Inhibitor | 1 NA-PP1 (PP1 Analog)  

Compound name Brutto MW CAS PubChem CID Action Reference Reference
1 NA-PP1 (PP1 Analog)   C19H19N5 317.40 221243-82-9 4877 Src Bishop A. C. (2000) Nature 407 395 https://pubmed.ncbi.nlm.nih.gov/[pmid2]

Screening Results Chart

Screening Results Tables

Screen Conc: 1.00µM
Kinase % Activity Remaining Standard Deviation
AMPK 81 6
Aurora B 90 7
Aurora C 88 6
BRSK2 108 4
CAMK1 83 3
CAMKK alpha 94 5
CAMKK beta 90 1
CDK2-Cyclin A 94 3
CHK1 97 8
CHK2 75 3
CK1 delta 30 0
CK2 88 0
CSK 31 1
DYRK1A 91 4
DYRK2 95 1
DYRK3 84 1
EF2K 97 1
ERK1 103 1
ERK2 82 4
ERK8 81 1
GSK3 beta 95 1
HIPK2 99 2
HIPK3 101 3
IKK beta 92 1
JNK1 92 4
JNK2 84 0
JNK3 93 3
Lck 30 0
MAPKAP-K2 116 0
MAPKAP-K3 90 1
MARK3 67 2
MELK 84 2
MKK1 86 5
MNK1 109 1
MNK2 105 0
MSK1 81 6
MST2 46 3
NEK2a 99 4
NEK6 98 8
NEK7 93 6
p38 alpha MAPK 49 1
p38 beta MAPK 77 1
p38 delta MAPK 108 1
p38 gamma MAPK 97 0
PAK4 82 2
PAK5 73 9
PAK6 94 5
PDK1 97 5
PHK 84 1
PIM1 104 5
PIM2 100 5
PIM3 98 3
PKA 86 2
PKB alpha 102 9
PKB beta 95 2
PKC alpha 77 4
PKC zeta 86 0
PKD1 35 2
PLK1 94 2
PRAK 88 7
PRK2 110 1
ROCK 2 86 1
RSK1 89 2
RSK2 95 1
S6K1 86 6
SGK1 101 5
SmMLCK 78 0
Src 20 6
SRPK1 94 7
Screen Conc: 10.00µM
Kinase % Activity Remaining Standard Deviation
AMPK 73 2
Aurora B 74 8
Aurora C 55 1
BRSK2 75 0
CAMK1 63 2
CAMKK alpha 76 8
CAMKK beta 72 6
CDK2-Cyclin A 55 1
CHK1 95 2
CHK2 32 1
CK1 delta
4
0
CK2 87 0
CSK
5
1
DYRK1A 77 8
DYRK2 96 7
DYRK3 65 1
EF2K 99 2
ERK1 69 1
ERK2 62 0
ERK8 58 4
GSK3 beta 77 0
HIPK2 84 1
HIPK3 105 0
IKK beta 95 3
JNK1 93 1
JNK2 56 4
JNK3 87 3
Lck
6
1
MAPKAP-K2 97 3
MAPKAP-K3 87 5
MARK3 30 0
MELK 27 0
MKK1 65 4
MNK1 95 1
MNK2 85 7
MSK1 46 6
MST2
10
3
NEK2a 95 4
NEK6 91 7
NEK7 106 0
p38 alpha MAPK 17 4
p38 beta MAPK 24 2
p38 delta MAPK 80 2
p38 gamma MAPK 81 2
PAK4 35 0
PAK5 25 3
PAK6 57 6
PDK1 97 3
PHK 75 1
PIM1 91 4
PIM2 104 0
PIM3 83 4
PKA 56 2
PKB alpha 50 0
PKB beta 89 1
PKC alpha 39 8
PKC zeta 83 1
PKD1
8
3
PLK1 95 5
PRAK 76 0
PRK2 89 2
ROCK 2 30 0
RSK1 53 4
RSK2 71 1
S6K1 61 7
SGK1 91 2
SmMLCK 61 4
Src
3
2
SRPK1 89 7