Inhibitor | Blebbistatin  

Compound name Brutto MW CAS PubChem CID Action Reference Reference
Blebbistatin   C18H16N2O2 292.30 674289-55-5 3476986 myosin II Shu S. (2005) Proc. Natl. Acad. Sci. USA 102 1472 Kovacs M. (2004) J. Biol. Chem. 279 35557

Screening Results Chart

Screening Results Tables

Screen Conc: 100.00µM
Kinase % Activity Remaining Sort descending Standard Deviation
AMPK 60 2
SGK1 60 3
PRAK 64 1
GSK3 beta 66 2
CSK 67 9
PKA 70 0
S6K1 71 4
p38 beta MAPK 71 7
Lck 72 1
PDK1 74 3
PKC alpha 75 7
MSK1 75 7
ROCK 2 76 0
RSK1 77 5
JNK1 78 5
p38 alpha MAPK 80 1
p38 gamma MAPK 80 0
MAPKAP-K2 80 4
ERK2 82 3
NEK2a 82 6
NEK6 85 2
PHK 86 2
PKB alpha 88 3
DYRK1A 90 3
CK1 delta 91 3
CDK2-Cyclin A 92 7
CHK1 96 7
MKK1 99 6
CK2 101 5
p38 delta MAPK 116 4
Screen Conc: 10.00µM
Kinase % Activity Remaining Sort descending Standard Deviation
CSK 69 7
MINK1 72 9
RSK2 72 3
MLK3 73 7
PAK5 73 7
SmMLCK 74 15
PKB beta 74 6
CAMK1 74 4
DYRK2 76 10
RSK1 76 1
NEK2a 77 2
ROCK 2 77 4
Src 80 6
p38 delta MAPK 81 1
LKB1 81 1
MKK2 81 13
TAO1 82 5
MAPKAP-K2 82 4
PRAK 82 3
BTK 82 9
p38 beta MAPK 82 1
MSK1 83 0
PIM3 83 7
EF2K 83 5
PAK6 83 6
VEGFR1 85 2
IKK epsilon 85 6
IRAK4 86 6
MAPKAP-K3 86 1
HER4 87 8
TTK 87 3
CLK2 87 5
PAK2 87 5
PIM1 87 6
SRPK1 88 1
GSK3 beta 88 0
HIPK1 88 5
IGF-1R 88 2
IRR 88 7
Aurora B 88 2
JNK2 88 6
ERK8 89 5
MKK1 89 6
RIPK2 90 7
PAK4 90 8
CAMKK beta 90 3
CHK1 90 5
MARK3 91 4
ERK2 91 9
ASK1 91 3
AMPK 92 8
S6K1 92 3
JNK1 92 2
PDK1 93 3
MARK2 93 1
DAPK1 93 1
PIM2 93 3
MKK6 94 0
MARK4 94 5
TBK1 94 6
IR 95 15
PKB alpha 95 1
PRK2 95 0
MARK1 96 2
MELK 96 3
IKK beta 96 4
YES1 96 2
TAK1 96 3
DYRK1A 97 4
GCK 97 8
MNK1 97 2
EPH-B1 97 11
NUAK1 97 3
PKD1 97 11
HIPK2 98 0
BRSK2 98 4
p38 gamma MAPK 99 2
EPH-B4 99 2
DYRK3 99 9
PLK1 99 8
Aurora A 99 3
CK1 delta 99 4
JNK3 99 2
MST4 99 1
CHK2 100 12
MEKK1 100 8
JAK2 101 13
MLK1 101 8
SGK1 101 0
PKA 101 6
p38 alpha MAPK 101 2
ERK1 102 1
HIPK3 103 5
TrkA 103 3
PKC alpha 103 4
MNK2 104 3
MST2 104 1
SYK 105 12
BRSK1 106 5
Lck 106 6
NEK6 107 4
EPH-B3 107 4
EPH-A4 108 13
PKC zeta 108 5
EPH-A2 109 8
CK2 110 5
PHK 114 0
CDK2-Cyclin A 116 1
EPH-B2 116 3
FGF-R1 118 14