

Compound name | Brutto | MW | CAS | PubChem CID | Action | Reference | Reference |
---|---|---|---|---|---|---|---|
Blebbistatin | C18H16N2O2 | 292.30 | 674289-55-5 | 3476986 | myosin II | Shu S. (2005) Proc. Natl. Acad. Sci. USA 102 1472 | Kovacs M. (2004) J. Biol. Chem. 279 35557 |
Kinase | % Activity Remaining | Standard Deviation |
---|---|---|
AMPK | 92 | 8 |
ASK1 | 91 | 3 |
Aurora A | 99 | 3 |
Aurora B | 88 | 2 |
BRSK1 | 106 | 5 |
BRSK2 | 98 | 4 |
BTK | 82 | 9 |
CAMK1 | 74 | 4 |
CAMKK beta | 90 | 3 |
CDK2-Cyclin A | 116 | 1 |
CHK1 | 90 | 5 |
CHK2 | 100 | 12 |
CK1 delta | 99 | 4 |
CK2 | 110 | 5 |
CLK2 | 87 | 5 |
CSK | 69 | 7 |
DAPK1 | 93 | 1 |
DYRK1A | 97 | 4 |
DYRK2 | 76 | 10 |
DYRK3 | 99 | 9 |
EF2K | 83 | 5 |
EPH-A2 | 109 | 8 |
EPH-A4 | 108 | 13 |
EPH-B1 | 97 | 11 |
EPH-B2 | 116 | 3 |
EPH-B3 | 107 | 4 |
EPH-B4 | 99 | 2 |
ERK1 | 102 | 1 |
ERK2 | 91 | 9 |
ERK8 | 89 | 5 |
FGF-R1 | 118 | 14 |
GCK | 97 | 8 |
GSK3 beta | 88 | 0 |
HER4 | 87 | 8 |
HIPK1 | 88 | 5 |
HIPK2 | 98 | 0 |
HIPK3 | 103 | 5 |
IGF-1R | 88 | 2 |
IKK beta | 96 | 4 |
IKK epsilon | 85 | 6 |
IR | 95 | 15 |
IRAK4 | 86 | 6 |
IRR | 88 | 7 |
JAK2 | 101 | 13 |
JNK1 | 92 | 2 |
JNK2 | 88 | 6 |
JNK3 | 99 | 2 |
Lck | 106 | 6 |
LKB1 | 81 | 1 |
MAPKAP-K2 | 82 | 4 |
MAPKAP-K3 | 86 | 1 |
MARK1 | 96 | 2 |
MARK2 | 93 | 1 |
MARK3 | 91 | 4 |
MARK4 | 94 | 5 |
MEKK1 | 100 | 8 |
MELK | 96 | 3 |
MINK1 | 72 | 9 |
MKK1 | 89 | 6 |
MKK2 | 81 | 13 |
MKK6 | 94 | 0 |
MLK1 | 101 | 8 |
MLK3 | 73 | 7 |
MNK1 | 97 | 2 |
MNK2 | 104 | 3 |
MSK1 | 83 | 0 |
MST2 | 104 | 1 |
MST4 | 99 | 1 |
NEK2a | 77 | 2 |
NEK6 | 107 | 4 |
NUAK1 | 97 | 3 |
p38 alpha MAPK | 101 | 2 |
p38 beta MAPK | 82 | 1 |
p38 delta MAPK | 81 | 1 |
p38 gamma MAPK | 99 | 2 |
PAK2 | 87 | 5 |
PAK4 | 90 | 8 |
PAK5 | 73 | 7 |
PAK6 | 83 | 6 |
PDK1 | 93 | 3 |
PHK | 114 | 0 |
PIM1 | 87 | 6 |
PIM2 | 93 | 3 |
PIM3 | 83 | 7 |
PKA | 101 | 6 |
PKB alpha | 95 | 1 |
PKB beta | 74 | 6 |
PKC alpha | 103 | 4 |
PKC zeta | 108 | 5 |
PKD1 | 97 | 11 |
PLK1 | 99 | 8 |
PRAK | 82 | 3 |
PRK2 | 95 | 0 |
RIPK2 | 90 | 7 |
ROCK 2 | 77 | 4 |
RSK1 | 76 | 1 |
RSK2 | 72 | 3 |
S6K1 | 92 | 3 |
SGK1 | 101 | 0 |
SmMLCK | 74 | 15 |
Src | 80 | 6 |
SRPK1 | 88 | 1 |
SYK | 105 | 12 |
TAK1 | 96 | 3 |
TAO1 | 82 | 5 |
TBK1 | 94 | 6 |
TrkA | 103 | 3 |
TTK | 87 | 3 |
VEGFR1 | 85 | 2 |
YES1 | 96 | 2 |
Kinase | % Activity Remaining | Standard Deviation |
---|---|---|
AMPK | 60 | 2 |
CDK2-Cyclin A | 92 | 7 |
CHK1 | 96 | 7 |
CK1 delta | 91 | 3 |
CK2 | 101 | 5 |
CSK | 67 | 9 |
DYRK1A | 90 | 3 |
ERK2 | 82 | 3 |
GSK3 beta | 66 | 2 |
JNK1 | 78 | 5 |
Lck | 72 | 1 |
MAPKAP-K2 | 80 | 4 |
MKK1 | 99 | 6 |
MSK1 | 75 | 7 |
NEK2a | 82 | 6 |
NEK6 | 85 | 2 |
p38 alpha MAPK | 80 | 1 |
p38 beta MAPK | 71 | 7 |
p38 delta MAPK | 116 | 4 |
p38 gamma MAPK | 80 | 0 |
PDK1 | 74 | 3 |
PHK | 86 | 2 |
PKA | 70 | 0 |
PKB alpha | 88 | 3 |
PKC alpha | 75 | 7 |
PRAK | 64 | 1 |
ROCK 2 | 76 | 0 |
RSK1 | 77 | 5 |
S6K1 | 71 | 4 |
SGK1 | 60 | 3 |