 3
NEK6 105 0
NUAK1 97 5
p38 alpha MAPK 113 16
p38 beta MAPK 100 4
p38 delta MAPK 101 2
p38 gamma MAPK 114 9
PAK2 113 9
PAK4 139 28
PAK5 139 14
PAK6 103 11
PDK1 107 2
PHK 109 3
PIM1 105 1
PIM2 113 1
PIM3 87 4
PKA 112 6
PKB alpha 92 0
PKB beta 117 14
PKC alpha 96 13
PKC zeta 124 2
PKD1 110 7
PLK1 111 9
PRAK 93 8
PRK2 116 8
RIPK2 102 4
ROCK 2 110 2
RSK1 97 3
RSK2 109 5
S6K1 105 1
SGK1 102 17
SmMLCK 110 7
Src 135 27
SRPK1 111 3
SYK 97 1
TAK1 105 10
TBK1 111 2
TrkA 169 18
TTK 102 8
VEGFR1 94 4
YES1 115 7
Screen Conc: 10.00µM
Kinase % Activity Remaining Standard Deviation
AMPK 91 1
Aurora A 108 3
Aurora B 64 7
BRSK1 89 21
BRSK2 84 4
BTK 98 15
CAMK1 73 8
CAMKK beta 99 1
CDK2-Cyclin A 60 4
CHK1 86 3
CHK2 88 2
CK1 delta 55 5
CK2 79 1
CLK2 74 3
CSK 93 6
DAPK1 118 45
DYRK1A 77 3
DYRK2 46 0
DYRK3 71 2
EF2K 99 3
EPH-A2 65 0
EPH-A4 83 1
EPH-B2 92 12
EPH-B3 61 1
EPH-B4 132 13
ERK1 87 6
ERK2 97 2
ERK8 18 2
FGF-R1 73 18
GCK 87 5
GSK3 beta 82 7
HER4 105 9
HIPK1 96 14
HIPK2 67 1
HIPK3 96 9
IGF-1R 93 2
IKK beta 16 6
IKK epsilon 101 8
IR 109 1
IRAK4 97 7
IRR 76 3
JAK2 87 2
JNK1 101 0
JNK2 83 2
JNK3 81 3
Lck 79 4
LKB1 71 8
MAPKAP-K2 100 3
MAPKAP-K3 94 3
MARK1 110 3
MARK2 103 5
MARK3 109 11
MARK4 103 10
MEKK1 92 3
MELK 94 13
MINK1 93 7
MKK1 96 3
MLK1 89 6
MLK3 91 2
MNK1 88 3
MNK2 100 6
MSK1 82 2
MST2 92 7
MST4 89 5
NEK2a 90 7
NEK6 86 7
NUAK1 45 5
p38 alpha MAPK 101 3
p38 beta MAPK 101 2
p38 delta MAPK 91 3
p38 gamma MAPK 102 3
PAK2 110 1
PAK4 106 7
PAK5 97 7
PAK6 96 7
PDK1 98 6
PHK 88 4
PIM1 95 2
PIM2 83 5
PIM3 70 3
PKA 94 4
PKB alpha 88 5
PKB beta 103 1
PKC alpha 90 4
PKC zeta 102 8
PKD1 54 5
PLK1 116 2
PRAK 111 7
PRK2 100 3
RIPK2 113 19
ROCK 2 80 5
RSK1 101 2
RSK2 81 8
S6K1 83 3
SGK1 91 4
SmMLCK 77 2
Src 90 7
SRPK1 104 4
SYK 96 1
TAK1 101 13
TBK1 89 9
TrkA 99 8
TTK 85 4
VEGFR1 69 2
YES1 84 12