Inhibitor | (5Z)-7-Oxozeaenol  

Screen Conc: 0.10µM

Kinase Sort ascending	% Activity Remaining	Standard Deviation
ZAP70	110	4
YES1	105	40
VEGFR1	8	0
TTK	104	2
TrkA	46	0
TIE2	103	16
TBK1	105	1
TAO1	103	3
TAK1	5	1
SYK	88	3
STK33	120	13
SRPK1	104	10
Src	106	4
SmMLCK	108	4
SGK1	106	2
S6K1	112	8
RSK2	106	6
RSK1	113	1
ROCK 2	116	13
RIPK2	103	5
PRK2	102	2
PRAK	66	7
PLK1	103	1
PKD1	71	6
PKC zeta	105	1
PKC gamma	87	4
PKC alpha	107	3
PKB beta	86	9
PKB alpha	111	9
PKA	99	7
PIM3	126	6
PIM2	91	7
PIM1	102	1
PHK	100	2
PDK1	99	10
PAK6	100	5
PAK5	96	9
PAK4	94	11
PAK2	104	5
p38 gamma MAPK	99	1
p38 delta MAPK	99	2
p38 beta MAPK	90	9
p38 alpha MAPK	103	3
NUAK1	113	9
NEK6	122	5
NEK2a	108	0
MST4	129	6
MST2	120	14
MSK1	107	25
MPSK1	103	6
MNK2	41	3
MNK1	55	0
MLK3	114	16
MLK1	109	4
MKK6	12	4
MKK2	12	2
MKK1	13	2
MINK1	101	9
MELK	95	11
MEKK1	107	5
MARK4	107	1
MARK3	116	11
MARK2	109	1
MARK1	112	16
MAPKAP-K3	113	18
MAPKAP-K2	124	4
LKB1	138	6
Lck	78	1
JNK3	107	2
JNK2	109	12
JNK1	90	0
JAK2	108	11
IRR	107	52
IRAK4	99	4
IR	110	10
IKK epsilon	120	4
IKK beta	102	17
IGF-1R	100	16
HIPK3	90	2
HIPK2	98	9
HIPK1	102	11
HER4	100	2
GSK3 beta	102	13
GCK	121	3
FGF-R1	105	24
ERK8	40	2
ERK2	103	2
ERK1	106	15
EPH-B4	87	6
EPH-B3	111	8
EPH-B2	96	21
EPH-B1	99	11
EPH-A4	91	4
EPH-A2	99	8
EF2K	48	57
DYRK3	94	7
DYRK2	114	5
DYRK1A	117	0
DAPK1	108	1
CSK	118	16
CLK2	96	17
CK2	106	15
CK1 delta	102	4
CHK2	110	1
CHK1	114	13
CDK2-Cyclin A	119	7
CAMKK beta	87	4
CAMK1	88	2
BTK	90	5
BRSK2	84	11
BRSK1	113	12
BRK	65	13
Aurora B	94	1
Aurora A	106	20
ASK1	91	1
AMPK	100	7
ABL	108	5

Screen Conc: 1.00µM

Kinase Sort ascending	% Activity Remaining	Standard Deviation
ZAP70	96	6
YES1	60	2
VEGFR1	13	6
TTK	91	8
TrkA	24	11
TIE2	93	9
TBK1	102	13
TAO1	66	5
TAK1	3	1
SYK	77	5
STK33	85	2
SRPK1	88	5
Src	43	3
SmMLCK	80	5
SGK1	95	1
S6K1	82	4
RSK2	70	13
RSK1	90	2
ROCK 2	83	6
RIPK2	39	2
PRK2	91	15
PRAK	14	11
PLK1	100	6
PKD1	31	11
PKC zeta	99	12
PKC gamma	87	10
PKC alpha	85	3
PKB beta	84	10
PKB alpha	91	1
PKA	93	1
PIM3	80	3
PIM2	106	4
PIM1	72	9
PHK	89	5
PDK1	76	3
PAK6	87	1
PAK5	103	6
PAK4	81	6
PAK2	110	8
p38 gamma MAPK	92	6
p38 delta MAPK	114	14
p38 beta MAPK	72	0
p38 alpha MAPK	85	4
NUAK1	78	3
NEK6	93	5
NEK2a	89	1
MST4	72	9
MST2	89	4
MSK1	100	1
MPSK1	101	10
MNK2	26	1
MNK1	13	5
MLK3	79	18
MLK1	75	1
MKK6	10	2
MKK2	3	2
MKK1	2	1
MINK1	83	1
MELK	94	4
MEKK1	92	2
MARK4	86	4
MARK3	77	14
MARK2	114	3
MARK1	99	0
MAPKAP-K3	94	5
MAPKAP-K2	79	4
LKB1	65	1
Lck	30	4
JNK3	90	11
JNK2	81	4
JNK1	52	14
JAK2	75	0
IRR	96	14
IRAK4	28	2
IR	94	7
IKK epsilon	92	10
IKK beta	95	6
IGF-1R	93	8
HIPK3	103	10
HIPK2	82	4
HIPK1	98	9
HER4	95	1
GSK3 beta	74	5
GCK	80	0
FGF-R1	87	7
ERK8	4	4
ERK2	65	7
ERK1	64	0
EPH-B4	90	5
EPH-B3	100	4
EPH-B2	75	5
EPH-B1	81	8
EPH-A4	46	8
EPH-A2	55	2
EF2K	85	3
DYRK3	101	2
DYRK2	89	5
DYRK1A	97	1
DAPK1	94	2
CSK	56	7
CLK2	90	2
CK2	77	1
CK1 delta	104	6
CHK2	87	1
CHK1	92	3
CDK2-Cyclin A	88	3
CAMKK beta	57	2
CAMK1	105	11
BTK	93	0
BRSK2	88	11
BRSK1	90	4
BRK	25	0
Aurora B	74	6
Aurora A	105	2
ASK1	95	6
AMPK	92	5
ABL	71	6