| Compound name | Brutto | MW | CAS | PubChem CID | Action | Reference | Reference |
|---|---|---|---|---|---|---|---|
| Staurosporine | C28H26N4O3 | 466.54 | 62996-74-1 | 451705 | Broad spectrum | Boix J. (1997) Neuropharmacology 36 811-821 | Wiesner D.A. and Dawson G. (1996) J. Neurochem. 66 1418-1425 |
| Kinase | % Activity Remaining | Standard Deviation |
|---|---|---|
| ABL |
3
|
1 |
| AMPK | 22 | 3 |
| ASK1 |
8
|
0 |
| Aurora A |
1
|
0 |
| Aurora B | 41 | 3 |
| BRK |
7
|
4 |
| BRSK1 |
8
|
2 |
| BRSK2 |
2
|
1 |
| BTK | 16 | 1 |
| CAMK1 |
4
|
2 |
| CAMKK beta |
4
|
1 |
| CDK2-Cyclin A |
5
|
2 |
| CHK1 | 16 | 11 |
| CHK2 |
3
|
0 |
| CK1 delta | 63 | 11 |
| CK2 | 69 | 10 |
| CLK2 |
2
|
0 |
| CSK | 36 | 9 |
| DAPK1 |
7
|
0 |
| DYRK1A |
0
|
0 |
| DYRK2 | 13 | 4 |
| DYRK3 |
6
|
2 |
| EF2K | 112 | 2 |
| EIF2AK3 | 18 | 3 |
| EPH-A2 | 11 | 3 |
| EPH-A4 | 16 | 0 |
| EPH-B1 | 118 | 11 |
| EPH-B2 |
3
|
0 |
| EPH-B3 |
7
|
0 |
| EPH-B4 | 12 | 2 |
| ERK1 | 33 | 8 |
| ERK2 | 22 | 1 |
| ERK8 | 17 | 5 |
| FGF-R1 |
3
|
0 |
| GCK |
7
|
2 |
| GSK3 beta |
1
|
1 |
| HER4 |
10
|
2 |
| HIPK1 | 26 | 5 |
| HIPK2 |
5
|
3 |
| HIPK3 | 13 | 2 |
| IGF-1R |
1
|
0 |
| IKK beta | 11 | 1 |
| IKK epsilon | 14 | 7 |
| IR |
1
|
1 |
| IRAK1 |
2
|
0 |
| IRAK4 |
3
|
1 |
| IRR |
4
|
0 |
| JAK2 |
5
|
0 |
| JNK1 |
6
|
0 |
| JNK2 | 21 | 1 |
| JNK3 | 15 | 2 |
| Lck |
6
|
0 |
| LKB1 | 11 | 0 |
| MAPKAP-K2 |
1
|
0 |
| MAPKAP-K3 | 33 | 7 |
| MARK1 | 23 | 1 |
| MARK2 | 38 | 11 |
| MARK3 |
1
|
2 |
| MARK4 |
8
|
0 |
| MEKK1 | 33 | 8 |
| MELK | 20 | 1 |
| MINK1 | 19 | 0 |
| MKK1 | 15 | 15 |
| MKK2 |
8
|
3 |
| MKK6 | 37 | 0 |
| MLK1 | 24 | 9 |
| MLK3 | 14 | 4 |
| MNK1 | 38 | 5 |
| MNK2 | 39 | 0 |
| MPSK1 | 16 | 0 |
| MSK1 |
1
|
0 |
| MST2 | 30 | 9 |
| MST4 | 29 | 6 |
| NEK2a | 11 | 1 |
| NEK6 | 69 | 4 |
| NUAK1 |
4
|
1 |
| OSR1 |
2
|
1 |
| p38 alpha MAPK | 72 | 0 |
| p38 beta MAPK | 60 | 4 |
| p38 delta MAPK |
6
|
2 |
| p38 gamma MAPK | 13 | 6 |
| PAK2 |
1
|
0 |
| PAK4 |
8
|
7 |
| PAK5 |
3
|
1 |
| PAK6 |
0
|
0 |
| PDK1 | 18 | 7 |
| PHK | 26 | 6 |
| PIM1 |
8
|
2 |
| PIM2 |
3
|
1 |
| PIM3 |
7
|
11 |
| PKA |
2
|
0 |
| PKB alpha |
2
|
1 |
| PKB beta |
0
|
0 |
| PKC alpha |
4
|
1 |
| PKC gamma |
7
|
0 |
| PKC zeta |
3
|
1 |
| PKD1 |
5
|
0 |
| PLK1 | 28 | 1 |
| PRAK |
2
|
1 |
| PRK2 |
7
|
1 |
| RIPK2 | 21 | 2 |
| ROCK 2 | 24 | 9 |
| RSK1 |
3
|
1 |
| RSK2 |
-1
|
0 |
| S6K1 |
4
|
2 |
| SGK1 |
1
|
2 |
| SmMLCK |
9
|
3 |
| Src |
3
|
1 |
| SRPK1 |
2
|
0 |
| STK33 |
6
|
0 |
| SYK |
4
|
1 |
| TAK1 |
2
|
1 |
| TAO1 |
4
|
1 |
| TBK1 |
5
|
2 |
| TIE2 |
9
|
4 |
| TLK1 |
5
|
3 |
| TrkA |
1
|
0 |
| TTK | 23 | 6 |
| VEGFR1 |
2
|
0 |
| YES1 |
8
|
4 |
| ZAP70 |
6
|
0 |