Inhibitor | Blebbistatin  

Compound name Brutto MW CAS PubChem CID Action Reference Reference
Blebbistatin   C18H16N2O2 292.30 674289-55-5 3476986 myosin II Shu S. (2005) Proc. Natl. Acad. Sci. USA 102 1472 Kovacs M. (2004) J. Biol. Chem. 279 35557

Screening Results Chart

Screening Results Tables

Screen Conc: 10.00µM
Kinase % Activity Remaining Standard Deviation
AMPK 92 8
ASK1 91 3
Aurora A 99 3
Aurora B 88 2
BRSK1 106 5
BRSK2 98 4
BTK 82 9
CAMK1 74 4
CAMKK beta 90 3
CDK2-Cyclin A 116 1
CHK1 90 5
CHK2 100 12
CK1 delta 99 4
CK2 110 5
CLK2 87 5
CSK 69 7
DAPK1 93 1
DYRK1A 97 4
DYRK2 76 10
DYRK3 99 9
EF2K 83 5
EPH-A2 109 8
EPH-A4 108 13
EPH-B1 97 11
EPH-B2 116 3
EPH-B3 107 4
EPH-B4 99 2
ERK1 102 1
ERK2 91 9
ERK8 89 5
FGF-R1 118 14
GCK 97 8
GSK3 beta 88 0
HER4 87 8
HIPK1 88 5
HIPK2 98 0
HIPK3 103 5
IGF-1R 88 2
IKK beta 96 4
IKK epsilon 85 6
IR 95 15
IRAK4 86 6
IRR 88 7
JAK2 101 13
JNK1 92 2
JNK2 88 6
JNK3 99 2
Lck 106 6
LKB1 81 1
MAPKAP-K2 82 4
MAPKAP-K3 86 1
MARK1 96 2
MARK2 93 1
MARK3 91 4
MARK4 94 5
MEKK1 100 8
MELK 96 3
MINK1 72 9
MKK1 89 6
MKK2 81 13
MKK6 94 0
MLK1 101 8
MLK3 73 7
MNK1 97 2
MNK2 104 3
MSK1 83 0
MST2 104 1
MST4 99 1
NEK2a 77 2
NEK6 107 4
NUAK1 97 3
p38 alpha MAPK 101 2
p38 beta MAPK 82 1
p38 delta MAPK 81 1
p38 gamma MAPK 99 2
PAK2 87 5
PAK4 90 8
PAK5 73 7
PAK6 83 6
PDK1 93 3
PHK 114 0
PIM1 87 6
PIM2 93 3
PIM3 83 7
PKA 101 6
PKB alpha 95 1
PKB beta 74 6
PKC alpha 103 4
PKC zeta 108 5
PKD1 97 11
PLK1 99 8
PRAK 82 3
PRK2 95 0
RIPK2 90 7
ROCK 2 77 4
RSK1 76 1
RSK2 72 3
S6K1 92 3
SGK1 101 0
SmMLCK 74 15
Src 80 6
SRPK1 88 1
SYK 105 12
TAK1 96 3
TAO1 82 5
TBK1 94 6
TrkA 103 3
TTK 87 3
VEGFR1 85 2
YES1 96 2
Screen Conc: 100.00µM
Kinase % Activity Remaining Standard Deviation
AMPK 60 2
CDK2-Cyclin A 92 7
CHK1 96 7
CK1 delta 91 3
CK2 101 5
CSK 67 9
DYRK1A 90 3
ERK2 82 3
GSK3 beta 66 2
JNK1 78 5
Lck 72 1
MAPKAP-K2 80 4
MKK1 99 6
MSK1 75 7
NEK2a 82 6
NEK6 85 2
p38 alpha MAPK 80 1
p38 beta MAPK 71 7
p38 delta MAPK 116 4
p38 gamma MAPK 80 0
PDK1 74 3
PHK 86 2
PKA 70 0
PKB alpha 88 3
PKC alpha 75 7
PRAK 64 1
ROCK 2 76 0
RSK1 77 5
S6K1 71 4
SGK1 60 3