| Compound name | Brutto | MW | CAS | PubChem CID | Action | Reference | Reference |
|---|---|---|---|---|---|---|---|
| Blebbistatin | C18H16N2O2 | 292.30 | 674289-55-5 | 3476986 | myosin II | Shu S. (2005) Proc. Natl. Acad. Sci. USA 102 1472 | Kovacs M. (2004) J. Biol. Chem. 279 35557 |
| Kinase | % Activity Remaining | Standard Deviation |
|---|---|---|
| AMPK | 92 | 8 |
| ASK1 | 91 | 3 |
| Aurora A | 99 | 3 |
| Aurora B | 88 | 2 |
| BRSK1 | 106 | 5 |
| BRSK2 | 98 | 4 |
| BTK | 82 | 9 |
| CAMK1 | 74 | 4 |
| CAMKK beta | 90 | 3 |
| CDK2-Cyclin A | 116 | 1 |
| CHK1 | 90 | 5 |
| CHK2 | 100 | 12 |
| CK1 delta | 99 | 4 |
| CK2 | 110 | 5 |
| CLK2 | 87 | 5 |
| CSK | 69 | 7 |
| DAPK1 | 93 | 1 |
| DYRK1A | 97 | 4 |
| DYRK2 | 76 | 10 |
| DYRK3 | 99 | 9 |
| EF2K | 83 | 5 |
| EPH-A2 | 109 | 8 |
| EPH-A4 | 108 | 13 |
| EPH-B1 | 97 | 11 |
| EPH-B2 | 116 | 3 |
| EPH-B3 | 107 | 4 |
| EPH-B4 | 99 | 2 |
| ERK1 | 102 | 1 |
| ERK2 | 91 | 9 |
| ERK8 | 89 | 5 |
| FGF-R1 | 118 | 14 |
| GCK | 97 | 8 |
| GSK3 beta | 88 | 0 |
| HER4 | 87 | 8 |
| HIPK1 | 88 | 5 |
| HIPK2 | 98 | 0 |
| HIPK3 | 103 | 5 |
| IGF-1R | 88 | 2 |
| IKK beta | 96 | 4 |
| IKK epsilon | 85 | 6 |
| IR | 95 | 15 |
| IRAK4 | 86 | 6 |
| IRR | 88 | 7 |
| JAK2 | 101 | 13 |
| JNK1 | 92 | 2 |
| JNK2 | 88 | 6 |
| JNK3 | 99 | 2 |
| Lck | 106 | 6 |
| LKB1 | 81 | 1 |
| MAPKAP-K2 | 82 | 4 |
| MAPKAP-K3 | 86 | 1 |
| MARK1 | 96 | 2 |
| MARK2 | 93 | 1 |
| MARK3 | 91 | 4 |
| MARK4 | 94 | 5 |
| MEKK1 | 100 | 8 |
| MELK | 96 | 3 |
| MINK1 | 72 | 9 |
| MKK1 | 89 | 6 |
| MKK2 | 81 | 13 |
| MKK6 | 94 | 0 |
| MLK1 | 101 | 8 |
| MLK3 | 73 | 7 |
| MNK1 | 97 | 2 |
| MNK2 | 104 | 3 |
| MSK1 | 83 | 0 |
| MST2 | 104 | 1 |
| MST4 | 99 | 1 |
| NEK2a | 77 | 2 |
| NEK6 | 107 | 4 |
| NUAK1 | 97 | 3 |
| p38 alpha MAPK | 101 | 2 |
| p38 beta MAPK | 82 | 1 |
| p38 delta MAPK | 81 | 1 |
| p38 gamma MAPK | 99 | 2 |
| PAK2 | 87 | 5 |
| PAK4 | 90 | 8 |
| PAK5 | 73 | 7 |
| PAK6 | 83 | 6 |
| PDK1 | 93 | 3 |
| PHK | 114 | 0 |
| PIM1 | 87 | 6 |
| PIM2 | 93 | 3 |
| PIM3 | 83 | 7 |
| PKA | 101 | 6 |
| PKB alpha | 95 | 1 |
| PKB beta | 74 | 6 |
| PKC alpha | 103 | 4 |
| PKC zeta | 108 | 5 |
| PKD1 | 97 | 11 |
| PLK1 | 99 | 8 |
| PRAK | 82 | 3 |
| PRK2 | 95 | 0 |
| RIPK2 | 90 | 7 |
| ROCK 2 | 77 | 4 |
| RSK1 | 76 | 1 |
| RSK2 | 72 | 3 |
| S6K1 | 92 | 3 |
| SGK1 | 101 | 0 |
| SmMLCK | 74 | 15 |
| Src | 80 | 6 |
| SRPK1 | 88 | 1 |
| SYK | 105 | 12 |
| TAK1 | 96 | 3 |
| TAO1 | 82 | 5 |
| TBK1 | 94 | 6 |
| TrkA | 103 | 3 |
| TTK | 87 | 3 |
| VEGFR1 | 85 | 2 |
| YES1 | 96 | 2 |
| Kinase | % Activity Remaining | Standard Deviation |
|---|---|---|
| AMPK | 60 | 2 |
| CDK2-Cyclin A | 92 | 7 |
| CHK1 | 96 | 7 |
| CK1 delta | 91 | 3 |
| CK2 | 101 | 5 |
| CSK | 67 | 9 |
| DYRK1A | 90 | 3 |
| ERK2 | 82 | 3 |
| GSK3 beta | 66 | 2 |
| JNK1 | 78 | 5 |
| Lck | 72 | 1 |
| MAPKAP-K2 | 80 | 4 |
| MKK1 | 99 | 6 |
| MSK1 | 75 | 7 |
| NEK2a | 82 | 6 |
| NEK6 | 85 | 2 |
| p38 alpha MAPK | 80 | 1 |
| p38 beta MAPK | 71 | 7 |
| p38 delta MAPK | 116 | 4 |
| p38 gamma MAPK | 80 | 0 |
| PDK1 | 74 | 3 |
| PHK | 86 | 2 |
| PKA | 70 | 0 |
| PKB alpha | 88 | 3 |
| PKC alpha | 75 | 7 |
| PRAK | 64 | 1 |
| ROCK 2 | 76 | 0 |
| RSK1 | 77 | 5 |
| S6K1 | 71 | 4 |
| SGK1 | 60 | 3 |